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Results: 1-12 |
Results: 12
DISCOVERY OF YDROXYPROPYL]-(4S)-(4-HYDROXYPHENYL)-2-AZETIDINONE (SCH-58235) - A DESIGNED, POTENT, ORALLY-ACTIVE INHIBITOR OF CHOLESTEROL ABSORPTION
Authors: ROSENBLUM SB HUYNH T AFONSO A DAVIS HR YUMIBE N CLADER JW BURNETT DA
Citation: Sb. Rosenblum et al., DISCOVERY OF YDROXYPROPYL]-(4S)-(4-HYDROXYPHENYL)-2-AZETIDINONE (SCH-58235) - A DESIGNED, POTENT, ORALLY-ACTIVE INHIBITOR OF CHOLESTEROL ABSORPTION, Journal of medicinal chemistry, 41(6), 1998, pp. 973-980
SYNTHESIS OF C3 HETEROATOM-SUBSTITUTED AZETIDINONES THAT DISPLAY POTENT CHOLESTEROL ABSORPTION INHIBITORY ACTIVITY
Authors: MCKITTRICK BA MA K HUIE K YUMIBE N DAVIS H CLADER JW CZARNIECKI M MCPHAIL AT
Citation: Ba. Mckittrick et al., SYNTHESIS OF C3 HETEROATOM-SUBSTITUTED AZETIDINONES THAT DISPLAY POTENT CHOLESTEROL ABSORPTION INHIBITORY ACTIVITY, Journal of medicinal chemistry, 41(5), 1998, pp. 752-759
(-)-SCH-57939 - SYNTHESIS AND PHARMACOLOGICAL PROPERTIES OF A POTENT,METABOLICALLY STABLE CHOLESTEROL ABSORPTION INHIBITOR
Authors: KIRKUP MP RIZVI R SHANKAR BB DUGAR S CLADER JW MCCOMBIE SW LIN SI YUMIBE N HUIE K VANHEEK M COMPTON DS DAVIS HR MCPHAIL AT
Citation: Mp. Kirkup et al., (-)-SCH-57939 - SYNTHESIS AND PHARMACOLOGICAL PROPERTIES OF A POTENT,METABOLICALLY STABLE CHOLESTEROL ABSORPTION INHIBITOR, Bioorganic & medicinal chemistry letters, 6(17), 1996, pp. 2069-2072
STEREOSELECTIVE SYNTHESIS AND BIOLOGICAL-ACTIVITY OF CIS AZETIDINONESAS CHOLESTEROL ABSORPTION INHIBITORS
Authors: MCKITTRICK BA MA K DUGAR S CLADER JW DAVIS H CZARNIECKI M MCPHAIL AT
Citation: Ba. Mckittrick et al., STEREOSELECTIVE SYNTHESIS AND BIOLOGICAL-ACTIVITY OF CIS AZETIDINONESAS CHOLESTEROL ABSORPTION INHIBITORS, Bioorganic & medicinal chemistry letters, 6(16), 1996, pp. 1947-1950
METABOLISM AND STRUCTURE-ACTIVITY DATA-BASED DRUG DESIGN - DISCOVERY OF (-) SCH-53079 AN ANALOG OF THE POTENT CHOLESTEROL ABSORPTION INHIBITOR (-) SCH-48461
Authors: DUGAR S YUMIBE N CLADER JW VIZZIANO M HUIE K VANHEEK M COMPTON DS DAVIS HR
Citation: S. Dugar et al., METABOLISM AND STRUCTURE-ACTIVITY DATA-BASED DRUG DESIGN - DISCOVERY OF (-) SCH-53079 AN ANALOG OF THE POTENT CHOLESTEROL ABSORPTION INHIBITOR (-) SCH-48461, Bioorganic & medicinal chemistry letters, 6(11), 1996, pp. 1271-1274
2-AZETIDINONE CHOLESTEROL ABSORPTION INHIBITORS - STRUCTURE-ACTIVITY-RELATIONSHIPS ON THE HETEROCYCLIC NUCLEUS
Authors: CLADER JW BURNETT DA CAPLEN MA DOMALSKI MS DUGAR S VACCARO W SHER R BROWNE ME ZHAO HR BURRIER RE SALISBURY B DAVIS HR
Citation: Jw. Clader et al., 2-AZETIDINONE CHOLESTEROL ABSORPTION INHIBITORS - STRUCTURE-ACTIVITY-RELATIONSHIPS ON THE HETEROCYCLIC NUCLEUS, Journal of medicinal chemistry, 39(19), 1996, pp. 3684-3693
GAMMA-LACTAMS AND RELATED-COMPOUNDS AS CHOLESTEROL ABSORPTION INHIBITORS - HOMOLOGS OF THE BETA-LACTAM CHOLESTEROL ABSORPTION INHIBITOR SCH-48461
Authors: DUGAR S KIRKUP MP CLADER JW LIN SI RIZVI R SNOW ME DAVIS HR MCCOMBIE SW
Citation: S. Dugar et al., GAMMA-LACTAMS AND RELATED-COMPOUNDS AS CHOLESTEROL ABSORPTION INHIBITORS - HOMOLOGS OF THE BETA-LACTAM CHOLESTEROL ABSORPTION INHIBITOR SCH-48461, Bioorganic & medicinal chemistry letters, 5(24), 1995, pp. 2947-2952
TRANS DIASTEREOSELECTIVE SYNTHESIS OF 3-ALKYL SUBSTITUTED BETA-LACTAMS VIA THE ACID CHLORIDE-IMINE REACTION OF NONACTIVATED ACID-CHLORIDES
Authors: BROWNE M BURNETT DA CAPLEN MA CHEN LY CLADER JW DOMALSKI M DUGAR S PUSHPAVANAM P SHER R VACCARO W VIZIANO M ZHAO HR
Citation: M. Browne et al., TRANS DIASTEREOSELECTIVE SYNTHESIS OF 3-ALKYL SUBSTITUTED BETA-LACTAMS VIA THE ACID CHLORIDE-IMINE REACTION OF NONACTIVATED ACID-CHLORIDES, Tetrahedron letters, 36(15), 1995, pp. 2555-2558
SUBSTITUTED 2-AZASPIRO[5.3]NONAN-1-ONES AS POTENT CHOLESTEROL ABSORPTION INHIBITORS - DEFINING A BINDING CONFORMATION FOR SCH-48461
Authors: DUGAR S CLADER JW CHAN TM DAVIS H
Citation: S. Dugar et al., SUBSTITUTED 2-AZASPIRO[5.3]NONAN-1-ONES AS POTENT CHOLESTEROL ABSORPTION INHIBITORS - DEFINING A BINDING CONFORMATION FOR SCH-48461, Journal of medicinal chemistry, 38(25), 1995, pp. 4875-4877
SUBSTITUTED (1,2-DIARYLETHYL)AMIDE ACYL-COA-CHOLESTEROL ACYLTRANSFERASE INHIBITORS - EFFECT OF POLAR GROUPS ON IN-VITRO AND IN-VIVO ACTIVITY
Authors: CLADER JW BERGER JG BURRIER RE DAVIS HR DOMALSKI M DUGAR S KOGAN TP SALISBURY B VACCARO W
Citation: Jw. Clader et al., SUBSTITUTED (1,2-DIARYLETHYL)AMIDE ACYL-COA-CHOLESTEROL ACYLTRANSFERASE INHIBITORS - EFFECT OF POLAR GROUPS ON IN-VITRO AND IN-VIVO ACTIVITY, Journal of medicinal chemistry, 38(10), 1995, pp. 1600-1607
HYPOCHOLESTEROLEMIC ACTIVITY OF A NOVEL INHIBITOR OF CHOLESTEROL ABSORPTION, SCH-48461
Authors: SALISBURY BG DAVIS HR BURRIER RE BURNETT DA BOYKOW G CAPLEN MA CLEMMONS AL COMPTON DS HOOS LM MCGREGOR DG SCHNITZERPOLOKOFF R SMITH AA WEIG BC ZILLI DL CLADER JW SYBERTZ EJ
Citation: Bg. Salisbury et al., HYPOCHOLESTEROLEMIC ACTIVITY OF A NOVEL INHIBITOR OF CHOLESTEROL ABSORPTION, SCH-48461, Atherosclerosis, 115(1), 1995, pp. 45-63
2-AZETIDINONES AS INHIBITORS OF CHOLESTEROL ABSORPTION
Authors: BURNETT DA CAPLEN MA DAVIS HR BURRIER RE CLADER JW
Citation: Da. Burnett et al., 2-AZETIDINONES AS INHIBITORS OF CHOLESTEROL ABSORPTION, Journal of medicinal chemistry, 37(12), 1994, pp. 1733-1736
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