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Results: 1-7 |
Results: 7
-5-ALPHA-ANDROST-1-ENE-17-BETA-N-ARYL-CARBOXAMIDES - AN APPROACH TO COMBINED ANDROGEN BLOCKADE [5-ALPHA-REDUCTASE INHIBITION WITH ANDROGEN RECEPTOR-BINDING IN-VITRO]
Authors: TOLMAN RL SAHOO SP BAKSHI RK GRATALE D PATEL G PATEL S TONEY J CHANG B HARRIS GS
Citation: Rl. Tolman et al., -5-ALPHA-ANDROST-1-ENE-17-BETA-N-ARYL-CARBOXAMIDES - AN APPROACH TO COMBINED ANDROGEN BLOCKADE [5-ALPHA-REDUCTASE INHIBITION WITH ANDROGEN RECEPTOR-BINDING IN-VITRO], Journal of steroid biochemistry and molecular biology, 60(5-6), 1997, pp. 303-309
MK386 - A POTENT, SELECTIVE INHIBITOR OF THE HUMAN TYPE-1 5-ALPHA-REDUCTASE
Authors: ELLSWORTH K AZZOLINA B BAGINSKY W BULL H CHANG B CIMIS G MITRA S TONEY J BAKSHI RK RASMUSSON GR TOLMAN RL HARRIS GS
Citation: K. Ellsworth et al., MK386 - A POTENT, SELECTIVE INHIBITOR OF THE HUMAN TYPE-1 5-ALPHA-REDUCTASE, Journal of steroid biochemistry and molecular biology, 58(4), 1996, pp. 377-384
O-5-ALPHA-ANDROST-1-ENE-17-BETA-N-ARYLCARBOXAMIDES AS DUAL INHIBITORSOF HUMAN TYPE-1 AND TYPE-2 STEROID 5-ALPHA-REDUCTASES - DRAMATIC EFFECT OF N-ARYL SUBSTITUENTS ON TYPE-1 AND TYPE-2 5-ALPHA-REDUCTASE INHIBITORY POTENCY (VOL 38, PG 3190, 1995)
Authors: BAKSHI RK RASMUSSON GH PATEL GF MOSLEY RT CHANG B ELLSWORTH K HARRIS GS TOLMAN RL
Citation: Rk. Bakshi et al., O-5-ALPHA-ANDROST-1-ENE-17-BETA-N-ARYLCARBOXAMIDES AS DUAL INHIBITORSOF HUMAN TYPE-1 AND TYPE-2 STEROID 5-ALPHA-REDUCTASES - DRAMATIC EFFECT OF N-ARYL SUBSTITUENTS ON TYPE-1 AND TYPE-2 5-ALPHA-REDUCTASE INHIBITORY POTENCY (VOL 38, PG 3190, 1995), Journal of medicinal chemistry, 39(5), 1996, pp. 1192-1192
MECHANISM-BASED INHIBITION OF HUMAN STEROID 5-ALPHA-REDUCTASE BY FINASTERIDE - ENZYME-CATALYZED FORMATION OF NADP-DIHYDROFINASTERIDE, A POTENT BISUBSTRATE ANALOG INHIBITOR
Authors: BULL HG GARCIACALVO M ANDERSSON S BAGINSKY WF CHAN HK ELLSWORTH DE MILLER RR STEARNS RA BAKSHI RK RASMUSSON GH TOLMAN RL MYERS RW KOZARICH JW HARRIS GS
Citation: Hg. Bull et al., MECHANISM-BASED INHIBITION OF HUMAN STEROID 5-ALPHA-REDUCTASE BY FINASTERIDE - ENZYME-CATALYZED FORMATION OF NADP-DIHYDROFINASTERIDE, A POTENT BISUBSTRATE ANALOG INHIBITOR, Journal of the American Chemical Society, 118(10), 1996, pp. 2359-2365
4-AZASTEROIDS AS 5-ALPHA-REDUCTASE INHIBITORS - IDENTIFICATION OF 4,7-BETA-DIMETHYL-4-AZA-5-ALPHA-CHOLESTAN-3-ONE (MK-386) AS A SCALP ISOZYME-SELECTIVE INHIBITOR
Authors: TOLMAN RL ASTER S BAKSHI RK BERGMAN JP BULL HG CHANG B CIMIS G DOLENGA MP DURETTE P ELLSWORTH K ESSER C GRAHAM DW HAGMANN WK HARRIS G KOPKA I LANZA T PATEL G POLO S RASMUSSON GH SAHOO S TONEY JH VONLANGEN D WITZEL B
Citation: Rl. Tolman et al., 4-AZASTEROIDS AS 5-ALPHA-REDUCTASE INHIBITORS - IDENTIFICATION OF 4,7-BETA-DIMETHYL-4-AZA-5-ALPHA-CHOLESTAN-3-ONE (MK-386) AS A SCALP ISOZYME-SELECTIVE INHIBITOR, European journal of medicinal chemistry, 30, 1995, pp. 311-316
-5-ALPHA-ANDROST-1-ENE-17-BETA-N-ARYL-CARBOXAMIDES AS DUAL INHIBITORSOF HUMAN TYPE-1 AND TYPE-2 STEROID 5-ALPHA-REDUCTASES - DRAMATIC EFFECT OF N-ARYL SUBSTITUENTS ON TYPE-1 AND TYPE-2 5-ALPHA-REDUCTASE INHIBITORY POTENCY
Authors: BAKSHI RK RASMUSSON GH PATEL GF MOSLEY RT CHANG B ELLSWORTH K HARRIS GS TOLMAN RL
Citation: Rk. Bakshi et al., -5-ALPHA-ANDROST-1-ENE-17-BETA-N-ARYL-CARBOXAMIDES AS DUAL INHIBITORSOF HUMAN TYPE-1 AND TYPE-2 STEROID 5-ALPHA-REDUCTASES - DRAMATIC EFFECT OF N-ARYL SUBSTITUENTS ON TYPE-1 AND TYPE-2 5-ALPHA-REDUCTASE INHIBITORY POTENCY, Journal of medicinal chemistry, 38(17), 1995, pp. 3189-3192
4,7-BETA-DIMETHYL-4-AZACHOLESTAN-3-ONE (MK-386) AND RELATED 4-AZASTEROIDS AS SELECTIVE INHIBITORS OF HUMAN TYPE-1 5-ALPHA-REDUCTASE
Authors: BAKSHI RK PATEL GF RASMUSSON GH BAGINSKY WF CIMIS G ELLSWORTH K CHANG B BULL H TOLMAN RL HARRIS GS
Citation: Rk. Bakshi et al., 4,7-BETA-DIMETHYL-4-AZACHOLESTAN-3-ONE (MK-386) AND RELATED 4-AZASTEROIDS AS SELECTIVE INHIBITORS OF HUMAN TYPE-1 5-ALPHA-REDUCTASE, Journal of medicinal chemistry, 37(23), 1994, pp. 3871-3874
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