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Results: 1-25/32
Authors:
Lee, A
Ellman, JA
Citation: A. Lee et Ja. Ellman, Parallel solution-phase synthesis of mechanism-based cysteine protease inhibitors, ORG LETT, 3(23), 2001, pp. 3707-3709
Authors:
Szewczyk, JW
Zuckerman, RL
Bergman, RG
Ellman, JA
Citation: Jw. Szewczyk et al., A mass spectrometric labeling strategy for high-throughput reaction evaluation and optimization: Exploring C-H activation, ANGEW CHEM, 40(1), 2001, pp. 216-219
Authors:
Borg, G
Chino, M
Ellman, JA
Citation: G. Borg et al., Asymmetric synthesis of pre-protected alpha,alpha-disubstituted amino acids from tert-butanesulfinyl ketimines, TETRAHEDR L, 42(8), 2001, pp. 1433-1436
Authors:
Souers, AJ
Ellman, JA
Citation: Aj. Souers et Ja. Ellman, beta-turn mimetic library synthesis: scaffolds and applications, TETRAHEDRON, 57(35), 2001, pp. 7431-7448
Authors:
Harris, JL
Niles, A
Burdick, K
Maffitt, M
Backes, BJ
Ellman, JA
Kuntz, I
Haak-Frendscho, M
Craik, CS
Citation: Jl. Harris et al., Definition of the extended substrate specificity determinants for beta-tryptases I and II, J BIOL CHEM, 276(37), 2001, pp. 34941-34947
Authors:
Souers, AJ
Owens, TD
Oliver, AG
Hollander, FJ
Ellman, JA
Citation: Aj. Souers et al., Synthesis and crystal structure of a unique and homochiral N,S-bonded N,N '-bis(tert-butanesulfinyl)amidinate rhodium(I) complex, INORG CHEM, 40(20), 2001, pp. 5299
Authors:
Owens, TD
Hollander, FJ
Oliver, AG
Ellman, JA
Citation: Td. Owens et al., Synthesis, utility, and structure of novel bis(sulfinyl)imidoamidine ligands for asymmetric Lewis acid catalysis, J AM CHEM S, 123(7), 2001, pp. 1539-1540
Authors:
Dragoli, DR
Burdett, MT
Ellman, JA
Citation: Dr. Dragoli et al., Design, synthesis, and utility of a support-bound tert-butanesulfinamide, J AM CHEM S, 123(41), 2001, pp. 10127-10128
Authors:
Thalji, RK
Ahrendt, KA
Bergman, RG
Ellman, JA
Citation: Rk. Thalji et al., Annulation of aromatic imines via directed C-H activation with Wilkinson'scatalyst, J AM CHEM S, 123(39), 2001, pp. 9692-9693
Authors:
Tan, KL
Bergman, RG
Ellman, JA
Citation: Kl. Tan et al., Annulation of alkenyl-substituted heterocycles via rhodium-catalyzed intramolecular C-H activated coupling reactions, J AM CHEM S, 123(11), 2001, pp. 2685-2686
Authors:
Backes, BJ
Harris, JL
Leonetti, F
Craik, CS
Ellman, JA
Citation: Bj. Backes et al., Synthesis of positional-scanning libraries of fluorogenic peptide substrates to define the extended substrate specificity of plasmin and thrombin (vol 18, pg 188, 2000), NAT BIOTECH, 18(5), 2000, pp. 559-559
Authors:
Backes, BJ
Harris, JL
Leonetti, F
Craik, CS
Ellman, JA
Citation: Bj. Backes et al., Synthesis of positional-scanning libraries of fluorogenic peptide substrates to define the extended substrate specificity of plasmin and thrombin, NAT BIOTECH, 18(2), 2000, pp. 187-193
Authors:
Souers, AJ
Rosenquist, A
Jarvie, EM
Ladlow, M
Feniuk, W
Ellman, JA
Citation: Aj. Souers et al., Optimization of a somatostatin mimetic via constrained amino acid and backbone incorporation, BIOORG MED, 10(24), 2000, pp. 2731-2733
Authors:
Maly, DJ
Choong, IC
Ellman, JA
Citation: Dj. Maly et al., Combinatorial target-guided ligand assembly: Identification of potent subtype-selective c-Src inhibitors, P NAS US, 97(6), 2000, pp. 2419-2424
Authors:
Harris, JL
Backes, BJ
Leonetti, F
Mahrus, S
Ellman, JA
Craik, CS
Citation: Jl. Harris et al., Rapid and general profiling of protease specificity by using combinatorialfluorogenic substrate libraries, P NAS US, 97(14), 2000, pp. 7754-7759
Authors:
Souers, AJ
Ellman, JA
Citation: Aj. Souers et Ja. Ellman, Asymmetric synthesis of a C-3 substituted pipecolic acid, J ORG CHEM, 65(4), 2000, pp. 1222-1224
Novel cathepsin D inhibitors block the formation of hyperphosphorylated tau fragments in hippocampus
Authors:
Bi, XN
Haque, TS
Zhou, J
Skillman, AG
Lin, B
Lee, CE
Kuntz, ID
Ellman, JA
Lynch, G
Citation: Xn. Bi et al., Novel cathepsin D inhibitors block the formation of hyperphosphorylated tau fragments in hippocampus, J NEUROCHEM, 74(4), 2000, pp. 1469-1477
Authors:
Dragoli, DR
Thompson, LA
O'Brien, J
Ellman, JA
Citation: Dr. Dragoli et al., Parallel synthesis of prostaglandin E-1 analogues, J COMB CHEM, 1(6), 1999, pp. 534-539
Authors:
Borg, G
Cogan, DA
Ellman, JA
Citation: G. Borg et al., One-pot asymmetric synthesis of tert-butanesulfinyl-protected amines from ketones by the in situ reduction of tert-butanesulfinyl ketimines, TETRAHEDR L, 40(37), 1999, pp. 6709-6712
Authors:
Souers, AJ
Schurer, S
Kwack, H
Virgilio, AA
Ellman, JA
Citation: Aj. Souers et al., Preparation of enantioenriched alpha-bromo acids incorporating diverse functionality, SYNTHESIS-S, (4), 1999, pp. 583-585
Authors:
Backes, BJ
Ellman, JA
Citation: Bj. Backes et Ja. Ellman, An alkanesulfonamide "safety-catch" linker for solid-phase synthesis, J ORG CHEM, 64(7), 1999, pp. 2322-2330
Authors:
Liu, GC
Cogan, DA
Owens, TD
Tang, TP
Ellman, JA
Citation: Gc. Liu et al., Synthesis of enantiomerically pure N-tert-butanesulfinyl imines (tert-butanesulfinimines) by the direct condensation of tert-butanesulfinamide with aldehydes and ketones, J ORG CHEM, 64(4), 1999, pp. 1278-1284
Authors:
Choong, IC
Ellman, JA
Citation: Ic. Choong et Ja. Ellman, Synthesis of alkoxylamines by alkoxide amination with 3,3 '-Di-tert-butyloxaziridine, J ORG CHEM, 64(18), 1999, pp. 6528-6529
Authors:
Backes, BJ
Dragoli, DR
Ellman, JA
Citation: Bj. Backes et al., Chiral N-acyl-tert-butanesulfinamides: The "safety-catch" principle applied to diastereoselective enolate alkylations, J ORG CHEM, 64(15), 1999, pp. 5472-5478
Authors:
Tang, TP
Ellman, JA
Citation: Tp. Tang et Ja. Ellman, The tert-butanesulfinyl group: An ideal chiral directing group and boc-surrogate for the asymmetric synthesis and applications of beta-amino acids, J ORG CHEM, 64(1), 1999, pp. 12-13