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Showalter, HDH
Zhou, HR
Bridges, AJ
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Fry, DW
Nelson, JM
Sherwood, V
Vincent, PW
Roberts, BJ
Elliott, WL
Denny, WA
Citation: Jb. Smaill et al., Tyrosine kinase inhibitors. 18. 6-substituted 4-anilinoquinazolines and 4-anilinopyrido [3,4-d]pyrimidines as soluble, irreversible inhibitors of theepidermal growth factor receptor, J MED CHEM, 44(3), 2001, pp. 429-440
Authors:
Schroeder, MC
Hamby, JM
Connolly, CJC
Grohar, PJ
Winters, RT
Barvian, MR
Moore, CW
Boushelle, SL
Crean, SM
Kraker, AJ
Driscoll, DL
Vincent, PW
Elliott, WL
Lu, GH
Batley, BL
Dahring, TK
Major, TC
Panek, RL
Doherty, AM
Showalter, HDH
Citation: Mc. Schroeder et al., Soluble 2-substituted aminopyrido[2,3-d]pyrimidin-7-yl ureas. Structure-activity relationships against selected tyrosine kinases and exploration of in vitro and in vivo anticancer activity, J MED CHEM, 44(12), 2001, pp. 1915-1926
Authors:
Vincent, PW
Bridges, AJ
Dykes, DJ
Fry, DW
Leopold, WR
Patmore, SJ
Roberts, BJ
Rose, S
Sherwood, V
Zhou, HR
Elliott, WL
Citation: Pw. Vincent et al., Anticancer efficacy of the irreversible EGFr tyrosine kinase inhibitor PD 0169414 against human tumor xenografts, CANC CHEMOT, 45(3), 2000, pp. 231-238
Authors:
Thompson, AM
Connolly, CJC
Hamby, JM
Boushelle, S
Hartl, BG
Amar, AM
Kraker, AJ
Driscoll, DL
Steinkampf, RW
Patmore, SJ
Vincent, PW
Roberts, BJ
Elliott, WL
Klohs, W
Leopold, WR
Showalter, HDH
Denny, WA
Citation: Am. Thompson et al., 3-(3,5-dimethoxyphenyl)-1,6-naphthyridine-2,7-diamines and related 2-urea derivatives are potent and selective inhibitors of the FGF receptor-1 tyrosine kinase, J MED CHEM, 43(22), 2000, pp. 4200-4211
Authors:
Smaill, JB
Rewcastle, GW
Bridges, AJ
Zhou, HR
Showalter, HDH
Fry, DW
Nelson, JM
Sherwood, V
Elliott, WL
Vincent, PW
DeJohn, DE
Loo, JA
Greis, KD
Chan, OH
Reyner, EL
Lipka, E
Denny, WA
Citation: Jb. Smaill et al., Tyrosine kinase inhibitors. 17. Irreversible inhibitors of the epidermal growth factor receptor: 4-(phenylamino)quinazoline- and 4-(phenylamino)pyrido[3,2-d]-pyrimidine-6-acrylamides bearing additional solubilizing functions(vol 43, pg 1380, 2000), J MED CHEM, 43(16), 2000, pp. 3199-3199