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CREGGE RJ
DURHAM SL
FARR RA
GALLION SL
HARE CM
HOFFMAN RV
JANUSZ MJ
KIM HO
KOEHL JR
MEHDI S
METZ WA
PEET NP
PELTON JT
SCHREUDER HA
SUNDER S
TARDIF C
Citation: Rj. Cregge et al., INHIBITION OF HUMAN NEUTROPHIL ELASTASE - 4 - DESIGN, SYNTHESIS, X-RAY CRYSTALLOGRAPHIC ANALYSIS, AND STRUCTURE-ACTIVITY-RELATIONSHIPS FOR A SERIES OF P-2-MODIFIED, ORALLY-ACTIVE PEPTIDYL PENTAFLUOROETHYL KETONES, Journal of medicinal chemistry, 41(14), 1998, pp. 2461-2480
Authors:
BURKHART JP
KOEHL JR
MEHDI S
DURHAM SL
JANUSZ MJ
HUBER EW
ANGELASTRO MR
SUNDER S
METZ WA
SHUM PW
CHEN TM
BEY P
CREGGE RJ
PEET NP
Citation: Jp. Burkhart et al., INHIBITION OF HUMAN NEUTROPHIL ELASTASE .3. AN ORALLY-ACTIVE ENOL ACETATE PRODRUG, Journal of medicinal chemistry, 38(2), 1995, pp. 223-233
Authors:
PODLOGAR BL
FARR RA
FRIEDRICH D
TARNUS C
HUBER EW
CREGGE RJ
SCHIRLIN D
Citation: Bl. Podlogar et al., DESIGN, SYNTHESIS, AND CONFORMATIONAL-ANALYSIS OF A NOVEL MACROCYCLICHIV-PROTEASE INHIBITOR, Journal of medicinal chemistry, 37(22), 1994, pp. 3684-3692