Authors:
Boyle, CD
Chackalamannil, S
Clader, JW
Greenlee, WJ
Josien, HB
Kaminski, JJ
Kozlowski, JA
McCombie, SW
Nazareno, DV
Tagat, JR
Wang, YG
Zhou, GW
Billard, W
Binch, H
Crosby, G
Cohen-Williams, M
Coffin, VL
Cox, KA
Grotz, DE
Duffy, RA
Ruperto, V
Lachowicz, JE
Citation: Cd. Boyle et al., Metabolic stabilization of benzylidene ketal M-2 muscarinic receptor antagonists via halonaphthoic acid substitution, BIOORG MED, 11(17), 2001, pp. 2311-2314
Authors:
Strizki, JM
Xu, S
Wagner, NE
Wojcik, L
Liu, J
Hou, Y
Endres, M
Palani, A
Shapiro, S
Clader, JW
Greenlee, WJ
Tagat, JR
McCombie, S
Cox, K
Fawzi, AB
Chou, CC
Pugliese-Sivo, C
Davies, L
Moreno, ME
Ho, DD
Trkola, A
Stoddart, CA
Moore, JP
Reyes, GR
Baroudy, BM
Citation: Jm. Strizki et al., SCH-C (SCH 351125), an orally bioavailable, small molecule antagonist of the chemokine receptor CCR5, is a potent inhibitor of HIV-1 infection in vitro and in vivo, P NAS US, 98(22), 2001, pp. 12718-12723
Authors:
Palani, A
Shapiro, S
Clader, JW
Greenlee, WJ
Cox, K
Strizki, J
Endres, M
Baroudy, BM
Citation: A. Palani et al., Discovery of 4-[(Z)-(4-bromophenyl)-(ethoxyimino)methyll-1 '-[(2,4-dimethyl-3-pyridinyl)carbonyl]-4 '-methyl-1,4 '-bipiperidine N-oxide (SCH 351125):An orally bioavailable human CCR5 antagonist for the treatment of HIV infection, J MED CHEM, 44(21), 2001, pp. 3339-3342
Authors:
Wang, YG
Chackalamannil, S
Hu, ZY
Clader, JW
Greenlee, W
Billard, W
Binch, H
Crosby, G
Ruperto, V
Duffy, RA
McQuade, R
Lachowicz, JE
Citation: Yg. Wang et al., Design and synthesis of piperidinyl piperidine analogues as potent and selective M-2 muscarinic receptor antagonists, BIOORG MED, 10(20), 2000, pp. 2247-2250
Authors:
Billard, W
Binch, H
Bratzler, K
Chen, LY
Crosby, G
Duffy, RA
Dugar, S
Lachowicz, J
McQuade, R
Pushpavanam, P
Ruperto, VB
Taylor, LA
Clader, JW
Citation: W. Billard et al., Diphenylsulfone muscarinic antagonists: Piperidine derivatives with high M-2 selectivity and improved potency, BIOORG MED, 10(19), 2000, pp. 2209-2212