Authors:
HEWLETT WA
SCHMIDT DE
MASON NS
TRIVEDI BL
EBERT MH
DEPAULIS T
Citation: Wa. Hewlett et al., SYNTHESIS AND 5-HT-3 RECEPTOR-BINDING OF 2-(HALO)ALKOXYL AND 3-(HALO)ALKOXYL SUBSTITUTED N-(1-AZABICYCLO[2.2.2]OCT-3-YL)-5-CHLOROBENZAMIDESAS POTENTIAL RADIOLIGANDS, Nuclear medicine and biology, 25(2), 1998, pp. 141-153
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HEWLETT WA
FRIDMAN S
TRIVEDI BL
SCHMIDT DE
DEPAULIS T
EBERT MH
Citation: Wa. Hewlett et al., CHARACTERIZATION OF DESAMINO-5-[I-125]IODO-3-METHOXYZACOPRIDE ([I-125]MIZAC) BINDING TO 5-HT3 RECEPTORS IN THE RAT-BRAIN, Progress in neuro-psychopharmacology & biological psychiatry, 22(2), 1998, pp. 397-410
Authors:
DEPAULIS T
HEWLETT WA
SCHMIDT DE
MASON NS
TRIVEDI BL
EBERT MH
Citation: T. Depaulis et al., SYNTHESIS AND 5-HT-3 RECEPTOR-BINDING ACTIVITY OF DIMETHOXY-N-(1-AZABICYCLO[2.2.2]OCT-3-YL)BENZAMIDE AND ITS 5-HALOGEN-2-ALKOXYL HOMOLOGS, European journal of medicinal chemistry, 32(5), 1997, pp. 385-396
Authors:
HEWLETT WA
DEPAULIS T
MASON NS
SCHMIDT DE
TRIVEDI BL
ZHANG ZJ
EBERT MH
Citation: Wa. Hewlett et al., SYNTHESIS AND RADIOLABELING OF -METHOXY-N-(1-AZABICYCLO[2.2.2]OCT-3-YL)BENZAMIDE, THE ACTIVE ENANTIOMER OF [I-125] IODOZACOPRIDE, AND REEVALUATION OF ITS 5-HT3 RECEPTOR AFFINITY, Chemical and Pharmaceutical Bulletin, 45(12), 1997, pp. 2079-2084
Authors:
DEPAULIS T
TRIVEDI BL
ZHANG ZJ
SCHMIDT DE
EBERT MH
HEWLETT WA
Citation: T. Depaulis et al., 2-METHOXY-N-(1-AZABICYCLO[2.2.2]OCT-3-YL)BENZAMIDE (TRIZAC), A HIGH-AFFINITY LIGAND FOR THE 5-HT-3 RECEPTOR, Bioorganic & medicinal chemistry letters, 6(22), 1996, pp. 2657-2662
Authors:
MASON NS
HEWLETT WA
EBERT MH
SCHMIDT DE
DEPAULIS T
Citation: Ns. Mason et al., LABELING OF (S)-DES-4-AMINO-3-[I-125]IODOZACOPRIDE (DAIZAC), A HIGH-AFFINITY RADIOLIGAND FOR THE 5-HT-3 RECEPTOR, Journal of labelled compounds & radiopharmaceuticals, 38(11), 1996, pp. 955-961
Authors:
VOTAW JR
ANSARI MS
MASON NS
SCHMIDT D
DEPAULIS T
HOLBURN G
CLANTON JA
VOTAW DB
MANNING RG
KESSLER RM
Citation: Jr. Votaw et al., DOSIMETRY OF IODINE-123-EPIDEPRIDE - A DOPAMINE D2 RECEPTOR-LIGAND, The Journal of nuclear medicine, 36(7), 1995, pp. 1316-1321
Authors:
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DEPAULIS T
NEERGAARD JR
BARON BM
SIEGEL BW
SEEMAN P
VANTOL HHM
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SMITH HE
Citation: St. Phillips et al., BINDING OF 5H-DIBENZO[A,D]CYCLOHEPTENE AND DIBENZ[B,F]OXEPIN ANALOGS OF CLOZAPINE TO DOPAMINE AND SEROTONIN RECEPTORS, Journal of medicinal chemistry, 38(4), 1995, pp. 708-714
Authors:
HEWLETT WA
DEPAULIS T
SCHMIDT DE
TRIVEDI BL
MASON NS
EBERT MH
Citation: Wa. Hewlett et al., I-125 LIZAC, A NOVEL LIGAND-BINDING WITH HIGH-AFFINITY TO 5-HT-3 CNS RECEPTORS, Biological psychiatry, 37(9), 1995, pp. 668-668
Authors:
KESSLER RM
MASON NS
ANSARI MS
DEPAULIS T
CLANTON JA
MANNING RG
HOLBURN G
FORRESTER JW
Citation: Rm. Kessler et al., N-ALLYL EPIDEPRIDE - AN EXTREMELY POTENT SPECT RADIOLIGAND FOR THE DOPAMINE D2 RECEPTOR, The Journal of nuclear medicine, 35(5), 1994, pp. 160000199-160000199
Authors:
SCHMIDT DE
VOTAW JR
KESSLER RM
DEPAULIS T
Citation: De. Schmidt et al., AROMATIC AND AMINE SUBSTITUENT EFFECTS ON THE APPARENT LIPOPHILICITIES OF N-[(2-PYRROLIDINYL)METHYL]-SUBSTITUTED BENZAMIDES, Journal of pharmaceutical sciences, 83(3), 1994, pp. 305-315
Authors:
PHILLIPS ST
DEPAULIS T
BARON BM
SIEGEL BW
SEEMAN P
VANTOL HHM
GUAN HC
SMITH HE
Citation: St. Phillips et al., BINDING OF 5H-DIBENZO[B,E][1,4]DIAZEPINE AND CHIRAL 5H-DIBENZO[A,D]CYCLOHEPTENE ANALOGS OF CLOZAPINE TO DOPAMINE AND SEROTONIN RECEPTORS, Journal of medicinal chemistry, 37(17), 1994, pp. 2686-2696
Authors:
KESSLER RM
VOTAW JR
DEPAULIS T
BINGHAM DR
ANSARI MS
MASON NS
HOLBURN G
SCHMIDT DE
VOTAW DB
MANNING RG
EBERT MH
Citation: Rm. Kessler et al., EVALUATION OF 5-[F-18]FLUOROPROPYLEPIDEPRIDE AS A POTENTIAL PET RADIOLIGAND FOR IMAGING DOPAMINE D2 RECEPTORS, Synapse, 15(3), 1993, pp. 169-176
Citation: Jr. Votaw et al., FAILURE OF THE 3-COMPARTMENT MODEL TO DESCRIBE THE PHARMACOKINETICS IN BRAIN OF A HIGH-AFFINITY SUBSTITUTED BENZAMIDE, Synapse, 15(3), 1993, pp. 177-190
Authors:
KESSLER RM
MASON NS
VOTAW JR
ANSARI MS
DEPAULIS T
SCHMIDT DE
MANNING RG
Citation: Rm. Kessler et al., FACTORS UNDERLYING THE D-AMPHETAMINE INDUCED DISPLACEMENT OF DOPAMINED2 RADIOLIGANDS IN RHESUS-MONKEYS, The Journal of nuclear medicine, 34(5), 1993, pp. 132-132
Authors:
VOTAW JR
KESSLER RM
DEPAULIS T
ANSARI MS
MASON NS
SCHMIDT DE
MANNING RG
HOLBURN G
Citation: Jr. Votaw et al., QUANTIFICATION OF STRIATAL AND EXTRASTRIATAL DOPAMINE D2 RECEPTORS USING N-ALLYL-[18F]FPE, The Journal of nuclear medicine, 34(5), 1993, pp. 132-132
Authors:
KESSLER RM
DEPAULIS T
ANSARI MS
VOTAW JR
SCHMIDT DE
MANNING RG
Citation: Rm. Kessler et al., N-ALLYL-5-FLUOROPROPYLEPIDEPRIDE - A VERY POTENT AND SPECIFIC DOPAMINE-D2 PET RADIOLIGAND, The Journal of nuclear medicine, 34(5), 1993, pp. 202-202
Authors:
KESSLER RM
VOTAW JR
SCHMIDT DE
ANSARI MS
HOLDEMAN KP
DEPAULIS T
CLANTON JA
PFEFFER R
MANNING RG
EBERT MH
Citation: Rm. Kessler et al., HIGH-AFFINITY DOPAMINE D2 RECEPTOR RADIOLIGANDS .3. [I-123] AND [I-125] EPIDEPRIDE - INVIVO STUDIES IN RHESUS-MONKEY BRAIN AND COMPARISON WITH INVITRO PHARMACOKINETICS IN RAT-BRAIN, Life sciences, 53(3), 1993, pp. 241-250
Authors:
KESSLER RM
WHETSELL WO
ANSARI MS
VOTAW JR
DEPAULIS T
CLANTON JA
SCHMIDT DE
MASON NS
MANNING RG
Citation: Rm. Kessler et al., IDENTIFICATION OF EXTRASTRIATAL DOPAMINE D2 RECEPTORS IN POSTMORTEM HUMAN BRAIN WITH [I-125] EPIDEPRIDE, Brain research, 609(1-2), 1993, pp. 237-243