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Results: 1-13 |
Results: 13
29-METHYLIDENE-2,3-OXIDOSQUALENE DERIVATIVES AS STEREOSPECIFIC MECHANISM-BASED INHIBITORS OF LIVER AND YEAST OXIDOSQUALENE CYCLASE
Authors: CERUTI M ROCCO F VIOLA F BALLIANO G MILLA P ARPICCO S CATTEL L
Citation: M. Ceruti et al., 29-METHYLIDENE-2,3-OXIDOSQUALENE DERIVATIVES AS STEREOSPECIFIC MECHANISM-BASED INHIBITORS OF LIVER AND YEAST OXIDOSQUALENE CYCLASE, Journal of medicinal chemistry, 41(4), 1998, pp. 540-554
HUMAN ALPHA-THROMBIN INHIBITION BY THE HIGHLY SELECTIVE COMPOUNDS ARBONYL-D-PHE-PRO-ALPHA-ARALYS-P-NITROPHENYL-ESTER AND -CARBOBENZOXY-PRO-ALPHA-AZALYS-P-NITROPHENYL-ESTER - A KINETIC, THERMODYNAMIC AND X-RAY CRYSTALLOGRAPHIC STUDY
Authors: DESIMONE G BALLIANO G MILLA P GALLINA C GIORDANO C TARRICONE C RIZZI M BOLOGNESI M ASCENZI P
Citation: G. Desimone et al., HUMAN ALPHA-THROMBIN INHIBITION BY THE HIGHLY SELECTIVE COMPOUNDS ARBONYL-D-PHE-PRO-ALPHA-ARALYS-P-NITROPHENYL-ESTER AND -CARBOBENZOXY-PRO-ALPHA-AZALYS-P-NITROPHENYL-ESTER - A KINETIC, THERMODYNAMIC AND X-RAY CRYSTALLOGRAPHIC STUDY, Journal of Molecular Biology, 269(4), 1997, pp. 558-569
HUMAN ALPHA-THROMBIN INHIBITION BY THE ACTIVE-SITE TITRANT N-ALPHA-(N,N-DIMETHYLCARBAMOYL)-ALPHA-AZALYSINE P-NITROPHENYL ESTER - A COMPARATIVE KINETIC AND X-RAY CRYSTALLOGRAPHIC STUDY (VOL 258, PG 851, 1996)
Authors: NARDINI M PEACE A RIZZI M CASALE E FERRACCIOLI R BALLIANO G MILLA P ASCENZI P BOLOGNESI M
Citation: M. Nardini et al., HUMAN ALPHA-THROMBIN INHIBITION BY THE ACTIVE-SITE TITRANT N-ALPHA-(N,N-DIMETHYLCARBAMOYL)-ALPHA-AZALYSINE P-NITROPHENYL ESTER - A COMPARATIVE KINETIC AND X-RAY CRYSTALLOGRAPHIC STUDY (VOL 258, PG 851, 1996), Journal of Molecular Biology, 263(1), 1996, pp. 99-99
HUMAN ALPHA-THROMBIN INHIBITION BY THE ACTIVE-SITE TITRANT N-ALPHA-(N,N-DIMETHYLCARBAMOYL)-ALPHA-AZALYSINE P-NITROPHENYL ESTER - A COMPARATIVE KINETIC AND X-RAY CRYSTALLOGRAPHIC STUDY
Authors: NARDINI M PESCE A RIZZI M CASALE E FERRACCIOLI R BALLIANO G MILLA P ASCENZI P BOLOGNESI M
Citation: M. Nardini et al., HUMAN ALPHA-THROMBIN INHIBITION BY THE ACTIVE-SITE TITRANT N-ALPHA-(N,N-DIMETHYLCARBAMOYL)-ALPHA-AZALYSINE P-NITROPHENYL ESTER - A COMPARATIVE KINETIC AND X-RAY CRYSTALLOGRAPHIC STUDY, Journal of Molecular Biology, 258(5), 1996, pp. 851-859
XYCARBONYL-D-PHENYLALANYL-L-PROLYL-ALPHA-AZALYSINE P-NITROPHENYL ESTER - A NOVEL, HIGH SELECTIVE AND OPTIMAL CHROMOGENIC ACTIVE-SITE TITRANT FOR HUMAN AND BOVINE ALPHA-THROMBIN, BETA-THROMBIN AND GAMMA-THROMBIN
Authors: BALLIANO G MILLA P GIORDANO C GALLINA C COLETTA M MENEGATTI E RIZZI M BOLOGNESI M ASCENZI P
Citation: G. Balliano et al., XYCARBONYL-D-PHENYLALANYL-L-PROLYL-ALPHA-AZALYSINE P-NITROPHENYL ESTER - A NOVEL, HIGH SELECTIVE AND OPTIMAL CHROMOGENIC ACTIVE-SITE TITRANT FOR HUMAN AND BOVINE ALPHA-THROMBIN, BETA-THROMBIN AND GAMMA-THROMBIN, Biochemical and biophysical research communications, 225(2), 1996, pp. 557-561
INHIBITION OF BOVINE BETA-TRYPSIN, HUMAN ALPHA-THROMBIN AND PORCINE PANCREATIC BETA-KALLIKREIN-B BY 4',6-DIAMIDINO-2-PHENYLINDOLE, 6-AMIDINOINDOLE AND BENZAMIDINE - A COMPARATIVE THERMODYNAMIC AND X-RAY STRUCTURAL STUDY
Authors: CASALE E COLLYER C ASCENZI P BALLIANO G MILLA P VIOLA F FASANO M MENEGATTI E BOLOGNESI M
Citation: E. Casale et al., INHIBITION OF BOVINE BETA-TRYPSIN, HUMAN ALPHA-THROMBIN AND PORCINE PANCREATIC BETA-KALLIKREIN-B BY 4',6-DIAMIDINO-2-PHENYLINDOLE, 6-AMIDINOINDOLE AND BENZAMIDINE - A COMPARATIVE THERMODYNAMIC AND X-RAY STRUCTURAL STUDY, Biophysical chemistry, 54(1), 1995, pp. 75-81
2,3-OXIDOSQUALENE CYCLASE - FROM AZASQUALENES TO NEW SITE-DIRECTED INHIBITORS
Authors: CATTEL L CERUTI M BALLIANO G VIOLA F GROSA G ROCCO F BRUSA P
Citation: L. Cattel et al., 2,3-OXIDOSQUALENE CYCLASE - FROM AZASQUALENES TO NEW SITE-DIRECTED INHIBITORS, Lipids, 30(3), 1995, pp. 235-246
ACTIVE-SITE TITRATION OF BOVINE BETA-TRYPSIN BY N-ALPHA-(N,N-DIMETHYLCARBAMOYL)-ALPHA-AZA-LYSINE P-NITROPHENYL ESTER - KINETIC AND CRYSTALLOGRAPHIC ANALYSIS
Authors: SARTORI P CARUGO KD FERRACCIOLI R BALLIANO G MILLA P ASCENZI P BOLOGNESI M
Citation: P. Sartori et al., ACTIVE-SITE TITRATION OF BOVINE BETA-TRYPSIN BY N-ALPHA-(N,N-DIMETHYLCARBAMOYL)-ALPHA-AZA-LYSINE P-NITROPHENYL ESTER - KINETIC AND CRYSTALLOGRAPHIC ANALYSIS, FEBS letters, 358(1), 1995, pp. 53-56
INHIBITION OF 2,3-OXIDOSQUALENE CYCLASE AND STEROL BIOSYNTHESIS BY 10-AZASQUALENE AND 19-AZASQUALENE DERIVATIVES
Authors: VIOLA F BRUSA P BALLIANO G CERUTI M BOUTAUD O SCHUBER F CATTEL L
Citation: F. Viola et al., INHIBITION OF 2,3-OXIDOSQUALENE CYCLASE AND STEROL BIOSYNTHESIS BY 10-AZASQUALENE AND 19-AZASQUALENE DERIVATIVES, Biochemical pharmacology, 50(6), 1995, pp. 787-796
INHIBITION OF BOVINE BETA-TRYPSIN BY THE ACTIVE-SITE TITRANT (N)UNDER-BAR-DIMETHYLCARBAMOYL)-ALPHA-AZAORNITHINE (P)UNDER-BAR-NITROPHENYL ESTER - A KINETIC AND X-RAY CRYSTALLOGRAPHIC STUDY
Authors: ASCENZI P BALLIANO G MILLA P FERRACCIOLI R SARTORI P DJINOVICCARUGO K BOLOGNESI M
Citation: P. Ascenzi et al., INHIBITION OF BOVINE BETA-TRYPSIN BY THE ACTIVE-SITE TITRANT (N)UNDER-BAR-DIMETHYLCARBAMOYL)-ALPHA-AZAORNITHINE (P)UNDER-BAR-NITROPHENYL ESTER - A KINETIC AND X-RAY CRYSTALLOGRAPHIC STUDY, Biochemical and biophysical research communications, 217(2), 1995, pp. 437-444
INHIBITION OF STEROL BIOSYNTHESIS IN SACCHAROMYCES-CEREVISIAE AND CANDIDA-ALBICANS BY 22,23-EPOXY-2-AZA-2,3-DIHYDROSQUALENE AND THE CORRESPONDING N-OXIDE
Authors: BALLIANO G MILLA P CERUTI M CARRANO L VIOLA F BRUSA P CATTEL L
Citation: G. Balliano et al., INHIBITION OF STEROL BIOSYNTHESIS IN SACCHAROMYCES-CEREVISIAE AND CANDIDA-ALBICANS BY 22,23-EPOXY-2-AZA-2,3-DIHYDROSQUALENE AND THE CORRESPONDING N-OXIDE, Antimicrobial agents and chemotherapy, 38(9), 1994, pp. 1904-1908
SYNTHESIS AND BIOLOGICAL-ACTIVITY OF 19-AZASQUALENE 2,3-EPOXIDE AS INHIBITOR OF 2,3-OXIDOSQUALENE CYCLASE
Authors: CERUTI M ROCCO F VIOLA F BALLIANO G GROSA G DOSIO F CATTEL L
Citation: M. Ceruti et al., SYNTHESIS AND BIOLOGICAL-ACTIVITY OF 19-AZASQUALENE 2,3-EPOXIDE AS INHIBITOR OF 2,3-OXIDOSQUALENE CYCLASE, European journal of medicinal chemistry, 28(9), 1993, pp. 675-682
ARBOXY-4-NITROPHENYL-DITHIO-1,1',2-TRISNORSQUALENE - A SITE-DIRECTED INACTIVATOR OF YEAST OXIDOSQUALENE CYCLASE
Authors: BALLIANO G GROSA G MILLA P VIOLA F CATTEL L
Citation: G. Balliano et al., ARBOXY-4-NITROPHENYL-DITHIO-1,1',2-TRISNORSQUALENE - A SITE-DIRECTED INACTIVATOR OF YEAST OXIDOSQUALENE CYCLASE, Lipids, 28(10), 1993, pp. 903-906
Risultati: 1-13 |