Authors:
DeVita, RJ
Walsh, TF
Young, JR
Jiang, JL
Ujjainwalla, F
Toupence, RB
Parikh, M
Huang, SX
Fair, JA
Goulet, MT
Wyvratt, MJ
Lo, JL
Ren, N
Yudkovitz, JB
Yang, YT
Cheng, K
Cui, JS
Mount, G
Rohrer, SP
Schaeffer, JM
Rhodes, L
Drisko, JE
McGowan, E
MacIntyre, DE
Vincent, S
Carlin, JR
Cameron, J
Smith, RG
Citation: Rj. Devita et al., A potent, nonpeptidyl 1H-quinolone antagonist for the gonadotropin-releasing hormone receptor, J MED CHEM, 44(6), 2001, pp. 917-922
Authors:
Young, JR
Huang, SX
Chen, I
Walsh, TF
DeVita, RJ
Wyvratt, MJ
Goulet, MT
Ren, N
Lo, J
Yang, YT
Yudkovitz, JB
Cheng, K
Smith, RG
Citation: Jr. Young et al., Quinolones as gonadotropin releasing hormone (GnRH) antagonists: Simultaneous optimization of the C(3)-aryl and C(6)-substituents, BIOORG MED, 10(15), 2000, pp. 1723-1727
Authors:
Cui, JS
Smith, RG
Mount, GR
Lo, JL
Yu, JH
Walsh, TF
Singh, SB
DeVita, RJ
Goulet, MT
Schaeffer, JM
Cheng, K
Citation: Js. Cui et al., Identification of Phe(313) of the gonadotropin-releasing hormone (GnRH) receptor as a site critical for the binding of nonpeptide GnRH antagonists, MOL ENDOCR, 14(5), 2000, pp. 671-681
Citation: Rj. Devita et al., Identification and initial structure-activity relationships of a novel non-peptide quinolone GnRH receptor antagonist, BIOORG MED, 9(17), 1999, pp. 2615-2620
Citation: Rj. Devita et al., Investigation of the 4-O-alkylamine substituent of non-peptide quinolone GnRH receptor antagonists, BIOORG MED, 9(17), 1999, pp. 2621-2624
Citation: Jl. Jiang et al., Asymmetric synthesis of chiral, nonracemic trifluoromethyl-substituted piperidines and decahydroquinolines, J AM CHEM S, 121(3), 1999, pp. 593-594