Authors:
CREGGE RJ
DURHAM SL
FARR RA
GALLION SL
HARE CM
HOFFMAN RV
JANUSZ MJ
KIM HO
KOEHL JR
MEHDI S
METZ WA
PEET NP
PELTON JT
SCHREUDER HA
SUNDER S
TARDIF C
Citation: Rj. Cregge et al., INHIBITION OF HUMAN NEUTROPHIL ELASTASE - 4 - DESIGN, SYNTHESIS, X-RAY CRYSTALLOGRAPHIC ANALYSIS, AND STRUCTURE-ACTIVITY-RELATIONSHIPS FOR A SERIES OF P-2-MODIFIED, ORALLY-ACTIVE PEPTIDYL PENTAFLUOROETHYL KETONES, Journal of medicinal chemistry, 41(14), 1998, pp. 2461-2480