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BUTLER BS
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SILVA M
FREIDINGER RM
SMITH RG
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SCHAEFFER JM
PATCHETT AA
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BELL IM
ERB JM
FREIDINGER RM
GALLICCHIO SN
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HALPIN RA
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PAWLUCZYK JM
PETTIBONE DJ
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Citation: Im. Bell et al., DEVELOPMENT OF ORALLY-ACTIVE OXYTOCIN ANTAGONISTS - STUDIES ON DIN-3-YLMETHYL)PIPERIDIN-4-YLOXY]-2-METHOXYBENZOYL IPERIDIN-4-YL)-1,4-DIHYDROBENZ[D][1,3]OXAZIN-2-ONE (L-372,662) AND RELATED PYRIDINES, Journal of medicinal chemistry, 41(12), 1998, pp. 2146-2163
Authors:
LEWIS SD
LUCAS BJ
BRADY SF
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CUTRONA KJ
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Citation: Sd. Lewis et al., CHARACTERIZATION OF THE 2-STEP PATHWAY FOR INHIBITION OF THROMBIN BY ALPHA-KETOAMIDE TRANSITION-STATE ANALOGS, The Journal of biological chemistry, 273(9), 1998, pp. 4843-4854
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Citation: Tj. Tucker et al., DESIGN OF HIGHLY POTENT NONCOVALENT THROMBIN INHIBITORS THAT UTILIZE A NOVEL LIPOPHILIC BINDING POCKET IN THE THROMBIN ACTIVE-SITE, Journal of medicinal chemistry, 40(6), 1997, pp. 830-832
Authors:
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SMITH GR
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SIEGL PKS
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Citation: Hg. Selnick et al., CLASS-III ANTIARRHYTHMIC ACTIVITY IN-VIVO BY SELECTIVE BLOCKADE OF THE SLOWLY ACTIVATING CARDIAC DELAYED RECTIFIER POTASSIUM CURRENT I-KS BY ,3-DIHYDRO-1H-BENZO[E][1,4]DIAZEPIN-3-YL]ACETAMIDE, Journal of medicinal chemistry, 40(24), 1997, pp. 3865-3868
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ERB JM
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Citation: Pd. Williams et al., ENZOYL]PIPERIDIN-4-YL)-4H-3,1-BENZOXAZIN-2(1H)-ONE (L-371,257) - A NEW, ORALLY BIOAVAILABLE, NONPEPTIDE OXYTOCIN ANTAGONIST, Journal of medicinal chemistry, 38(23), 1995, pp. 4634-4636
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Citation: Mg. Bock et al., 2ND-GENERATION BENZODIAZEPINE CCK-B ANTAGONISTS - DEVELOPMENT OF SUBNANOMOLAR ANALOGS WITH SELECTIVITY AND WATER SOLUBILITY, Journal of medicinal chemistry, 37(6), 1994, pp. 722-724
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Citation: Pd. Williams et al., )-YL)METHYL)SULFONYL)-4-(2-METHYLPHENYL)PIPERAZINE (L-368,899) - AN ORALLY BIOAVAILABLE, NONPEPTIDE OXYTOCIN ANTAGONIST WITH POTENTIAL UTILITY FOR MANAGING PRETERM LABOR, Journal of medicinal chemistry, 37(5), 1994, pp. 565-571
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CLINESCHMIDT BV
GUIDOTTI MT
LIS EV
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Citation: Dj. Pettibone et al., L-368,899, A POTENT ORALLY-ACTIVE OXYTOCIN ANTAGONIST FOR POTENTIAL USE IN PRETERM LABOR, Drug development research, 30(3), 1993, pp. 129-142
Authors:
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CLINESCHMIDT BV
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Citation: Sf. Brady et al., APPROACHES TO PEPTIDOMIMETICS WHICH SERVE AS SURROGATES FOR THE CIS AMIDE BOND - NOVEL DISULFIDE-CONSTRAINED BICYCLIC HEXAPEPTIDE ANALOGS OF SOMATOSTATIN, Tetrahedron, 49(17), 1993, pp. 3449-3466
Authors:
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VEBER DF
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Citation: Mg. Bock et al., DEVELOPMENT OF 1,4-BENZODIAZEPINE CHOLECYSTOKININ TYPE-B ANTAGONISTS, Journal of medicinal chemistry, 36(26), 1993, pp. 4276-4292
Authors:
EVANS BE
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GILBERT KF
BOCK MG
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DIPARDO RM
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CLINESCHMIDT BV
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FREIDINGER RM
Citation: Be. Evans et al., NANOMOLAR-AFFINITY, NONPEPTIDE OXYTOCIN RECEPTOR ANTAGONISTS, Journal of medicinal chemistry, 36(25), 1993, pp. 3993-4005
Authors:
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NICOLAOU KC
PIETRANICO S
LEAHY EM
SALVINO J
ARISON B
CICHY MA
SPOORS PG
SHAKESPEARE WC
SPRENGELER PA
HAMLEY P
SMITH AB
REISINE T
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DONALDSON C
VALE W
FREIDINGER RM
CASCIERI MR
STRADER CD
Citation: R. Hirschmann et al., DE-NOVO DESIGN AND SYNTHESIS OF SOMATOSTATIN NONPEPTIDE PEPTIDOMIMETICS UTILIZING BETA-D-GLUCOSE AS A NOVEL SCAFFOLDING, Journal of the American Chemical Society, 115(26), 1993, pp. 12550-12568