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Results: 1-11 |
Results: 11
UNIQUE PRECLINICAL CHARACTERISTICS OF GG745, A POTENT DUAL INHIBITOR OF 5AR
Authors: BRAMSON HN HERMANN D BATCHELOR KW LEE FW JAMES MK FRYE SV
Citation: Hn. Bramson et al., UNIQUE PRECLINICAL CHARACTERISTICS OF GG745, A POTENT DUAL INHIBITOR OF 5AR, The Journal of pharmacology and experimental therapeutics, 282(3), 1997, pp. 1496-1502
INHIBITION OF HUMAN STEROID 5-ALPHA REDUCTASES TYPE-I AND TYPE-II BY 6-AZA-STEROIDS - STRUCTURAL DETERMINANTS OF ONE-STEP VS 2-STEP MECHANISM
Authors: MOSS ML KUZMIC P STUART JD TIAN GC PERANTEAU AG FRYE SV KADWELL SH KOST TA OVERTON LK PATEL IR
Citation: Ml. Moss et al., INHIBITION OF HUMAN STEROID 5-ALPHA REDUCTASES TYPE-I AND TYPE-II BY 6-AZA-STEROIDS - STRUCTURAL DETERMINANTS OF ONE-STEP VS 2-STEP MECHANISM, Biochemistry, 35(11), 1996, pp. 3457-3464
STRUCTURE-ACTIVITY-RELATIONSHIPS FOR INHIBITION OF TYPE-1 AND 2 HUMAN5-ALPHA-REDUCTASE AND HUMAN ADRENAL 3-BETA-HYDROXY-DELTA(5)-STEROID DEHYDROGENASE 3-KETO-DELTA(5)-STEROID ISOMERASE BY 6-AZAANDROST-4-EN-3-ONES - OPTIMIZATION OF THE C17 SUBSTITUENT/
Authors: FRYE SV HAFFNER CD MALONEY PR HINER RN DORSEY GF NOE RA UNWALLA RJ BATCHELOR KW BRAMSON HN STUART JD SCHWEIKER SL VANAMOLD J BICKETT DM MOSS ML TIAN GC LEE FW TIPPIN TK JAMES MK GRIZZLE MK LONG JE CROOM DK
Citation: Sv. Frye et al., STRUCTURE-ACTIVITY-RELATIONSHIPS FOR INHIBITION OF TYPE-1 AND 2 HUMAN5-ALPHA-REDUCTASE AND HUMAN ADRENAL 3-BETA-HYDROXY-DELTA(5)-STEROID DEHYDROGENASE 3-KETO-DELTA(5)-STEROID ISOMERASE BY 6-AZAANDROST-4-EN-3-ONES - OPTIMIZATION OF THE C17 SUBSTITUENT/, Journal of medicinal chemistry, 38(14), 1995, pp. 2621-2627
MECHANISM OF TIME-DEPENDENT INHIBITION OF 5-ALPHA-REDUCTASES BY DELTA(1)-4-AZASTEROIDS - TOWARD PERFECTION OF RATES OF TIME-DEPENDENT INHIBITION BY USING LIGAND-BINDING ENERGIES
Authors: TIAN GC MOOK RA MOSS ML FRYE SV
Citation: Gc. Tian et al., MECHANISM OF TIME-DEPENDENT INHIBITION OF 5-ALPHA-REDUCTASES BY DELTA(1)-4-AZASTEROIDS - TOWARD PERFECTION OF RATES OF TIME-DEPENDENT INHIBITION BY USING LIGAND-BINDING ENERGIES, Biochemistry, 34(41), 1995, pp. 13453-13459
REDUCTION IN THE PROSTATE WEIGHT OF RATS BY A SERIES OF 6-AZASTEROID 5-ALPHA-REDUCTASE (5AR) INHIBITORS
Authors: GRIZZLE MK JAMES MK SCHUSTER SV LONG JE FRYE SV HAFFNER CD MALONEY PR MOOK RA DORSEY GF HINER RN
Citation: Mk. Grizzle et al., REDUCTION IN THE PROSTATE WEIGHT OF RATS BY A SERIES OF 6-AZASTEROID 5-ALPHA-REDUCTASE (5AR) INHIBITORS, The FASEB journal, 8(5), 1994, pp. 10000638-10000638
REDUCTION OF PROSTATIC DIHYDROTESTOSTERONE (DHT) IN RATS BY A SERIES OF 6-AZASTEROID 5-ALPHA REDUCTASE (5AR) INHIBITORS
Authors: JAMES MK GRIZZLE MK SCHUSTER SV LONG JE FRYE SV HAFFNER CD MALONEY PR MOOK RA DORSEY GF HINER RN
Citation: Mk. James et al., REDUCTION OF PROSTATIC DIHYDROTESTOSTERONE (DHT) IN RATS BY A SERIES OF 6-AZASTEROID 5-ALPHA REDUCTASE (5AR) INHIBITORS, The FASEB journal, 8(5), 1994, pp. 10000638-10000638
TIME-DEPENDENT INHIBITION OF RAT 5-ALPHA-REDUCTASE ISOZYMES 1 AND 2 BY 4-AZA-STEROID AND 6-AZA-STEROID
Authors: BATCHELOR KW STUART JD BRAMSON HN FRYE SV
Citation: Kw. Batchelor et al., TIME-DEPENDENT INHIBITION OF RAT 5-ALPHA-REDUCTASE ISOZYMES 1 AND 2 BY 4-AZA-STEROID AND 6-AZA-STEROID, Journal of cellular biochemistry, 1994, pp. 235-235
SLOW, TIGHT-BINDING INHIBITORS OF TYPE-II HUMAN STEROID 5-ALPHA-REDUCTASE
Authors: MOSS ML STUART JD KUZMIC P BRAMSON HN TIAN G MCGEEHAN J BATCHELOR KW FRYE SV WISEMAN JS
Citation: Ml. Moss et al., SLOW, TIGHT-BINDING INHIBITORS OF TYPE-II HUMAN STEROID 5-ALPHA-REDUCTASE, Journal of cellular biochemistry, 1994, pp. 238-238
6-AZASTEROIDS - STRUCTURE-ACTIVITY-RELATIONSHIPS FOR INHIBITION OF TYPE-1 AND TYPE-2 HUMAN 5-ALPHA-REDUCTASE AND HUMAN ADRENAL 3-BETA-HYDROXY-DELTA(5)-STEROID DEHYDROGENASE 3-KETO-DELTA(5)-STEROID ISOMERASE
Authors: FRYE SV HAFFNER CD MALONEY PR MOOK RA DORSEY GF HINER RN CRIBBS CM WHEELER TN RAY JA ANDREWS RC BATCHELOR KW BRAMSON HN STUART JD SCHWEIKER SL VANARNOLD J CROOM S BICKETT DM MOSS ML TIAN GC UNWALLA RJ LEE FW TIPPIN TK JAMES MK GRIZZLE MK LONG JE SCHUSTER SV
Citation: Sv. Frye et al., 6-AZASTEROIDS - STRUCTURE-ACTIVITY-RELATIONSHIPS FOR INHIBITION OF TYPE-1 AND TYPE-2 HUMAN 5-ALPHA-REDUCTASE AND HUMAN ADRENAL 3-BETA-HYDROXY-DELTA(5)-STEROID DEHYDROGENASE 3-KETO-DELTA(5)-STEROID ISOMERASE, Journal of medicinal chemistry, 37(15), 1994, pp. 2352-2360
BUTYLCARBAMOYL)-4-AZA-5-ALPHA-ANDROSTAN-1-EN-3-ONE IS AN ACTIVE-SITE-DIRECTED SLOW TIME-DEPENDENT INHIBITOR OF HUMAN STEROID 5-ALPHA-REDUCTASE-1
Authors: TIAN GC STUART JD MOSS ML DOMANICO PL BRAMSON HN PATEL IR KADWELL SH OVERTON LK KOST TA MOOK RA FRYE SV BATCHELOR KW WISEMAN JS
Citation: Gc. Tian et al., BUTYLCARBAMOYL)-4-AZA-5-ALPHA-ANDROSTAN-1-EN-3-ONE IS AN ACTIVE-SITE-DIRECTED SLOW TIME-DEPENDENT INHIBITOR OF HUMAN STEROID 5-ALPHA-REDUCTASE-1, Biochemistry, 33(8), 1994, pp. 2291-2296
6-AZASTEROIDS - POTENT DUAL INHIBITORS OF HUMAN TYPE-1 AND 2 STEROID 5-ALPHA-REDUCTASE
Authors: FRYE SV HAFFNER CD MALONEY PR MOOK RA HINER RN BATCHELOR KW BRAMSON HN STUART JD SCHWEIKER SL VANARNOLD J BICKETT DM MOSS ML TIAN GC UNWALLA RJ LEE FW TIPPIN TK JAMES MK GRIZZLE MK LONG JE SCHUSTER SV DORSEY GF
Citation: Sv. Frye et al., 6-AZASTEROIDS - POTENT DUAL INHIBITORS OF HUMAN TYPE-1 AND 2 STEROID 5-ALPHA-REDUCTASE, Journal of medicinal chemistry, 36(26), 1993, pp. 4313-4315
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