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Results: 1-22 |
Results: 22

Authors: KUO MS BOCK MG FREIDINGER RM GUIDOTTI MT LIS EV PAWLUCZYK JM PERLOW DS PETTIBONE DJ QUIGLEY AG REISS DR WILLIAMS PD WOYDEN CJ
Citation: Ms. Kuo et al., NONPEPTIDE OXYTOCIN ANTAGONISTS - POTENT, ORALLY BIOAVAILABLE ANALOGSOF L-371,257 CONTAINING A 1-R-(PYRIDYL)ETHYL ETHER TERMINUS, Bioorganic & medicinal chemistry letters, 8(21), 1998, pp. 3081-3086

Authors: YANG LH BERK SC ROHRER SP MOSLEY RT GUO LQ UNDERWOOD DJ ARISON BH BIRZIN ET HAYES EC MITRA SW PARMAR RM CHENG K WU TJ BUTLER BS FOOR F PASTERNAK A PAN YP SILVA M FREIDINGER RM SMITH RG CHAPMAN K SCHAEFFER JM PATCHETT AA
Citation: Lh. Yang et al., SYNTHESIS AND BIOLOGICAL-ACTIVITIES OF POTENT PEPTIDOMIMETICS SELECTIVE FOR SOMATOSTATIN RECEPTOR SUBTYPE-2, Proceedings of the National Academy of Sciences of the United Statesof America, 95(18), 1998, pp. 10836-10841

Authors: BELL IM ERB JM FREIDINGER RM GALLICCHIO SN GUARE JP GUIDOTTI MT HALPIN RA HOBBS DW HOMNICK CF KUO MS LIS EV MATHRE DJ MICHELSON SR PAWLUCZYK JM PETTIBONE DJ REISS DR VICKERS S WILLIAMS PD WOYDEN CJ
Citation: Im. Bell et al., DEVELOPMENT OF ORALLY-ACTIVE OXYTOCIN ANTAGONISTS - STUDIES ON DIN-3-YLMETHYL)PIPERIDIN-4-YLOXY]-2-METHOXYBENZOYL IPERIDIN-4-YL)-1,4-DIHYDROBENZ[D][1,3]OXAZIN-2-ONE (L-372,662) AND RELATED PYRIDINES, Journal of medicinal chemistry, 41(12), 1998, pp. 2146-2163

Authors: LEWIS SD LUCAS BJ BRADY SF SISKO JT CUTRONA KJ SANDERSON PEJ FREIDINGER RM MAO SS GARDELL SJ SHAFER JA
Citation: Sd. Lewis et al., CHARACTERIZATION OF THE 2-STEP PATHWAY FOR INHIBITION OF THROMBIN BY ALPHA-KETOAMIDE TRANSITION-STATE ANALOGS, The Journal of biological chemistry, 273(9), 1998, pp. 4843-4854

Authors: LYLE TA CHEN ZG APPLEBY SD FREIDINGER RM GARDELL SJ LEWIS SD LI Y LYLE EA LYNCH JJ MULICHAK AM NG AS NAYLOROLSEN AM SANDERS WM
Citation: Ta. Lyle et al., SYNTHESIS, EVALUATION, AND CRYSTALLOGRAPHIC ANALYSIS OF L-371,912 - APOTENT AND SELECTIVE ACTIVE-SITE THROMBIN INHIBITOR, Bioorganic & medicinal chemistry letters, 7(1), 1997, pp. 67-72

Authors: PETTIBONE DJ FREIDINGER RM
Citation: Dj. Pettibone et Rm. Freidinger, DISCOVERY AND DEVELOPMENT OF NONPEPTIDE ANTAGONISTS OF PEPTIDE-HORMONE RECEPTORS, Biochemical Society transactions, 25(3), 1997, pp. 1051-1057

Authors: FREIDINGER RM PETTIBONE DJ
Citation: Rm. Freidinger et Dj. Pettibone, SMALL-MOLECULE LIGANDS FOR OXYTOCIN AND VASOPRESSIN RECEPTORS, Medicinal research reviews, 17(1), 1997, pp. 1-16

Authors: TUCKER TJ LUMMA WC MULICHAK AM CHEN ZG NAYLOROLSEN AM LEWIS SD LUCAS R FREIDINGER RM KUO LC
Citation: Tj. Tucker et al., DESIGN OF HIGHLY POTENT NONCOVALENT THROMBIN INHIBITORS THAT UTILIZE A NOVEL LIPOPHILIC BINDING POCKET IN THE THROMBIN ACTIVE-SITE, Journal of medicinal chemistry, 40(6), 1997, pp. 830-832

Authors: SELNICK HG LIVERTON NJ BALDWIN JJ BUTCHER JW CLAREMON DA ELLIOTT JM FREIDINGER RM KING SA LIBBY BE MCINTYRE CJ PRIBUSH DA REMY DC SMITH GR TEBBEN AJ JURKIEWICZ NK LYNCH JJ SALATA JJ SANGUINETTI MC SIEGL PKS SLAUGHTER DE VYAS K
Citation: Hg. Selnick et al., CLASS-III ANTIARRHYTHMIC ACTIVITY IN-VIVO BY SELECTIVE BLOCKADE OF THE SLOWLY ACTIVATING CARDIAC DELAYED RECTIFIER POTASSIUM CURRENT I-KS BY ,3-DIHYDRO-1H-BENZO[E][1,4]DIAZEPIN-3-YL]ACETAMIDE, Journal of medicinal chemistry, 40(24), 1997, pp. 3865-3868

Authors: FENG DM GARDELL SJ LEWIS SD BOCK MG CHEN ZG FREIDINGER RM NAYLOROLSEN AM RAMJIT HG WOLTMANN R BASKIN EP LYNCH JJ LUCAS R SHAFER JA DANCHECK KB CHEN IW MAO SS KRUEGER JA HARE TR MULICHAK AM VACCA JP
Citation: Dm. Feng et al., DISCOVERY OF A NOVEL, SELECTIVE, AND ORALLY BIOAVAILABLE CLASS OF THROMBIN INHIBITORS INCORPORATING AMINOPYRIDYL MOIETIES AT THE P1 POSITION, Journal of medicinal chemistry, 40(23), 1997, pp. 3726-3733

Authors: HOBBS DW GOULD NP HOFFMAN JB CLINESCHMIDT BV PETTIBONE DJ VEBER DF FREIDINGER RM
Citation: Dw. Hobbs et al., NONPEPTIDE OXYTOCIN ANTAGONISTS - IDENTIFICATION AND SYNTHESIS OF A POTENT CAMPHOR AMINOSUCCINIMIDE, Bioorganic & medicinal chemistry letters, 5(2), 1995, pp. 119-122

Authors: WILLIAMS PD CLINESCHMIDT BV ERB JM FREIDINGER RM GUIDOTTI MT LIS EV PAWLUCZYK JM PETTIBONE DJ REISS DR VEBER DF WOYDEN CJ
Citation: Pd. Williams et al., ENZOYL]PIPERIDIN-4-YL)-4H-3,1-BENZOXAZIN-2(1H)-ONE (L-371,257) - A NEW, ORALLY BIOAVAILABLE, NONPEPTIDE OXYTOCIN ANTAGONIST, Journal of medicinal chemistry, 38(23), 1995, pp. 4634-4636

Authors: BOCK MG DIPARDO RM MELLIN EC NEWTON RC VEBER DF FREEDMAN SB SMITH AJ PATEL S KEMP JA MARSHALL GR FLETCHER AE CHAPMAN KL ANDERSON PS FREIDINGER RM
Citation: Mg. Bock et al., 2ND-GENERATION BENZODIAZEPINE CCK-B ANTAGONISTS - DEVELOPMENT OF SUBNANOMOLAR ANALOGS WITH SELECTIVITY AND WATER SOLUBILITY, Journal of medicinal chemistry, 37(6), 1994, pp. 722-724

Authors: WILLIAMS PD ANDERSON PS BALL RG BOCK MG CARROLL L CHIU SHL CLINESCHMIDT BV CULBERSON JC ERB JM EVANS BE FITZPATRICK SL FREIDINGER RM KAUFMAN MJ LUNDELL GF MURPHY JS PAWLUCZYK JM PERLOW DS PETTIBONE DJ PITZENBERGER SM THOMPSON KL VEBER DF
Citation: Pd. Williams et al., )-YL)METHYL)SULFONYL)-4-(2-METHYLPHENYL)PIPERAZINE (L-368,899) - AN ORALLY BIOAVAILABLE, NONPEPTIDE OXYTOCIN ANTAGONIST WITH POTENTIAL UTILITY FOR MANAGING PRETERM LABOR, Journal of medicinal chemistry, 37(5), 1994, pp. 565-571

Authors: EVANS BE RITTLE KE CHANG RSL LOTTI VJ FREEDMAN SB FREIDINGER RM
Citation: Be. Evans et al., MULTIPURPOSE RECEPTOR LIGANDS - BETA-CARBOLINE CHOLECYSTOKININ ANTAGONISTS, Bioorganic & medicinal chemistry letters, 3(5), 1993, pp. 867-870

Authors: BOCK MG DIPARDO RM VEBER DF CHANG RSL LOTTI VJ FREEDMAN SB FREIDINGER RM
Citation: Mg. Bock et al., BENZOLACTAMS AS NONPEPTIDE CHOLECYSTOKININ RECEPTOR LIGANDS, Bioorganic & medicinal chemistry letters, 3(5), 1993, pp. 871-874

Authors: PETTIBONE DJ CLINESCHMIDT BV GUIDOTTI MT LIS EV REISS DR WOYDEN CJ BOCK MG EVANS BE FREIDINGER RM HOBBS DW VEBER DF WILLIAMS PD CHIU SHL THOMPSON KL SCHORN TW SIEGL PKS KAUFMAN MJ CUKIERSKI MA HALUSKA GJ COOK MJ NOVY MJ
Citation: Dj. Pettibone et al., L-368,899, A POTENT ORALLY-ACTIVE OXYTOCIN ANTAGONIST FOR POTENTIAL USE IN PRETERM LABOR, Drug development research, 30(3), 1993, pp. 129-142

Authors: PETTIBONE DJ CLINESCHMIDT BV BOCK MG EVANS BE FREIDINGER RM VEBER DF WILLIAMS PD
Citation: Dj. Pettibone et al., DEVELOPMENT AND PHARMACOLOGICAL ASSESSMENT OF NOVEL PEPTIDE AND NONPEPTIDE OXYTOCIN ANTAGONISTS, Regulatory peptides, 45(1-2), 1993, pp. 289-293

Authors: BRADY SF PALEVEDA WJ ARISON BH SAPERSTEIN R BRADY EJ RAYNOR K REISINE T VEBER DF FREIDINGER RM
Citation: Sf. Brady et al., APPROACHES TO PEPTIDOMIMETICS WHICH SERVE AS SURROGATES FOR THE CIS AMIDE BOND - NOVEL DISULFIDE-CONSTRAINED BICYCLIC HEXAPEPTIDE ANALOGS OF SOMATOSTATIN, Tetrahedron, 49(17), 1993, pp. 3449-3466

Authors: BOCK MG DIPARDO RM EVANS BE RITTLE KE WHITTER WL GARSKY VM GILBERT KF LEIGHTON JL CARSON KL MELLIN EC VEBER DF CHANG RSL LOTTI VJ FREEDMAN SB SMITH AJ PATEL S ANDERSON PS FREIDINGER RM
Citation: Mg. Bock et al., DEVELOPMENT OF 1,4-BENZODIAZEPINE CHOLECYSTOKININ TYPE-B ANTAGONISTS, Journal of medicinal chemistry, 36(26), 1993, pp. 4276-4292

Authors: EVANS BE LUNDELL GF GILBERT KF BOCK MG RITTLE KE CARROLL LA WILLIAMS PD PAWLUCZYK JM LEIGHTON JL YOUNG MB ERB JM HOBBS DW GOULD NP DIPARDO RM HOFFMAN JB PERLOW DS WHITTER WL VEBER DF PETTIBONE DJ CLINESCHMIDT BV ANDERSON PS FREIDINGER RM
Citation: Be. Evans et al., NANOMOLAR-AFFINITY, NONPEPTIDE OXYTOCIN RECEPTOR ANTAGONISTS, Journal of medicinal chemistry, 36(25), 1993, pp. 3993-4005

Authors: HIRSCHMANN R NICOLAOU KC PIETRANICO S LEAHY EM SALVINO J ARISON B CICHY MA SPOORS PG SHAKESPEARE WC SPRENGELER PA HAMLEY P SMITH AB REISINE T RAYNOR K MAECHLER L DONALDSON C VALE W FREIDINGER RM CASCIERI MR STRADER CD
Citation: R. Hirschmann et al., DE-NOVO DESIGN AND SYNTHESIS OF SOMATOSTATIN NONPEPTIDE PEPTIDOMIMETICS UTILIZING BETA-D-GLUCOSE AS A NOVEL SCAFFOLDING, Journal of the American Chemical Society, 115(26), 1993, pp. 12550-12568
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