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Schols, D
Citation: S. Hatse et al., Mutation of Asp(171) and Asp(262) of the chemokine receptor CXCR4 impairs its coreceptor function for human immunodeficiency virus-1 entry and abrogates the antagonistic activity of AMD3100, MOLEC PHARM, 60(1), 2001, pp. 164-173
Authors:
Matthys, P
Hatse, S
Vermeire, K
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Bridger, G
Henson, GW
De Clercq, E
Billiau, A
Schols, D
Citation: P. Matthys et al., AMD3100, a potent and specific antagonist of the stromal cell-derived factor-1 chemokine receptor CXCR4, inhibits autoimmune joint inflammation in IFN-gamma receptor-deficient mice, J IMMUNOL, 167(8), 2001, pp. 4686-4692
Authors:
Hendrix, CW
Flexner, C
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Fuchs, EJ
Redpath, E
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Henson, GW
Citation: Cw. Hendrix et al., Pharmacokinetics and safety of AMD-3100, a novel antagonist of the CXCR-4 chemokine receptor, in human volunteers, ANTIM AG CH, 44(6), 2000, pp. 1667-1673
Authors:
Blanco, J
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Citation: J. Blanco et al., The CXCR4 antagonist AMD3100 efficiently inhibits cell-surface-expressed human immunodeficiency virus type 1 envelope-induced apoptosis, ANTIM AG CH, 44(1), 2000, pp. 51-56
Authors:
Van Gelder, J
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Citation: J. Van Gelder et al., Evaluation of the potential of ion pair formation to improve the oral absorption of two potent antiviral compounds, AMD3100 and PMPA, INT J PHARM, 186(2), 1999, pp. 127-136
Authors:
Este, JA
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Citation: Ja. Este et al., Activity of different bicyclam derivatives against human immunodeficiency virus depends on their interaction with the CXCR4 chemokine receptor, MOLEC PHARM, 55(1), 1999, pp. 67-73
Authors:
Este, JA
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Bridger, G
Henson, G
Clotet, B
Schols, D
De Clercq, E
Citation: Ja. Este et al., Shift of clinical human immunodeficiency virus type 1 isolates from X4 to R5 and prevention of emergence of the syncytium-inducing phenotype by blockade of CXCR4, J VIROLOGY, 73(7), 1999, pp. 5577-5585