Citation: Yf. Hu et al., SYNTHESIS OF 17R)-17-HYDROXY-14,15-SECOANDROST-4-EN-15-YN-3-ONE AND 17S)-17-HYDROXY-14,15-SECOANDROST-4-EN-15-YN-3-ONE AND THE X-RAY CRYSTAL-STRUCTURE OF THE (17S)-DIASTEREOMER, Steroids, 60(6), 1995, pp. 491-496
Citation: Yf. Hu et al., SYNTHESIS OF 17R)-17-HYDROXY-14,15-SECOANDROST-4-EN-15-YN-3-ONE AND 17S)-17-HYDROXY-14,15-SECOANDROST-4-EN-15-YN-3-ONE AND THE X-RAY CRYSTAL-STRUCTURE OF THE (17S)-DIASTEREOMER (VOL 60, PG 250, 1995), Steroids, 60(6), 1995, pp. 497-497
Citation: Yf. Hu et al., SYNTHESIS OF (17R) AND 17S)-17-HYDROXY-14,15-SECOANDROST-4-EN-16-YN-3-ONE AND THE X-RAY CRYSTAL-STRUCTURE OF THE (17S)-DIASTEREOMER, Steroids, 60(3), 1995, pp. 250-255
Citation: Ra. Gross et al., UNIQUE ACTION OF ANTICONVULSANT ALKYL-SUBSTITUTED THIOBUTYROLACTONES - REDUCTION OF LOW-THRESHOLD AND HIGH-THRESHOLD NEURONAL CA CURRENTS, Neurology, 45(4), 1995, pp. 362-362
Authors:
HOLLAND KD
MATHEWS GC
BOLOSSY AM
TUCKER JB
REDDY PA
COVEY DF
FERRENDELLI JA
ROTHMAN SM
Citation: Kd. Holland et al., DUAL MODULATION OF THE GAMMA-AMINOBUTYRIC-ACID TYPE-A RECEPTOR IONOPHORE BY ALKYL-SUBSTITUTED GAMMA-BUTYROLACTONES, Molecular pharmacology, 47(6), 1995, pp. 1217-1223
Citation: Yf. Hu et al., NEUROSTEROID ANALOGS .2. TOTAL SYNTHESIS AND ELECTROPHYSIOLOGICAL EVALUATION OF BENZ[E]INDENE ANALOGS OF THE ANESTHETIC STEROID ALPHAXALONE, Journal of organic chemistry, 60(12), 1995, pp. 3619-3625
Citation: Mc. Han et al., NEUROSTEROID ANALOGS .3. THE SYNTHESIS AND ELECTROPHYSIOLOGICAL EVALUATION OF BENZ[E]INDENE CONGENERS OF NEUROACTIVE STEROIDS HAVING THE 5-BETA CONFIGURATION, Journal of medicinal chemistry, 38(22), 1995, pp. 4548-4556
Citation: M. Xu et al., INTERACTION OF PICROTOXIN WITH GABA(A) RECEPTOR CHANNEL-LINING RESIDUES PROBED IN CYSTEINE MUTANTS, Biophysical journal, 69(5), 1995, pp. 1858-1867
Citation: Mg. Jakoby et al., LOCALIZATION OF TOLBUTAMIDE BINDING SITES ON HUMAN SERUM-ALBUMIN USING TITRATION CALORIMETRY AND HETERONUCLEAR 2-D NMR, Biochemistry, 34(27), 1995, pp. 8780-8787
Authors:
MATHEWS GC
BOLOSSY AM
HOLLAND KD
ISENBERG KE
COVEY DF
FERRENDELLI JA
ROTHMAN SM
Citation: Gc. Mathews et al., DEVELOPMENTAL ALTERATION IN GABA(A) RECEPTOR STRUCTURE AND PHYSIOLOGICAL-PROPERTIES IN CULTURED CEREBELLAR GRANULE NEURONS, Neuron, 13(1), 1994, pp. 149-158
Citation: Sj. Weiner et al., SYNTHESIS OF C-13, N-15-ENRICHED ALPHA-DICARBONYL MODEL ADDUCTS TO DETERMINE THE UTILITY OF C-13 AND N-15 NMR FOR STUDYING MECHANISM-BASED INACTIVATION OF CYTOCHROMES-P-450 BY SUBSTITUTED DICHLOROACETAMIDES, Magnetic resonance in chemistry, 32(2), 1994, pp. 122-127
Authors:
PETERSON EM
XU K
HOLLAND KD
MCKEON AC
ROTHMAN SM
FERRENDELLI JA
COVEY DF
Citation: Em. Peterson et al., ALPHA-SPIROCYCLOPENTYL- AND ALPHA-SPIROCYCLOPROPYL-GAMMA-BUTYROLACTONES - CONFORMATIONALLY CONSTRAINED DERIVATIVES OF ANTICONVULSANT AND CONVULSANT ALPHA,ALPHA-DISUBSTITUTED GAMMA-BUTYROLACTONES, Journal of medicinal chemistry, 37(2), 1994, pp. 275-286
Authors:
SCHLEGEL BP
PAWLOWSKI JE
HU YF
SCOLNICK DM
COVEY DF
PENNING TM
Citation: Bp. Schlegel et al., SECOSTEROID MECHANISM-BASED INACTIVATORS AND SITE-DIRECTED MUTAGENESIS AS PROBES FOR STEROID-HORMONE RECOGNITION BY 3-ALPHA-HYDROXYSTEROID DEHYDROGENASE, Biochemistry, 33(34), 1994, pp. 10367-10374
Citation: Sj. Zimniski et al., INHIBITION OF GROWTH AND APPEARANCE OF ESTROGEN-DEPENDENT RAT MAMMARY-TUMORS BY 10-PROPARGYLESTR-4-ENE-3,17-DIONE, AN AROMATASE INHIBITOR, Breast cancer research and treatment, 26(1), 1993, pp. 15-21
Citation: Kw. Yoon et al., MULTIPLE MECHANISMS OF PICROTOXIN BLOCK OF GABA-INDUCED CURRENTS IN RAT HIPPOCAMPAL-NEURONS, Journal of physiology, 464, 1993, pp. 423-439
Citation: Yf. Hu et al., NEUROSTEROID ANALOGS - STRUCTURE-ACTIVITY STUDIES OF BENZ[E]INDENE MODULATORS OF GABA(A) RECEPTOR FUNCTION .1. THE EFFECT OF 6-METHYL SUBSTITUTION ON THE ELECTROPHYSIOLOGICAL ACTIVITY OF 7-SUBSTITUTED BENZ[E]INDENE-3-CARBONITRILES, Journal of medicinal chemistry, 36(24), 1993, pp. 3956-3967
Authors:
HOLLAND KD
BOULEY MG
COVEY DF
FERRENDELLI JA
Citation: Kd. Holland et al., ALKYL-SUBSTITUTED GAMMA-BUTYROLACTONES ACT AT A DISTINCT SITE ALLOSTERICALLY LINKED TO THE TBPS PICROTOXININ SITE ON THE GABA(A)RECEPTOR COMPLEX, Brain research, 615(1), 1993, pp. 170-174