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Results: 1-9 |
Results: 9
SYNTHESIS AND TYROSINE KINASE INHIBITORY ACTIVITY OF A SERIES OF 2-AMINO-8H-PYRIDO[2,3-D]PYRIMIDINES - IDENTIFICATION OF POTENT, SELECTIVE PLATELET-DERIVED GROWTH-FACTOR RECEPTOR TYROSINE KINASE INHIBITORS
Authors: BOSCHELLI DH WU ZP KLUTCHKO SR SHOWALTER HDH HAMBY JM LU GH MAJOR TC DAHRING TK BATLEY B PANEK RL KEISER J HARTL BG KRAKER AJ KLOHS WD ROBERTS BJ PATMORE S ELLIOTT WL STEINKAMPF R BRADFORD LA HALLAK H DOHERTY AM
Citation: Dh. Boschelli et al., SYNTHESIS AND TYROSINE KINASE INHIBITORY ACTIVITY OF A SERIES OF 2-AMINO-8H-PYRIDO[2,3-D]PYRIMIDINES - IDENTIFICATION OF POTENT, SELECTIVE PLATELET-DERIVED GROWTH-FACTOR RECEPTOR TYROSINE KINASE INHIBITORS, Journal of medicinal chemistry, 41(22), 1998, pp. 4365-4377
2-SUBSTITUTED AMINOPYRIDO[2,3-D]PYRIMIDIN-7(8H) ONES - STRUCTURE-ACTIVITY-RELATIONSHIPS AGAINST SELECTED TYROSINE KINASES AND IN-VITRO AND IN-VIVO ANTICANCER ACTIVITY
Authors: KLUTCHKO SR HAMBY JM BOSCHELLI DH WU ZP KRAKER AJ AMAR AM HARTL BG SHEN C KLOHS WD STEINKAMPF RW DRISCOLL DL NELSON JM ELLIOTT WL ROBERTS BJ STONER CL VINCENT PW DYKES DJ PANEK RL LU GH MAJOR TC DAHRING TK HALLAK H BRADFORD LA SHOWALTER HDH DOHERTY AM
Citation: Sr. Klutchko et al., 2-SUBSTITUTED AMINOPYRIDO[2,3-D]PYRIMIDIN-7(8H) ONES - STRUCTURE-ACTIVITY-RELATIONSHIPS AGAINST SELECTED TYROSINE KINASES AND IN-VITRO AND IN-VIVO ANTICANCER ACTIVITY, Journal of medicinal chemistry, 41(17), 1998, pp. 3276-3292
PREPARATION OF BENZOTHIENO[2,3-F]-1,4-OXAZEPIN-5(2H)-ONES AND BENZOTHIENO[2,3-F]-1,4-THIAZEPIN-5(2H)-ONES AND OF BENZOTHIENO[3,2-E]-1,4-DIAZEPIN-5-ONES
Authors: KHATANA SS BOSCHELLI DH KRAMER JB CONNOR DT BARTH H STOSS P
Citation: Ss. Khatana et al., PREPARATION OF BENZOTHIENO[2,3-F]-1,4-OXAZEPIN-5(2H)-ONES AND BENZOTHIENO[2,3-F]-1,4-THIAZEPIN-5(2H)-ONES AND OF BENZOTHIENO[3,2-E]-1,4-DIAZEPIN-5-ONES, Journal of organic chemistry, 61(17), 1996, pp. 6060-6062
INHIBITION OF E-SELECTIN-MEDIATED, ICAM-1-MEDIATED, AND VCAM-1-MEDIATED CELL-ADHESION BY BENZO[B]THIOPHENE-CARBOXAMIDES, BENZOFURAN-CARBOXAMIDES, INDOLE-, AND NAPHTHALENE-2-CARBOXAMIDES - IDENTIFICATION OF PD-144795 AS AN ANTIINFLAMMATORY AGENT
Authors: BOSCHELLI DH KRAMER JB KHATANA SS SORENSON RJ CONNOR DT FERIN MA WRIGHT CD LESCH ME IMRE K OKONKWO GC SCHRIER DJ CONROY MC FERGUSON E WOELLE J SAXENA U
Citation: Dh. Boschelli et al., INHIBITION OF E-SELECTIN-MEDIATED, ICAM-1-MEDIATED, AND VCAM-1-MEDIATED CELL-ADHESION BY BENZO[B]THIOPHENE-CARBOXAMIDES, BENZOFURAN-CARBOXAMIDES, INDOLE-, AND NAPHTHALENE-2-CARBOXAMIDES - IDENTIFICATION OF PD-144795 AS AN ANTIINFLAMMATORY AGENT, Journal of medicinal chemistry, 38(22), 1995, pp. 4597-4614
INHIBITION OF TUMOR-NECROSIS-FACTOR INDUCED HUMAN AORTIC ENDOTHELIAL-CELL ADHESION MOLECULE GENE-EXPRESSION BY AN ALKOXYBENZO[B]THIOPHENE-2-CARBOXAMIDE
Authors: WOLLE J FERGUSON E KESHAVA C DEVALL LJ BOSCHELLI DH NEWTON RS SAXENA U
Citation: J. Wolle et al., INHIBITION OF TUMOR-NECROSIS-FACTOR INDUCED HUMAN AORTIC ENDOTHELIAL-CELL ADHESION MOLECULE GENE-EXPRESSION BY AN ALKOXYBENZO[B]THIOPHENE-2-CARBOXAMIDE, Biochemical and biophysical research communications, 214(1), 1995, pp. 6-10
3-ALKOXYBENZO[B]THIOPHENE-2-CARBOXAMIDES AS INHIBITORS OF NEUTROPHIL-ENDOTHELIAL CELL-ADHESION
Authors: BOSCHELLI DH KRAMER JB CONNOR DT LESCH ME SCHRIER DJ FERIN MA WRIGHT CD
Citation: Dh. Boschelli et al., 3-ALKOXYBENZO[B]THIOPHENE-2-CARBOXAMIDES AS INHIBITORS OF NEUTROPHIL-ENDOTHELIAL CELL-ADHESION, Journal of medicinal chemistry, 37(6), 1994, pp. 717-718
SYNTHESIS OF 2,6-DI-TERT-BUTYLPHENOLS LINKED TO 1,3,4-OXADIAZOLES AND1,3,4-THIADIAZOLES
Authors: KRAMER JB BOSCHELLI DH CONNOR DT
Citation: Jb. Kramer et al., SYNTHESIS OF 2,6-DI-TERT-BUTYLPHENOLS LINKED TO 1,3,4-OXADIAZOLES AND1,3,4-THIADIAZOLES, Journal of heterocyclic chemistry, 31(6), 1994, pp. 1439-1443
CYCLOOXYGENASE AND 5-LIPOXYGENASE INHIBITORY ACTIVITY OF 2,6 DI-T-BUTYLPHENOLS LINKED BY A SULFUR ATOM TO 1,3,4-THIADIAZOLES AND 1,3,4-OXADIAZOLES
Authors: KRAMER JB BOSCHELLI DH CONNOR DT KOSTLAN CR KUIPERS PJ KENNEDY JA WRIGHT CD BORNEMEIER DA DYER RD
Citation: Jb. Kramer et al., CYCLOOXYGENASE AND 5-LIPOXYGENASE INHIBITORY ACTIVITY OF 2,6 DI-T-BUTYLPHENOLS LINKED BY A SULFUR ATOM TO 1,3,4-THIADIAZOLES AND 1,3,4-OXADIAZOLES, Bioorganic & medicinal chemistry letters, 3(12), 1993, pp. 2827-2830
1,3,4-OXADIAZOLE, 1,3,4-THIADIAZOLE, AND 1,2,4-TRIAZOLE ANALOGS OF THE FENAMATES - IN-VITRO INHIBITION OF CYCLOOXYGENASE AND 5-LIPOXYGENASEACTIVITIES
Authors: BOSCHELLI DH CONNOR DT BORNEMEIER DA DYER RD KENNEDY JA KUIPERS PJ OKONKWO GC SCHRIER DJ WRIGHT CD
Citation: Dh. Boschelli et al., 1,3,4-OXADIAZOLE, 1,3,4-THIADIAZOLE, AND 1,2,4-TRIAZOLE ANALOGS OF THE FENAMATES - IN-VITRO INHIBITION OF CYCLOOXYGENASE AND 5-LIPOXYGENASEACTIVITIES, Journal of medicinal chemistry, 36(13), 1993, pp. 1802-1810
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