Authors:
EDWARDS PD
ANDISIK DW
BRYANT CA
EWING B
GOMES B
LEWIS JJ
RAKIEWICZ D
STEELMAN G
STRIMPLER A
TRAINOR DA
TUTHILL PA
MAUGER RC
VEALE CA
WILDONGER RA
WILLIAMS JC
WOLANIN DJ
ZOTTOLA M
Citation: Pd. Edwards et al., DISCOVERY AND BIOLOGICAL-ACTIVITY OR ORALLY-ACTIVE PEPTIDYL TRIFLUOROMETHYL KETONE INHIBITORS OF HUMAN NEUTROPHIL ELASTASE, Journal of medicinal chemistry, 40(12), 1997, pp. 1876-1885
Authors:
EDWARDS PD
ANDISIK DW
STRIMPLER AM
GOMES B
TUTHILL PA
Citation: Pd. Edwards et al., NONPEPTIDIC INHIBITORS OF HUMAN NEUTROPHIL ELASTASE .7. DESIGN, SYNTHESIS, AND IN-VITRO ACTIVITY OF A SERIES OF PYRIDOPYRIMIDINE TRIFLUOROMETHYL KETONES, Journal of medicinal chemistry, 39(5), 1996, pp. 1112-1124
Authors:
EDWARDS PD
WOLANIN DJ
ANDISIK DW
DAVIS MW
Citation: Pd. Edwards et al., PEPTIDYL ALPHA-KETOHETEROCYCLIC INHIBITORS OF HUMAN NEUTROPHIL ELASTASE .2. EFFECT OF VARYING THE HETEROCYCLIC RING ON IN-VITRO POTENCY, Journal of medicinal chemistry, 38(1), 1995, pp. 76-85
Authors:
BROWN FJ
ANDISIK DW
BERNSTEIN PR
BRYANT CB
CECCARELLI C
DAMEWOOD JR
WOOLSON SA
EDWARDS PD
EARLEY RA
FEENEY S
GREEN RC
GOMES B
KOSMIDER BJ
KRELL RD
SHAW A
STEELMAN GB
THOMAS RN
VACEK EP
VEALE CA
TUTHILL PA
WARNER P
WILLIAMS JC
WOLANIN DJ
Citation: Fj. Brown et al., DESIGN OF ORALLY-ACTIVE, NONPEPTIDIC INHIBITORS OF HUMAN-LEUKOCYTE ELASTASE, Journal of medicinal chemistry, 37(9), 1994, pp. 1259-1261