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Results: 1-13 |
Results: 13
Highly potent side-chain to side-chain cyclized enkephalin analogues containing a carbonyl bridge: Synthesis, biology and conformation
Authors: Pawlak, D Oleszczuk, M Wojcik, J Pachulska, M Chung, NN Schiller, PW Izdebski, J
Citation: D. Pawlak et al., Highly potent side-chain to side-chain cyclized enkephalin analogues containing a carbonyl bridge: Synthesis, biology and conformation, J PEPT SCI, 7(3), 2001, pp. 128-140
Stereospecific synthesis of (2S)-2-methyl-3-(2 ',6 '-dimethyl-4 '-hydroxyphenyl)-propionic acid (Mdp) and its incorporation into an opioid peptide
Authors: Lu, YX Weltrowska, G Lemieux, C Chung, NN Schiller, PW
Citation: Yx. Lu et al., Stereospecific synthesis of (2S)-2-methyl-3-(2 ',6 '-dimethyl-4 '-hydroxyphenyl)-propionic acid (Mdp) and its incorporation into an opioid peptide, BIOORG MED, 11(3), 2001, pp. 323-325
Induction chemotherapy with mitomycin, epirubicin, cisplatin, fluorouracil, and leucovorin followed by radiotherapy in the treatment of locoregionally advanced nasopharyngeal carcinoma
Authors: Hong, RL Ting, LL Ko, JY Hsu, MM Sheen, TS Lou, PJ Wang, CC Chung, NN Lui, LT
Citation: Rl. Hong et al., Induction chemotherapy with mitomycin, epirubicin, cisplatin, fluorouracil, and leucovorin followed by radiotherapy in the treatment of locoregionally advanced nasopharyngeal carcinoma, J CL ONCOL, 19(23), 2001, pp. 4305-4313
Pseudoproline-containing analogues of morphiceptin and endomorphin-2: Evidence for a cis Tyr-Pro amide bond in the bioactive conformation
Authors: Keller, M Boissard, C Patiny, L Chung, NN Lemieux, C Mutter, M Schiller, PW
Citation: M. Keller et al., Pseudoproline-containing analogues of morphiceptin and endomorphin-2: Evidence for a cis Tyr-Pro amide bond in the bioactive conformation, J MED CHEM, 44(23), 2001, pp. 3896-3903
[2 ',6 '-dimethyltyrosine]dynorphin A(1-11)-NH2 analogues lacking an N-terminal amino group: Potent and selective kappa opioid antagonists
Authors: Lu, YX Nguyen, TMD Weltrowska, G Berezowska, I Lemieux, C Chung, NN Schiller, PW
Citation: Yx. Lu et al., [2 ',6 '-dimethyltyrosine]dynorphin A(1-11)-NH2 analogues lacking an N-terminal amino group: Potent and selective kappa opioid antagonists, J MED CHEM, 44(19), 2001, pp. 3048-3053
Synthesis and in vitro opioid activity profiles of DALDA analogues
Authors: Schiller, PW Nguyen, TMD Berezowska, I Dupuis, S Weltrowska, G Chung, NN Lemieux, C
Citation: Pw. Schiller et al., Synthesis and in vitro opioid activity profiles of DALDA analogues, EUR J MED C, 35(10), 2000, pp. 895-901
Novel ligands lacking a positive charge for the delta- and mu-opioid receptors
Authors: Schiller, PW Berezowska, I Nguyen, TMD Schmidt, R Lemieux, C Chung, NN Falcone-Hindley, ML Yao, WQ Liu, J Iwama, S Smith, AB Hirschmann, R
Citation: Pw. Schiller et al., Novel ligands lacking a positive charge for the delta- and mu-opioid receptors, J MED CHEM, 43(4), 2000, pp. 551-559
[Pro(3)]Dyn A(1-11)-NH2: A dynorphin analogue with high selectivity for the kappa opioid receptor
Authors: Schlechtingen, G Zhang, L Maycock, A DeHaven, RN Daubert, JD Cassel, J Chung, NN Schiller, PW Goodman, M
Citation: G. Schlechtingen et al., [Pro(3)]Dyn A(1-11)-NH2: A dynorphin analogue with high selectivity for the kappa opioid receptor, J MED CHEM, 43(14), 2000, pp. 2698-2702
Subtleties of structure-agonist versus antagonist relationships of opioid peptides and peptidomimetics
Authors: Schiller, PW Weltrowska, G Schmidt, R Berezowska, I Nguyen, TMD Lemieux, C Chung, NN Carpenter, KA Wilkes, BC
Citation: Pw. Schiller et al., Subtleties of structure-agonist versus antagonist relationships of opioid peptides and peptidomimetics, J RECEPT SI, 19(1-4), 1999, pp. 573-588
The opioid mu agonist/delta antagonist DIPP-NH2[Psi] produces a potent analgesic effect, no physical dependence, and less tolerance than morphine in rats
Authors: Schiller, PW Fundytus, ME Merovitz, L Weltrowska, G Nguyen, TMD Lemieux, C Chung, NN Coderre, TJ
Citation: Pw. Schiller et al., The opioid mu agonist/delta antagonist DIPP-NH2[Psi] produces a potent analgesic effect, no physical dependence, and less tolerance than morphine in rats, J MED CHEM, 42(18), 1999, pp. 3520-3526
The TIPP opioid peptide family: Development of delta antagonists, delta agonists, and mixed mu agonist/delta antagonists
Authors: Schiller, PW Weltrowska, G Berezowska, I Nguyen, TMD Wilkes, BC Lemieux, C Chung, NN
Citation: Pw. Schiller et al., The TIPP opioid peptide family: Development of delta antagonists, delta agonists, and mixed mu agonist/delta antagonists, BIOPOLYMERS, 51(6), 1999, pp. 411-425
Enkephalin analogs containing 4,4-difluoro-2-aminobutyric acid: Synthesis and fluorine effect on the biological activity
Authors: Winkler, D Sewald, N Burger, K Chung, NN Schiller, PW
Citation: D. Winkler et al., Enkephalin analogs containing 4,4-difluoro-2-aminobutyric acid: Synthesis and fluorine effect on the biological activity, J PEPT SCI, 4(8), 1998, pp. 496-501
Side chain methyl substitution in the delta-opioid receptor antagonist TIPP has an important effect on the activity profile
Authors: Tourwe, D Mannekens, E Diem, TNT Verheyden, P Jaspers, H Toth, G Peter, A Kertesz, I Torok, G Chung, NN Schiller, PW
Citation: D. Tourwe et al., Side chain methyl substitution in the delta-opioid receptor antagonist TIPP has an important effect on the activity profile, J MED CHEM, 41(26), 1998, pp. 5167-5176
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