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Results: 1-19 |
Results: 19
Synthesis and receptor binding affinity of new selective GluR5 ligands
Authors: Bunch, L Johansen, TH Brauner-Osborne, H Stensbol, TB Johansen, TN Krogsgaard-Larsen, P Madsen, U
Citation: L. Bunch et al., Synthesis and receptor binding affinity of new selective GluR5 ligands, BIO MED CH, 9(4), 2001, pp. 875-879
Resolution, configurational assignment, and enantiopharmacology at glutamate receptors of 2-amino-3-(3-carboxy-5-methyl-4-isoxazolyl)propionic acid (ACPA) and demethyl-ACPA
Authors: Johansen, TN Stensbol, TB Nielsen, B Vogensen, SB Frydenvang, K Slok, FA Brauner-Osborne, H Madsen, U Krogsgaard-Larsen, P
Citation: Tn. Johansen et al., Resolution, configurational assignment, and enantiopharmacology at glutamate receptors of 2-amino-3-(3-carboxy-5-methyl-4-isoxazolyl)propionic acid (ACPA) and demethyl-ACPA, CHIRALITY, 13(9), 2001, pp. 523-532
Cloning and characterization of a human orphan family C G-protein coupled receptor GPRC5D
Authors: Brauner-Osborne, H Jensen, AA Sheppard, PO Brodin, B Krogsgaard-Larsen, P O'Hara, P
Citation: H. Brauner-osborne et al., Cloning and characterization of a human orphan family C G-protein coupled receptor GPRC5D, BBA-GENE ST, 1518(3), 2001, pp. 237-248
Synthesis and pharmacology of 3-isoxazolol amino acids as selective antagonists at group I metabotropic glutamic acid receptors
Authors: Madsen, U Brauner-Osborne, H Frydenvang, K Hvene, L Johansen, TN Nielsen, B Sanchez, C Stensbol, TB Bischoff, F Krogsgaard-Larsen, P
Citation: U. Madsen et al., Synthesis and pharmacology of 3-isoxazolol amino acids as selective antagonists at group I metabotropic glutamic acid receptors, J MED CHEM, 44(7), 2001, pp. 1051-1059
Construction of a high affinity zinc binding site in the metabotropic glutamate receptor mGluR1 - Noncompetitive antagonism originating from the amino-terminal domain of a family C G-protein-coupled receptor
Authors: Jensen, AA Sheppard, PO Jensen, LB O'Hara, PJ Brauner-Osborne, H
Citation: Aa. Jensen et al., Construction of a high affinity zinc binding site in the metabotropic glutamate receptor mGluR1 - Noncompetitive antagonism originating from the amino-terminal domain of a family C G-protein-coupled receptor, J BIOL CHEM, 276(13), 2001, pp. 10110-10118
Pharmacological characterization of homobaclofen on wild type and mutant GABA(B)1b receptors coexpressed with the GABA(B)2 receptor
Authors: Jensen, AA Madsen, BE Krogsgaard-Larsen, P Brauner-Osborne, H
Citation: Aa. Jensen et al., Pharmacological characterization of homobaclofen on wild type and mutant GABA(B)1b receptors coexpressed with the GABA(B)2 receptor, EUR J PHARM, 417(3), 2001, pp. 177-180
Sequence and expression pattern of a novel human orphan G-protein-coupled receptor, GPRC5B, a family C receptor with a short amino-terminal domain
Authors: Brauner-Osborne, H Krogsgaard-Larsen, P
Citation: H. Brauner-osborne et P. Krogsgaard-larsen, Sequence and expression pattern of a novel human orphan G-protein-coupled receptor, GPRC5B, a family C receptor with a short amino-terminal domain, GENOMICS, 65(2), 2000, pp. 121-128
Ionotropic excitatory amino acid receptor ligands. Synthesis and pharmacology of a new amino acid AMPA antagonist
Authors: Madsen, U Slok, FA Stensbol, TB Brauner-Osborne, H Lutzhoft, HCH Poulsen, MV Eriksen, L Krogsgaard-Larsen, P
Citation: U. Madsen et al., Ionotropic excitatory amino acid receptor ligands. Synthesis and pharmacology of a new amino acid AMPA antagonist, EUR J MED C, 35(1), 2000, pp. 69-76
Ligands for glutamate receptors: Design and therapeutic prospects
Authors: Brauner-Osborne, H Egebjerg, J Nielsen, EO Madsen, U Krogsgaard-Larsen, P
Citation: H. Brauner-osborne et al., Ligands for glutamate receptors: Design and therapeutic prospects, J MED CHEM, 43(14), 2000, pp. 2609-2645
Functional importance of the Ala(116)-Pro(136) region in the calcium-sensing receptor - Constitutive activity and inverse agonism in a family C G-protein-coupled receptor
Authors: Jensen, AA Spalding, TA Burstein, ES Sheppard, PO O'Hara, PJ Brann, MR Krogsgaard-Larsen, P Brauner-Osborne, H
Citation: Aa. Jensen et al., Functional importance of the Ala(116)-Pro(136) region in the calcium-sensing receptor - Constitutive activity and inverse agonism in a family C G-protein-coupled receptor, J BIOL CHEM, 275(38), 2000, pp. 29547-29555
A new structural class of subtype-selective inhibitor of cloned excitatoryamino acid transporter, EAAT2
Authors: Brauner-Osborne, H Hermit, MB Nielsen, B Krogsgaard-Larsen, P Johansen, TN
Citation: H. Brauner-osborne et al., A new structural class of subtype-selective inhibitor of cloned excitatoryamino acid transporter, EAAT2, EUR J PHARM, 406(1), 2000, pp. 41-44
The role of Arg(78) in the metabotropic glutamate receptor mGlu(1) for agonist binding and selectivity
Authors: Jensen, AA Sheppard, PO O'Hara, PJ Krogsgaard-Larsen, P Brauner-Osborne, H
Citation: Aa. Jensen et al., The role of Arg(78) in the metabotropic glutamate receptor mGlu(1) for agonist binding and selectivity, EUR J PHARM, 397(2-3), 2000, pp. 247-253
Synthesis and muscarinic receptor pharmacology of a series of 4,5,6,7-tetrahydroisothiazolo[4,5-c]pyridine bioisosteres of arecoline
Authors: Pedersen, H Brauner-Osborne, H Ball, RG Frydenvang, K Meier, E Bogeso, KP Krogsgaard-Larsen, P
Citation: H. Pedersen et al., Synthesis and muscarinic receptor pharmacology of a series of 4,5,6,7-tetrahydroisothiazolo[4,5-c]pyridine bioisosteres of arecoline, BIO MED CH, 7(5), 1999, pp. 795-809
Interaction of CPCCOEt with a chimeric mGlu(1b) and calcium sensing receptor
Authors: Brauner-Osborne, H Jensen, AA Krogsgaard-Larsen, P
Citation: H. Brauner-osborne et al., Interaction of CPCCOEt with a chimeric mGlu(1b) and calcium sensing receptor, NEUROREPORT, 10(18), 1999, pp. 3923-3925
3-Pyrazolone analogues of the 3-isoxazolol metabotropic excitatory amino acid receptor agonist homo-AMPA. Synthesis and pharmacological testing
Authors: Zimmermann, D Janin, YL Brehm, L Brauner-Osborne, H Ebert, B Johansen, TN Madsen, U Krogsgaard-Larsen, P
Citation: D. Zimmermann et al., 3-Pyrazolone analogues of the 3-isoxazolol metabotropic excitatory amino acid receptor agonist homo-AMPA. Synthesis and pharmacological testing, EUR J MED C, 34(11), 1999, pp. 967-976
Synthesis and enantiopharmacology of new AMPA-kainate receptor agonists
Authors: Conti, P De Amici, M De Sarro, G Rizzo, M Stensbol, TB Brauner-Osborne, H Madsen, U Toma, L De Micheli, C
Citation: P. Conti et al., Synthesis and enantiopharmacology of new AMPA-kainate receptor agonists, J MED CHEM, 42(20), 1999, pp. 4099-4107
The agonist-binding domain of the calcium-sensing receptor is located at the amino-terminal domain
Authors: Brauner-Osborne, H Jensen, AA Sheppard, PO O'Hara, P Krogsgaard-Larsen, P
Citation: H. Brauner-osborne et al., The agonist-binding domain of the calcium-sensing receptor is located at the amino-terminal domain, J BIOL CHEM, 274(26), 1999, pp. 18382-18386
Agonists and inverse agonists for the herpesvirus 8-encoded constitutivelyactive seven-transmembrane oncogene product, ORF-74
Authors: Rosenkilde, MM Kledal, TN Brauner-Osborne, H Schwartz, TW
Citation: Mm. Rosenkilde et al., Agonists and inverse agonists for the herpesvirus 8-encoded constitutivelyactive seven-transmembrane oncogene product, ORF-74, J BIOL CHEM, 274(2), 1999, pp. 956-961
Functional pharmacology of cloned heterodimeric GABA(B) receptors expressed in mammalian cells
Authors: Brauner-Osborne, H Krogsgaard-Larsen, P
Citation: H. Brauner-osborne et P. Krogsgaard-larsen, Functional pharmacology of cloned heterodimeric GABA(B) receptors expressed in mammalian cells, BR J PHARM, 128(7), 1999, pp. 1370-1374
Risultati: 1-19 |