Authors:
WURCH T
PALMIER C
RAULY I
COLPAERT FC
PAUWELS PJ
Citation: T. Wurch et al., MUTATION OF THR373 IN THE 3RD INTRACELLULAR LOOP OF THE HUMAN ALPHA(2A)-ADRENERGIC RECEPTOR PROMOTES PARTIAL AGONIST ACTIVITY FROM ANTAGONISTS, Naunyn-Schmiedeberg's archives of pharmacology, 358(1), 1998, pp. 642-642
Authors:
JOHN GW
VERSCHEURE Y
INFANTI F
BEL L
PEREZ M
HALAZY S
CHOPIN P
MARIEN M
COLPAERT FC
Citation: Gw. John et al., IN-VIVO PHARMACOLOGICAL ACTIONS OF F-11356, A NOVEL HIGH EFFICACY ANTIMIGRAINE 5-HT1B D RECEPTOR AGONIST/, Naunyn-Schmiedeberg's archives of pharmacology, 358(1), 1998, pp. 5261-5261
Authors:
JOHN GW
VALENTIN JP
LEGRAND B
BONNAFOUS R
PANISSIE A
VIE B
PEREZ M
HALAZY S
PAUWELS PJ
COLPAERT FC
Citation: Gw. John et al., IN-VITRO VASCULAR AND NEURONAL ACTIONS OF F-11356, A NOVEL HIGH EFFICACY 5HT(1B D) RECEPTOR AGONIST, IN MODELS RELEVANT TO MIGRAINE/, Naunyn-Schmiedeberg's archives of pharmacology, 358(1), 1998, pp. 5262-5262
Authors:
PAUWELS PJ
PALMIER C
TARDIF S
WURCH T
PEREZ M
CARILLADURAND E
JOHN GW
HALAZY S
COLPAERT FC
Citation: Pj. Pauwels et al., F-11356, A NEW 5-HT DERIVATIVE, WITH SELECTIVE, POTENT AND HIGH EFFICACY AGONIST PROPERTIES AT 5-HT1B D RECEPTORS/, Naunyn-Schmiedeberg's archives of pharmacology, 358(1), 1998, pp. 5263-5263
Authors:
PAUWELS PJ
PALMIER C
DUPUIS DS
COLPAERT FC
Citation: Pj. Pauwels et al., INTERACTION OF 5 HT1B D LIGANDS WITH RECOMBINANT-H 5-HT1A RECEPTORS -INTRINSIC ACTIVITY AND MODULATION BY G-PROTEIN ACTIVATION STATE/, Naunyn-Schmiedeberg's archives of pharmacology, 357(5), 1998, pp. 490-499
Authors:
KOEK W
PATOISEAU JF
ASSIE MB
COSI C
KLEVEN MS
DUPONTPASSELAIGUE E
CARILLADURAND E
PALMIER C
VALENTIN JP
JOHN G
PAUWELS PJ
TARAYRE JP
COLPAERT FC
Citation: W. Koek et al., F-11440, A POTENT, SELECTIVE, HIGH EFFICACY 5-HT1A RECEPTOR AGONIST WITH MARKED ANXIOLYTIC AND ANTIDEPRESSANT POTENTIAL, The Journal of pharmacology and experimental therapeutics, 287(1), 1998, pp. 266-283
Authors:
DUPUIS DS
PALMIER C
COLPAERT FC
PAUWELS PJ
Citation: Ds. Dupuis et al., AUTORADIOGRAPHY OF SEROTONIN 5-HT1A RECEPTOR-ACTIVATED G-PROTEINS IN GUINEA-PIG BRAIN SECTIONS BY AGONIST-STIMULATED [S-35] GTP-GAMMA-S BINDING, Journal of neurochemistry, 70(3), 1998, pp. 1258-1268
Citation: Ds. Dupuis et al., G-PROTEIN ACTIVATION AT 5-HT1A RECEPTORS BY THE 5-HT(1F) LIGAND LY334370 IN GUINEA-PIG BRAIN SECTIONS AND RECOMBINANT CELL-LINES, British Journal of Pharmacology, 124(2), 1998, pp. 283-290
Authors:
PAGNIEZ F
VALENTIN JP
VIEU S
COLPAERT FC
JOHN GW
Citation: F. Pagniez et al., PHARMACOLOGICAL ANALYSIS OF THE HEMODYNAMIC-EFFECTS OF 5-HT1B D RECEPTOR AGONISTS IN THE NORMOTENSIVE RAT/, British Journal of Pharmacology, 123(2), 1998, pp. 205-214
Citation: Pj. Pauwels et al., PHARMACOLOGICAL ANALYSIS OF G-PROTEIN ACTIVATION MEDIATED BY GUINEA-PIG RECOMBINANT 5-HT1B RECEPTORS IN C6-GLIAL CELLS - SIMILARITIES WITH THE HUMAN 5-HT1B RECEPTOR, British Journal of Pharmacology, 123(1), 1998, pp. 51-62
Authors:
AMOUREUX MC
VANGOOL D
HERRERO MT
DOM R
COLPAERT FC
PAUWELS PJ
Citation: Mc. Amoureux et al., REGULATION OF METALLOTHIONEIN-III (GIF) MESSENGER-RNA IN THE BRAIN OFPATIENTS WITH ALZHEIMER-DISEASE IS NOT IMPAIRED, Molecular and chemical neuropathology, 32(1-3), 1997, pp. 101-121
Authors:
PAUWELS PJ
TARDIF S
PALMIER C
WURCH T
COLPAERT FC
Citation: Pj. Pauwels et al., HOW EFFICACIOUS ARE 5-HT1B D RECEPTOR LIGANDS - AN ANSWER FROM GTP-GAMMA-S BINDING-STUDIES WITH STABLY TRANSFECTED C6-GLIAL CELL-LINES/, Neuropharmacology, 36(4-5), 1997, pp. 499-512
Citation: Pj. Pauwels et al., STIMULATED [S-35] GTP-GAMMA-S BINDING BY 5-HT1A RECEPTOR AGONISTS IN RECOMBINANT CELL-LINES - MODULATION OF APPARENT EFFICACY BY G-PROTEIN ACTIVATION STATE, Naunyn-Schmiedeberg's archives of pharmacology, 356(5), 1997, pp. 551-561
Authors:
BERTOLINO F
VALENTIN JP
PATOISEAU JF
RIEU JP
COLPAERT FC
JOHN GW
Citation: F. Bertolino et al., EVIDENCE FOR PARTIAL AGONIST PROPERTIES OF DALTROBAN (BM-13,505) AT TP RECEPTORS IN THE ANESTHETIZED OPEN-CHEST RAT, Naunyn-Schmiedeberg's archives of pharmacology, 356(4), 1997, pp. 462-466
Citation: T. Wurch et al., SEQUENCE AND FUNCTIONAL-ANALYSIS OF CLONED GUINEA-PIG AND RAT SEROTONIN 5-HT1D RECEPTORS, COMMON PHARMACOLOGICAL FEATURES WITHIN THE 5-HT1DRECEPTOR SUBFAMILY, Journal of neurochemistry, 68(1), 1997, pp. 410-418
Citation: T. Wurch et al., RECOMBINANT SAPHENOUS-VEIN 5-HT1B RECEPTORS OF THE RABBIT - COMPARATIVE PHARMACOLOGY WITH HUMAN 5-HT1B RECEPTORS, British Journal of Pharmacology, 120(1), 1997, pp. 153-159
Authors:
WURCH T
CHASTAGNIER C
PALMIER C
COLPAERT FC
PAUWELS PJ
Citation: T. Wurch et al., A 413 BP REGION UPSTREAM THE HUMAN 5-HT1A RECEPTOR GENE IS SUFFICIENTFOR ITS IN-VITRO EXPRESSION, Neuroscience research communications, 19(2), 1996, pp. 75-82
Authors:
WURCH T
CATHALA C
PALMIER C
VALENTIN JP
JOHN GW
COLPAERT FC
PAUWELS PJ
Citation: T. Wurch et al., MOLECULAR-CLONING AND IDENTIFICATION OF A RABBIT SAPHENOUS-VEIN 5-HT1D-BETA RECEPTOR GENE, Neuroscience research communications, 18(3), 1996, pp. 155-162
Citation: Pj. Pauwels et al., PROMOTION OF CELL-GROWTH BY STIMULATION OF CLONED HUMAN 5-HT1D RECEPTOR-SITES IN TRANSFECTED C6-GLIAL CELLS IS HIGHLY SENSITIVE TO INTRINSIC ACTIVITY AT 5-HT1D RECEPTORS, Naunyn-Schmiedeberg's archives of pharmacology, 354(2), 1996, pp. 136-144
Citation: Pj. Pauwels et al., PHARMACOLOGY OF CLONED HUMAN 5-HT1D RECEPTOR-MEDIATED FUNCTIONAL-RESPONSES IN STABLY TRANSFECTED RAT C6-GLIAL CELL-LINES - FURTHER EVIDENCEDIFFERENTIATING HUMAN 5-HT1D AND 5-HT1B RECEPTORS, Naunyn-Schmiedeberg's archives of pharmacology, 353(2), 1996, pp. 144-156
Authors:
PAUWELS PJ
WURCH T
AMOUREUX MC
PALMIER C
COLPAERT FC
Citation: Pj. Pauwels et al., STIMULATION OF CLONED HUMAN SEROTONIN 5-HT1D-BETA RECEPTOR-SITES IN STABLY TRANSFECTED C6 GLIAL-CELLS PROMOTES CELL-GROWTH, Journal of neurochemistry, 66(1), 1996, pp. 65-73
Citation: Pj. Pauwels et Fc. Colpaert, STEREOSELECTIVITY OF 8-OH-DPAT ENANTIOMERS AT CLONED HUMAN 5-HT1D RECEPTOR-SITES, European journal of pharmacology, 300(1-2), 1996, pp. 137-139