Authors:
LEGRAVEREND M
LUDWIG O
BISAGNI E
LECLERC S
MEIJER L
Citation: M. Legraverend et al., SYNTHESIS OF C2 ALKYNYLATED PURINES, A NEW FAMILY OF POTENT INHIBITORS OF CYCLIN-DEPENDENT KINASES, Bioorganic & medicinal chemistry letters, 8(7), 1998, pp. 793-798
Authors:
KUKRETI S
SUN JS
LOAKES D
BROWN DM
NGUYEN CH
BISAGNI E
GARESTIER T
HELENE C
Citation: S. Kukreti et al., TRIPLE HELICES FORMED AT OLIGOPYRIMIDINE-CENTER-DOT-OLIGOPURINE SEQUENCES WITH BASE-PAIR INVERSIONS - EFFECT OF A TRIPLEX-SPECIFIC LIGAND ON STABILITY AND SELECTIVITY, Nucleic acids research, 26(9), 1998, pp. 2179-2183
Authors:
COSTACHE E
NGUYEN CH
LEONCE S
PIERRE A
ATASSI G
BISAGNI E
Citation: E. Costache et al., 1-AMINO-SUBSTITUTED 8-HYDROXY-4,5-DIMETHY-5H-PYRIDO[4,3-B]INDOLES WITH PROPYL-SUBSTITUENTS OR METHYL-SUBSTITUENTS AT THE 9-POSITIONS, AND 7,9-POSITIONS - SYNTHESIS AND BIOLOGICAL EVALUATION, Anti-cancer drug design, 13(4), 1998, pp. 361-372
Authors:
COSTACHE E
NGUYEN CH
GUILBAUD N
LEONCE S
PIERRE A
ATASSI G
BISAGNI E
Citation: E. Costache et al., SYNTHESIS, PROPERTIES AND BIOLOGICAL EVALUATION OF SUBSTITUTED FURO[3,2-E] AND PYRANO[3,2-E]PYRIDO[4,3-B]INDOLES, Anti-cancer drug design, 13(4), 1998, pp. 373-386
Authors:
ESCUDE C
NGUYEN CH
KUKRETI S
JANIN Y
SUN JS
BISAGNI E
GARESTIER T
HELENE C
Citation: C. Escude et al., RATIONAL DESIGN OF A TRIPLE HELIX-SPECIFIC INTERCALATING LIGAND, Proceedings of the National Academy of Sciences of the United Statesof America, 95(7), 1998, pp. 3591-3596
Authors:
NGUYEN CH
MARCHAND C
DELAGE S
SUN JS
GARESTIER T
HELENE C
BISAGNI E
Citation: Ch. Nguyen et al., SYNTHESIS OF 13H-BENZO[6,7]INDOLO[3,2-C]QUINOLINES AND 13H-BENZO[4,5]INDOLO[3,2-C]QUINOLINES - A NEW SERIES OF POTENT SPECIFIC LIGANDS FOR TRIPLEX DNA, Journal of the American Chemical Society, 120(11), 1998, pp. 2501-2507
Authors:
ROUTIER S
BERNIER JL
CATTEAU JP
COLSON P
HOUSSIER C
RIVALLE C
BISAGNI E
BAILLY C
Citation: S. Routier et al., SYNTHESIS, DNA-BINDING, AND CLEAVING PROPERTIES OF AN ELLIPTICINE-SALEN-CENTER-DOT-COPPER CONJUGATE, Bioconjugate chemistry, 8(6), 1997, pp. 789-792
Authors:
SILVER GC
NGUYEN CH
BOUTORINE AS
BISAGNI E
GARESTIER T
HELENE C
Citation: Gc. Silver et al., CONJUGATES OF OLIGONUCLEOTIDES WITH TRIPLEX-SPECIFIC INTERCALATING AGENTS - STABILIZATION OF TRIPLE-HELICAL DNA IN THE PROMOTER REGION OF THE GENE FOR THE ALPHA-SUBUNIT OF INTERLEUKIN-2 (IL-2R-ALPHA), Bioconjugate chemistry, 8(1), 1997, pp. 15-22
Authors:
RENAULT E
FONTAINEAUPART MP
TFIBEL F
GARDESALBERT M
BISAGNI E
Citation: E. Renault et al., SPECTROSCOPIC STUDY OF THE INTERACTION OF PAZELLIPTINE WITH NUCLEIC-ACIDS, Journal of photochemistry and photobiology.B, Biology, 40(3), 1997, pp. 218-227
Authors:
CROISYDELCEY M
CROISY A
MOUSSET S
LETOURNEUR M
BISAGNI E
JACQUEMINSABLON A
PIERRE J
Citation: M. Croisydelcey et al., GENISTEIN ANALOGS - EFFECTS ON EPIDERMAL GROWTH-FACTOR RECEPTOR TYROSINE KINASE AND ON STRESS-ACTIVATED PATHWAYS, Biomedicine & pharmacotherapy, 51(6-7), 1997, pp. 286-294
Citation: M. Croisy et al., SYNTHESIS OF 4-METHOXYPHENYL)-5,7-DIMETHOXY(1H)-QUINOLIN-2-ONES OR 4-METHOXYPHENYL)-5,7-DIMETHOXY(1H)-QUINOLIN-4-ONES AND DERIVATIVES, Heterocycles, 45(4), 1997, pp. 683-690
Citation: C. Rivalle et E. Bisagni, ETHYL(4-N-ACYLAMINOPYRIDIN-3-YL)GLYOXYLATE AND 5-AZAISATIN AS NEW SYNTHONS FOR A ROUTE TO VARIOUS NEW POLYHETEROCYCLES, Journal of heterocyclic chemistry, 34(2), 1997, pp. 441-444
Authors:
KIM SK
SUN JS
GARESTIER T
HELENE C
NGUYEN CH
BISAGNI E
RODGER A
NORDEN B
Citation: Sk. Kim et al., BINDING GEOMETRIES OF TRIPLE-HELIX SELECTIVE BENZOPYRIDO[4,3-B]INDOLELIGANDS COMPLEXED WITH DOUBLE-HELICAL AND TRIPLE-HELICAL POLYNUCLEOTIDES, Biopolymers, 42(1), 1997, pp. 101-111
Authors:
SILVER GC
SUN JS
NGUYEN CH
BOUTORINE AS
BISAGNI E
HELENE C
Citation: Gc. Silver et al., STABLE TRIPLE-HELICAL DNA COMPLEXES FORMED BY BENZOPYRIDOINDOLE-OLIGONUCLEOTIDE AND BENZOPYRIDOQUINOXALINE-OLIGONUCLEOTIDE CONJUGATES, Journal of the American Chemical Society, 119(2), 1997, pp. 263-268
Authors:
RENAULT E
FONTAINEAUPART MP
GARDESALBERT M
RIVALLE C
BISAGNI E
Citation: E. Renault et al., RADICAL CHEMISTRY OF THE ANTITUMOR DRUG PAZELLIPTINE (PZE) IN AQUEOUS-SOLUTION OR INTERCALATED IN POLY(DA)-POLY(DT), Journal de chimie physique et de physico-chimie biologique, 93(1), 1996, pp. 194-202
Citation: C. Jolivet et al., SYNTHESIS AND BEHAVIOR OF FURO[2,3,4-K,L]ACRIDINES AND FURO[2,3,4-K,L]PYRANO[3,2-H]ACRIDINES, Heterocycles, 43(3), 1996, pp. 641-651
Authors:
GUILBAUD N
KRAUSBERTHIER L
SAINTDIZIER D
ROUILLON MH
JAN M
BURBRIDGE M
VISALLI M
BISAGNI E
PIERRE A
ATASSI G
Citation: N. Guilbaud et al., IN-VIVO ANTITUMOR-ACTIVITY OF S-16020-2, A NEW OLIVACINE DERIVATIVE, Cancer chemotherapy and pharmacology, 38(6), 1996, pp. 513-521
Authors:
DEBIZEMONT T
DUVALVALENTIN G
SUN JS
BISAGNI E
GARESTIER T
HELENE C
Citation: T. Debizemont et al., ALTERNATE STRAND RECOGNITION OF DOUBLE-HELICAL DNA BY (T,G)-CONTAINING OLIGONUCLEOTIDES IN THE PRESENCE OF A TRIPLE HELIX-SPECIFIC LIGAND, Nucleic acids research, 24(6), 1996, pp. 1136-1143
Authors:
FONTAINEAUPART MP
LAGUITTONPASQUIER H
PANSU R
BRIAN L
RENAULT E
MARDEN MC
RIVALLE C
BISAGNI E
Citation: Mp. Fontaineaupart et al., PROTON AND CHARGE-TRANSFER IN THE INTERCALATING ANTITUMOR DRUG PAZELLIPTINE, Perkin transactions. 2, (8), 1996, pp. 1767-1774
Authors:
JANIN YL
AUBERTIN AM
CHIARONI A
RICHE C
MONNERET C
BISAGNI E
GRIERSON DS
Citation: Yl. Janin et al., IMIDAZO[1,5-G][1,4]DIAZEPINES, TIBO ANALOGS LACKING THE PHENYL RING -SYNTHESIS AND EVALUATION AS ANTI-HIV AGENTS, Tetrahedron, 52(48), 1996, pp. 15157-15170