Authors: Sall, DJ Bailey, DL Bastian, JA Buben, JA Chirgadze, NY Clemens-Smith, AC Denney, ML Fisher, MJ Giera, DD Gifford-Moore, DS Harper, RW Johnson, LM Klimkowski, VJ Kohn, TJ Lin, HS McCowan, JR Palkowitz, AD Richett, ME Smith, GF Snyder, DW Takeuchi, K Toth, JE Zhang, MS

Citation: Dj. Sall et al., Diamino benzo[b]thiophene derivatives as a novel class of active site directed thrombin inhibitors. 5. Potency, efficacy, and pharmacokinetic properties of modified C-3 side chain derivatives, J MED CHEM, 43(4), 2000, pp. 649-663

Authors: Takeuchi, K Kohn, TJ Sall, DJ Denney, ML McCowan, JR Smith, GF Gifford-Moore, DS

Citation: K. Takeuchi et al., Dibasic benzo[b]thiophene derivatives as a novel class of active site directed thrombin inhibitors: 4. SAR studies on the conformationally restrictedC3-side chain of hydroxybenzo[b]thiophenes, BIOORG MED, 9(5), 1999, pp. 759-764

Authors: Zhang, MS Bailey, DL Bastian, JA Briggs, SL Chirgadze, NY Clawson, DK Denney, ML Gifford-Moore, DS Harper, RW Johnson, LM Klimkowski, VJ Kohn, TJ Lin, HS McCowan, JR Richett, ME Sall, DJ Smith, AJ Smith, GF Snyder, DW Takeuchi, K Utterback, BG Yan, SCB

Citation: Ms. Zhang et al., Dibasic benzo[b]thiophene derivatives as a novel class of active site directed thrombin inhibitors: 2. Sidechain optimization and demonstration of invivo efficacy, BIOORG MED, 9(5), 1999, pp. 775-780

Authors: Bastian, JA Chirgadze, N Denney, ML Gifford-Moore, DS Sall, DJ Smith, GF Wikel, JH

Citation: Ja. Bastian et al., Diamino benzo[b]thiophene derivatives as a novel class of active site directed thrombin inhibitors: 3. Enhancing activity by imposing conformational restriction in the C-4" side chain, BIOORG MED, 9(3), 1999, pp. 363-368