Authors:
LU YF
XU H
LIUCHEN LY
CHEN CG
PARTILLA JS
BRINE GA
CARROLL FI
RICE KC
LAI J
PORRECA F
SADEE W
ROTHMAN RB
Citation: Yf. Lu et al., OPIOID PEPTIDE RECEPTOR STUDIES - 7 - THE METHYLFENTANYL CONGENER RTI-4614-4 AND ITS 4 ENANTIOMERS BIND TO DIFFERENT DOMAINS OF THE RAT MU-OPIOID RECEPTOR, Synapse, 28(2), 1998, pp. 117-124
Authors:
FLIPPENANDERSON JL
DESCHAMPS JR
GEORGE C
REDDY PA
LEWIN AH
BRINE GA
SHELDRICK G
NIKIFOROVICH G
Citation: Jl. Flippenanderson et al., X-RAY STRUCTURE OF TYR-D-TIC-PHE-PHE-NH2 (D-TIPP-NH2), A HIGHLY POTENT MU-RECEPTOR SELECTIVE OPIOID AGONIST, The journal of peptide research, 49(5), 1997, pp. 384-393
Authors:
ZERNIG G
ISSAEVITCH T
BROADBEAR JH
BURKE TF
LEWIS JW
BRINE GA
WOODS JH
Citation: G. Zernig et al., RECEPTOR RESERVE AND AFFINITY OF MU-OPIOID AGONISTS IN MOUSE ANTINOCICEPTION - CORRELATION WITH RECEPTOR-BINDING, Life sciences, 57(23), 1995, pp. 2113-2125
Authors:
BRINE GA
STARK PA
LIU Y
CARROLL FI
SINGH P
XU H
ROTHMAN RB
Citation: Ga. Brine et al., ENANTIOMERS OF DIASTEREOMERIC LETHYL)-3-METHYL-4-PIPERIDYL]-N-PHENYLPROPANAMIDES - SYNTHESIS, X-RAY-ANALYSIS, AND BIOLOGICAL-ACTIVITIES, Journal of medicinal chemistry, 38(9), 1995, pp. 1547-1557
Citation: Ga. Brine et al., SYNTHESIS OF 4,4-DISUBSTITUTED PIPERIDINE ANALOGS OF (+ LETHYL)-3-METHYL-4-PIPERIDYL]-N-PHENYLPROPANAMIDE/, Journal of heterocyclic chemistry, 31(2), 1994, pp. 513-520
Authors:
NI Q
XU H
PARTILLA JS
STARK PA
CARROLL FI
BRINE GA
ROTHMAN RB
Citation: Q. Ni et al., STEREOCHEMICAL REQUIREMENTS FOR PSEUDOIRREVERSIBLE INHIBITION OF OPIOID MU RECEPTOR-BINDING BY THE 3-METHYLFENTANYL CONGENERS, RTI-46144 AND ITS ENANTIOMERS - EVIDENCE FOR DIFFERENT BINDING DOMAINS, Synapse, 15(4), 1993, pp. 296-306