Authors:
MOSS ML
JIN SLC
BECHERER JD
BICKETT DM
BURKHART W
CHEN WJ
HASSLER D
LEESNITZER MT
MCGEEHAN G
MILLA M
MOYER M
ROCQUE W
SEATON T
SCHOENEN F
WARNER J
WILLARD D
Citation: Ml. Moss et al., STRUCTURAL FEATURES AND BIOCHEMICAL-PROPERTIES OF TNF-ALPHA CONVERTING-ENZYME (TACE), Journal of neuroimmunology, 72(2), 1997, pp. 127-129
Authors:
MOSS ML
JIN SLC
MILLA ME
BICKETT DM
BURKHART W
CARTER HL
CHEN WJ
CLAY WC
DIDSBURY JR
HASSLER D
HOFFMAN CR
KOST TA
LAMBERT MH
LEESNITZER MA
MCCAULEY P
MCGEEHAN G
MITCHELL J
OVERTON LK
SCHOENEN F
SEATON T
SU JL
WARNER J
WILLARD D
BECHERER JD
Citation: Ml. Moss et al., CLONING OF A DISINTEGRIN METALLOPROTEINASE THAT PROCESSES PRECURSOR TUMOR-NECROSIS-FACTOR-ALPHA (VOL 385, PG 733, 1997), Nature, 386(6626), 1997, pp. 738-738
Authors:
FOLEY MA
HASSMAN AS
DREWRY DH
GREER DG
WAGNER CD
FELDMAN PL
BERMAN J
BICKETT DM
MCGEEHAN GM
LAMBERT MH
GREEN M
Citation: Ma. Foley et al., RAPID SYNTHESIS OF NOVEL DIPEPTIDE INHIBITORS OF HUMAN COLLAGENASE AND GELATINASE USING SOLID-PHASE CHEMISTRY, Bioorganic & medicinal chemistry letters, 6(16), 1996, pp. 1905-1910
Authors:
CONWAY JG
TREXLER SJ
WAKEFIELD JA
MARRON BE
EMERSON DL
BICKETT DM
DEATON DN
GARRISON D
ELDER M
MCELROY A
WILLMOTT N
DOCKERTY AJP
MCGEEHAN GM
Citation: Jg. Conway et al., EFFECT OF MATRIX METALLOPROTEINASE INHIBITORS ON TUMOR-GROWTH AND SPONTANEOUS METASTASIS, Clinical & experimental metastasis, 14(2), 1996, pp. 115-124
Authors:
FRYE SV
HAFFNER CD
MALONEY PR
HINER RN
DORSEY GF
NOE RA
UNWALLA RJ
BATCHELOR KW
BRAMSON HN
STUART JD
SCHWEIKER SL
VANAMOLD J
BICKETT DM
MOSS ML
TIAN GC
LEE FW
TIPPIN TK
JAMES MK
GRIZZLE MK
LONG JE
CROOM DK
Citation: Sv. Frye et al., STRUCTURE-ACTIVITY-RELATIONSHIPS FOR INHIBITION OF TYPE-1 AND 2 HUMAN5-ALPHA-REDUCTASE AND HUMAN ADRENAL 3-BETA-HYDROXY-DELTA(5)-STEROID DEHYDROGENASE 3-KETO-DELTA(5)-STEROID ISOMERASE BY 6-AZAANDROST-4-EN-3-ONES - OPTIMIZATION OF THE C17 SUBSTITUENT/, Journal of medicinal chemistry, 38(14), 1995, pp. 2621-2627
Authors:
BROWN FK
BROWN PJ
BICKETT DM
CHAMBERS CL
DAVIES HG
DEATON DN
DREWRY D
FOLEY M
MCELROY AB
GREGSON M
MCGEEHAN GM
MYERS PL
NORTON D
SALOVICH JM
SCHOENEN FJ
WARD P
Citation: Fk. Brown et al., MATRIX METALLOPROTEINASE INHIBITORS CONTAINING A (CARBOXYALKYL)AMINO ZINC LIGAND - MODIFICATION OF THE P1 AND P2' RESIDUES, Journal of medicinal chemistry, 37(5), 1994, pp. 674-688
Authors:
FRYE SV
HAFFNER CD
MALONEY PR
MOOK RA
DORSEY GF
HINER RN
CRIBBS CM
WHEELER TN
RAY JA
ANDREWS RC
BATCHELOR KW
BRAMSON HN
STUART JD
SCHWEIKER SL
VANARNOLD J
CROOM S
BICKETT DM
MOSS ML
TIAN GC
UNWALLA RJ
LEE FW
TIPPIN TK
JAMES MK
GRIZZLE MK
LONG JE
SCHUSTER SV
Citation: Sv. Frye et al., 6-AZASTEROIDS - STRUCTURE-ACTIVITY-RELATIONSHIPS FOR INHIBITION OF TYPE-1 AND TYPE-2 HUMAN 5-ALPHA-REDUCTASE AND HUMAN ADRENAL 3-BETA-HYDROXY-DELTA(5)-STEROID DEHYDROGENASE 3-KETO-DELTA(5)-STEROID ISOMERASE, Journal of medicinal chemistry, 37(15), 1994, pp. 2352-2360
Authors:
BROWN FK
BROWN PJ
BICKETT DM
CHAMBERS CL
DAVIES HG
DEATON DN
DREWRY D
FOLEY M
MCELROY AB
GREGSON M
MCGEEHAN GM
MYERS PL
NORTON D
SALOVICH JM
SCHOENEN FJ
WARD P
Citation: Fk. Brown et al., MATRIX METALLOPROTEINASE INHIBITORS CONTAINING A (CARBOXYALKYL)AMINO ZINC LIGAND - MODIFICATION OF THE P1 AND P2' RESIDUES (VOL 37, PG 674,1994), Journal of medicinal chemistry, 37(10), 1994, pp. 1546-1546
Authors:
MCGEEHAN GM
BICKETT DM
GREEN M
KASSEL D
WISEMAN JS
BERMAN J
Citation: Gm. Mcgeehan et al., CHARACTERIZATION OF THE PEPTIDE SUBSTRATE SPECIFICITIES OF INTERSTITIAL COLLAGENASE AND 92-KDA GELATINASE - IMPLICATIONS FOR SUBSTRATE OPTIMIZATION, The Journal of biological chemistry, 269(52), 1994, pp. 32814-32820
Authors:
WISEMAN J
GREEN M
BERMAN J
ANDEREGG R
KASSEL D
MILLINGTON DS
NORWOOD D
MCGEEHAN J
BICKETT DM
Citation: J. Wiseman et al., RAPID OPTIMIZATION OF ENZYME SUBSTRATES FOR MATRIX METALLOPROTEASES USING DEFINED SUBSTRATE MIXTURES, Journal of cellular biochemistry, 1993, pp. 118-118
Authors:
FRYE SV
HAFFNER CD
MALONEY PR
MOOK RA
HINER RN
BATCHELOR KW
BRAMSON HN
STUART JD
SCHWEIKER SL
VANARNOLD J
BICKETT DM
MOSS ML
TIAN GC
UNWALLA RJ
LEE FW
TIPPIN TK
JAMES MK
GRIZZLE MK
LONG JE
SCHUSTER SV
DORSEY GF
Citation: Sv. Frye et al., 6-AZASTEROIDS - POTENT DUAL INHIBITORS OF HUMAN TYPE-1 AND 2 STEROID 5-ALPHA-REDUCTASE, Journal of medicinal chemistry, 36(26), 1993, pp. 4313-4315
Authors:
BICKETT DM
GREEN MD
BERMAN J
DEZUBE M
HOWE AS
BROWN PJ
ROTH JT
MCGEEHAN GM
Citation: Dm. Bickett et al., A HIGH-THROUGHPUT FLUOROGENIC SUBSTRATE FOR INTERSTITIAL COLLAGENASE (MMP-1) AND GELATINASE (MMP-9), Analytical biochemistry, 212(1), 1993, pp. 58-64