Authors:
Chu, V
Brown, K
Colussi, D
Gao, JB
Bostwick, J
Kasiewski, C
Bentley, R
Morgan, S
Guertin, K
Pauls, HW
Gong, Y
Zulli, A
Perrone, MH
Dunwiddie, CT
Leadley, RJ
Citation: V. Chu et al., Pharmacological characterization of a novel factor Xa inhibitor, FXV673, THROMB RES, 103(4), 2001, pp. 309-324
Authors:
Bostwick, JS
Bentley, R
Morgan, S
Brown, K
Chu, V
Ewing, WR
Spada, AP
Pauls, H
Perrone, MH
Dunwiddie, CT
Leadley, RJ
Citation: Js. Bostwick et al., RPR120844, a novel, specific inhibitor of coagulation factor Xa inhibits venous thrombosis in the rabbit, THROMB HAEM, 81(1), 1999, pp. 157-160
Authors:
Leadley, RJ
Morgan, SR
Bentley, R
Bostwick, JS
Kasiewski, CJ
Heran, C
Chu, W
Brown, K
Moxey, P
Ewing, WR
Pauls, H
Spada, AP
Perrone, MH
Dunwiddie, CT
Citation: Rj. Leadley et al., Pharmacodynamic activity and antithrombotic efficacy of RPR120844, a novelinhibitor of coagulation factor Xa, J CARDIO PH, 34(6), 1999, pp. 791-799
Authors:
Ewing, WR
Becker, MR
Manetta, VE
Davis, RS
Pauls, HW
Mason, H
Choi-Sledeski, YM
Green, D
Cha, D
Spada, AP
Cheney, DL
Mason, JS
Maignan, S
Guilloteau, JP
Brown, K
Colussi, D
Bentley, R
Bostwick, J
Kasiewski, CJ
Morgan, SR
Leadley, RJ
Dunwiddie, CT
Perrone, MH
Chu, V
Citation: Wr. Ewing et al., Design and structure-activity relationships of potent and selective inhibitors of blood coagulation factor Xa, J MED CHEM, 42(18), 1999, pp. 3557-3571
Authors:
Choi-Sledeski, YM
McGarry, DG
Green, DM
Mason, HJ
Becker, MR
Davis, RS
Ewing, WR
Dankulich, WP
Manetta, VE
Morris, RL
Spada, AP
Cheney, DL
Brown, KD
Colussi, DJ
Chu, V
Heran, CL
Morgan, SR
Bentley, RG
Leadley, RJ
Maignan, S
Guilloteau, JP
Dunwiddie, CT
Pauls, HW
Citation: Ym. Choi-sledeski et al., Sulfonamidopyrrolidinone factor Xa inhibitors: Potency and selectivity enhancements via P-1 and P-4 optimization, J MED CHEM, 42(18), 1999, pp. 3572-3587