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Results: 1-11 |
Results: 11
Molecular modeling, structure-activity relationships and functional antagonism studies of 4-hydroxy-1-methyl-4-(4-methylphenyl)-3-piperidyl 4-methylphenyl ketones as a novel class of dopamine transporter inhibitors
Authors: Wang, SM Sakamuri, S Enyedy, IJ Kozikowski, AP Zaman, WA Johnson, KM
Citation: Sm. Wang et al., Molecular modeling, structure-activity relationships and functional antagonism studies of 4-hydroxy-1-methyl-4-(4-methylphenyl)-3-piperidyl 4-methylphenyl ketones as a novel class of dopamine transporter inhibitors, BIO MED CH, 9(7), 2001, pp. 1753-1764
Pharmacophore-based discovery of 3,4-disubstituted pyrrolidines as a novelglass of monoamine transporter inhibitors
Authors: Enyedy, IJ Zaman, WA Sakamuri, S Kozikowski, AP Johnson, KM Wang, SM
Citation: Ij. Enyedy et al., Pharmacophore-based discovery of 3,4-disubstituted pyrrolidines as a novelglass of monoamine transporter inhibitors, BIOORG MED, 11(9), 2001, pp. 1113-1118
Pharmacophore-based discovery, synthesis, and biological evaluation of 4-phenyl-1-arylalkyl piperidines as dopamine transporter inhibitors
Authors: Sakamuri, S Enyedy, IJ Kozikowski, AP Zaman, WA Johnson, KM Wang, SM
Citation: S. Sakamuri et al., Pharmacophore-based discovery, synthesis, and biological evaluation of 4-phenyl-1-arylalkyl piperidines as dopamine transporter inhibitors, BIOORG MED, 11(4), 2001, pp. 495-500
Synthesis and evaluation of the sunflower derived trypsin inhibitor as a potent inhibitor of the type II transmembrane serine protease, matriptase
Authors: Long, YQ Lee, SL Lin, CY Enyedy, IJ Wang, SM Li, P Dickson, RB Roller, PP
Citation: Yq. Long et al., Synthesis and evaluation of the sunflower derived trypsin inhibitor as a potent inhibitor of the type II transmembrane serine protease, matriptase, BIOORG MED, 11(18), 2001, pp. 2515-2519
Molecular dynamics study of active-site interactions with tetracoordinate transients in acetylcholinesterase and its mutants
Authors: Enyedy, IJ Kovach, IM Bencsura, A
Citation: Ij. Enyedy et al., Molecular dynamics study of active-site interactions with tetracoordinate transients in acetylcholinesterase and its mutants, BIOCHEM J, 353, 2001, pp. 645-653
Structure-based approach for the discovery of bis-benzamidines as novel inhibitors of matriptase
Authors: Enyedy, IJ Lee, SL Kuo, AH Dickson, RB Lin, CY Wang, SM
Citation: Ij. Enyedy et al., Structure-based approach for the discovery of bis-benzamidines as novel inhibitors of matriptase, J MED CHEM, 44(9), 2001, pp. 1349-1355
Discovery of small-molecule inhibitors of bcl-2 through structure-based computer screening
Authors: Enyedy, IJ Ling, Y Nacro, K Tomita, Y Wu, XH Cao, YY Guo, RB Li, BH Zhu, XF Huang, Y Long, YQ Roller, PP Yang, DJ Wang, SM
Citation: Ij. Enyedy et al., Discovery of small-molecule inhibitors of bcl-2 through structure-based computer screening, J MED CHEM, 44(25), 2001, pp. 4313-4324
Iridals are a novel class of ligands for phorbol ester receptors with modest selectivity for the RasGRP receptor subfamily
Authors: Shao, L Lewin, NE Lorenzo, PS Hu, ZJ Enyedy, IJ Garfield, SH Stone, JC Marner, FJ Blumberg, PM Wang, SM
Citation: L. Shao et al., Iridals are a novel class of ligands for phorbol ester receptors with modest selectivity for the RasGRP receptor subfamily, J MED CHEM, 44(23), 2001, pp. 3872-3880
Structural basis of binding of high-affinity ligands to protein kinase C: Prediction of the binding modes through a new molecular dynamics method andevaluation by site-directed mutagenesis
Authors: Pak, Y Enyedy, IJ Varady, J Kung, JW Lorenzo, PS Blumberg, PM Wang, SM
Citation: Y. Pak et al., Structural basis of binding of high-affinity ligands to protein kinase C: Prediction of the binding modes through a new molecular dynamics method andevaluation by site-directed mutagenesis, J MED CHEM, 44(11), 2001, pp. 1690-1701
Synthesis of 2-alkyl-3-aryl-substituted quinuclidines as novel dopamine transporter inhibitors
Authors: Sakamuri, S Enyedy, IJ Kozikowski, AP Wang, SM
Citation: S. Sakamuri et al., Synthesis of 2-alkyl-3-aryl-substituted quinuclidines as novel dopamine transporter inhibitors, TETRAHEDR L, 41(51), 2000, pp. 9949-9952
Discovery of a novel dopamine transporter inhibitor, 4-hydroxy-1-methyl-4-(4-methylphenyl)-3-piperidyl 4-methylphenyl ketone, as a potential cocaine antagonist through 3D-database pharmacophore searching. Molecular modeling,structure-activity relationships, and behavioral pharmacological studies
Authors: Wang, SM Sakamuri, S Enyedy, IJ Kozikowski, AP Deschaux, O Bandyopadhyay, BC Tella, SR Zaman, WA Johnson, KM
Citation: Sm. Wang et al., Discovery of a novel dopamine transporter inhibitor, 4-hydroxy-1-methyl-4-(4-methylphenyl)-3-piperidyl 4-methylphenyl ketone, as a potential cocaine antagonist through 3D-database pharmacophore searching. Molecular modeling,structure-activity relationships, and behavioral pharmacological studies, J MED CHEM, 43(3), 2000, pp. 351-360
Risultati: 1-11 |