Authors:
Dupuis, DS
Wurch, T
Tardif, S
Colpaert, FC
Pauwels, PJ
Citation: Ds. Dupuis et al., Modulation of 5-HT1A receptor activation by its interaction with wild-typeand mutant G(alpha i3) proteins, NEUROPHARM, 40(1), 2001, pp. 36-47
Authors:
Pauwels, PJ
Wurch, T
Tardif, S
Finana, F
Colpaert, FC
Citation: Pj. Pauwels et al., Analysis of ligand activation of alpha(2)-adrenoceptor subtypes under conditions of equal G alpha protein stoichiometry, N-S ARCH PH, 363(5), 2001, pp. 526-536
Authors:
Junquero, D
Bruniquel, F
N'Guyen, X
Autin, JM
Patoiseau, JF
Degryse, AD
Colpaert, FC
Delhon, A
Citation: D. Junquero et al., F 12511, a novel ACAT inhibitor, and atorvastatin regulate endogenous hypercholesterolemia in a synergistic manner in New Zealand rabbits fed a casein-enriched diet, ATHEROSCLER, 155(1), 2001, pp. 131-142
Authors:
Bardin, L
Tarayre, JP
Koek, W
Colpaert, FC
Citation: L. Bardin et al., In the formalin model of tonic nociceptive pain, 8-OH-DPAT produces 5-HT1Areceptor-mediated, behaviorally specific analgesia, EUR J PHARM, 421(2), 2001, pp. 109-114
Authors:
Koek, W
Vacher, B
Cosi, C
Assie, MB
Patoiseau, JF
Pauwels, PJ
Colpaert, FC
Citation: W. Koek et al., 5-HT1A receptor activation and antidepressant-like effects: F 13714 has high efficacy and marked antidepressant potential, EUR J PHARM, 420(2-3), 2001, pp. 103-112
Authors:
Pauwels, PJ
Tardif, S
Wurch, T
Colpaert, FC
Citation: Pj. Pauwels et al., Real-time analysis of dopamine: antagonist interactions at recombinant human D-2long receptor upon modulation of its activation state, BR J PHARM, 134(1), 2001, pp. 88-97
Citation: Pj. Pauwels et al., Differential signalling of both wild-type and Thr(343) Arg dopamine D-2short receptor by partial agonists in a G-protein-dependent manner, BIOCH PHARM, 62(6), 2001, pp. 723-732
Authors:
Pauwels, PJ
Tardif, S
Colpaert, FC
Wurch, T
Citation: Pj. Pauwels et al., Modulation of ligand responses by coupling of alpha(2A)-adrenoceptors to diverse G(alpha)-proteins, BIOCH PHARM, 61(9), 2001, pp. 1079-1092
Authors:
Junquero, D
Pilon, A
Carilla-Durand, E
Patoiseau, JF
Tarayre, JP
Torpier, G
Staels, B
Fruchart, JC
Colpaert, FC
Clavey, V
Delhon, A
Citation: D. Junquero et al., Lack of toxic effects of F 12511, a novel potent inhibitor of acylcoenzymeA: cholesterol O-acyltransferase, on human adrenocortical cells in culture, BIOCH PHARM, 61(4), 2001, pp. 387-398
Authors:
Junquero, D
Oms, P
Carilla-Durand, E
Autin, JM
Tarayre, JP
Degryse, AD
Patoiseau, JF
Colpaert, FC
Delhon, A
Citation: D. Junquero et al., Pharmacological profile of F 12511, (S)-2 ',3 ',5 '-trimethyl-4 '-hydroxy-alpha-dodecylthioacetanilide a powerful and systemic acylcoenzyme A: cholesterol acyltransferase inhibitor, BIOCH PHARM, 61(1), 2001, pp. 97-108
Authors:
Prinssen, EPM
Koek, W
Colpaert, FC
Kleven, MS
Citation: Epm. Prinssen et al., Repeated treatment with 8-OH-DPAT induces tolerance to its ability to produce the 5-HT1A behavioural syndrome, but not to its ability to attenuate haloperidol-induced, BEHAV PHARM, 11(3-4), 2000, pp. 299-305
Authors:
Colpaert, FC
Slot, LAB
Koek, W
Dupuis, DS
Citation: Fc. Colpaert et al., Memory of an operant response and of depressed mood retained in activationstates of 5-HT1A receptors: evidence from rodent models, BEH BRA RES, 117(1-2), 2000, pp. 41-51
Citation: Pj. Pauwels et Fc. Colpaert, Heterogeneous ligand-mediated Ca++ responses at wt and mutant alpha(2A)-adrenoceptors suggest multiple ligand activation binding sites at the alpha(2A)-adrenoceptor, NEUROPHARM, 39(11), 2000, pp. 2101-2111
Authors:
Pauwels, PJ
Finana, F
Tardif, S
Colpaert, FC
Wurch, T
Citation: Pj. Pauwels et al., Agonist efficacy at the alpha(2A)-adrenoceptor : G(alpha 15) fusion protein: an analysis based on Ca2+ responses, N-S ARCH PH, 361(6), 2000, pp. 672-679
Authors:
Pauwels, PJ
Tardif, S
Wurch, T
Colpaert, FC
Citation: Pj. Pauwels et al., Facilitation of constitutive alpha(2A)-adrenoceptor activity by both single amino acid mutation (Thr(373)Lys) and G(alpha o) protein coexpression: Evidence for inverse agonism, J PHARM EXP, 292(2), 2000, pp. 654-663
Authors:
Pauwels, PJ
Tardif, S
Finana, F
Wurch, T
Colpaert, FC
Citation: Pj. Pauwels et al., Ligand-receptor interactions as controlled by wild-type and mutant Thr(370)Lys alpha(2B)-adrenoceptor-G(alpha 15) fusion proteins, J NEUROCHEM, 74(1), 2000, pp. 375-384
Citation: Pj. Pauwels et Fc. Colpaert, Partial to complete antagonism by putative antagonists at the wild-type alpha(2C)-adrenoceptor based on kinetic analyses of agonist : antagonist interactions, BR J PHARM, 131(7), 2000, pp. 1385-1390