AAAAAA

   
Results: 1-16 |
Results: 16
THE SELECTIVE 5-HT1B RECEPTOR INVERSE AGONIST TETRAHYDROSPIRO[FURO[2,3-F]INDOLE-3,4'-PIPERIDINE] (SB-224289) POTENTLY BLOCKS TERMINAL 5-HT AUTORECEPTOR FUNCTION BOTH IN-VITRO AND IN-VIVO
Authors: GASTER LM BLANEY FE DAVIES S DUCKWORTH DM HAM P JENKINS S JENNINGS AJ JOINER GF KING FD MULHOLLAND KR WYMAN PA HAGAN JJ HATCHER J JONES BJ MIDDLEMISS DN PRICE GW RILEY G ROBERTS C ROUTLEDGE C SELKIRK J SLADE PD
Citation: Lm. Gaster et al., THE SELECTIVE 5-HT1B RECEPTOR INVERSE AGONIST TETRAHYDROSPIRO[FURO[2,3-F]INDOLE-3,4'-PIPERIDINE] (SB-224289) POTENTLY BLOCKS TERMINAL 5-HT AUTORECEPTOR FUNCTION BOTH IN-VITRO AND IN-VIVO, Journal of medicinal chemistry, 41(8), 1998, pp. 1218-1235
SB-224289 - A NOVEL SELECTIVE (HUMAN) 5-HT1B RECEPTOR ANTAGONIST WITHNEGATIVE INTRINSIC ACTIVITY
Authors: SELKIRK JV SCOTT C HO M BURTON MJ WATSON J GASTER LM COLLIN L JONES BJ MIDDLEMISS DN PRICE GW
Citation: Jv. Selkirk et al., SB-224289 - A NOVEL SELECTIVE (HUMAN) 5-HT1B RECEPTOR ANTAGONIST WITHNEGATIVE INTRINSIC ACTIVITY, British Journal of Pharmacology, 125(1), 1998, pp. 202-208
SEROTONIN 5-HT3 AND 5-HT4 RECEPTOR ANTAGONISTS
Authors: GASTER LM KING FD
Citation: Lm. Gaster et Fd. King, SEROTONIN 5-HT3 AND 5-HT4 RECEPTOR ANTAGONISTS, Medicinal research reviews, 17(2), 1997, pp. 163-214
INCREASED DEFECATION CAUSED BY 5-HT4 RECEPTOR ACTIVATION IN THE MOUSE
Authors: BANNER SE SMITH MI BYWATER D GASTER LM SANGER GJ
Citation: Se. Banner et al., INCREASED DEFECATION CAUSED BY 5-HT4 RECEPTOR ACTIVATION IN THE MOUSE, European journal of pharmacology, 308(2), 1996, pp. 181-186
SELECTIVE AND FUNCTIONAL 5-HYDROXYTRYPTAMINE(4) RECEPTOR ANTAGONISM BY SB-207266
Authors: WARDLE KA BINGHAM S ELLIS ES GASTER LM RUSHANT B SMITH MI SANGER GJ
Citation: Ka. Wardle et al., SELECTIVE AND FUNCTIONAL 5-HYDROXYTRYPTAMINE(4) RECEPTOR ANTAGONISM BY SB-207266, British Journal of Pharmacology, 118(3), 1996, pp. 665-670
SB-207266 - THE FIRST POTENT AND SELECTIVE 5-HT4 RECEPTOR ANTAGONIST AMIDE WITH ORAL ACTIVITY
Authors: WARDLE KA BINGHAM S ELLIS ES GASTER LM RUSHANT B SMITH MI BROWN AM YOUNG TJ SANGER GJ
Citation: Ka. Wardle et al., SB-207266 - THE FIRST POTENT AND SELECTIVE 5-HT4 RECEPTOR ANTAGONIST AMIDE WITH ORAL ACTIVITY, British Journal of Pharmacology, 117, 1996, pp. 126-126
IHYDRO-2H-[1,3]OXAZINO[3,2-A]INDOLE-10-CARBOXAMIDE HYDROCHLORIDE - THE FIRST POTENT AND SELECTIVE 5-HT4 RECEPTOR ANTAGONIST AMIDE WITH ORALACTIVITY
Authors: GASTER LM JOINER GF KING FD WYMAN PA SUTTON JM BINGHAM S ELLIS ES SANGER GJ WARDLE KA
Citation: Lm. Gaster et al., IHYDRO-2H-[1,3]OXAZINO[3,2-A]INDOLE-10-CARBOXAMIDE HYDROCHLORIDE - THE FIRST POTENT AND SELECTIVE 5-HT4 RECEPTOR ANTAGONIST AMIDE WITH ORALACTIVITY, Journal of medicinal chemistry, 38(24), 1995, pp. 4760-4763
5-HT(4) RECEPTOR ANTAGONISTS - OXAZOLO, OXAZINO AND OXAZEPINO[3,2-A]INDOLE DERIVATIVES
Authors: GASTER LM WYMAN PA ELLIS ES BROWN AM YOUNG TJ
Citation: Lm. Gaster et al., 5-HT(4) RECEPTOR ANTAGONISTS - OXAZOLO, OXAZINO AND OXAZEPINO[3,2-A]INDOLE DERIVATIVES, Bioorganic & medicinal chemistry letters, 4(5), 1994, pp. 667-668
BLOCKADE OF HUMAN ATRIAL 5-HT4 RECEPTORS BY SB-207710, A SELECTIVE AND HIGH-AFFINITY 5-HT4 RECEPTOR ANTAGONIST
Authors: KAUMANN AJ GASTER LM KING FD BROWN AM
Citation: Aj. Kaumann et al., BLOCKADE OF HUMAN ATRIAL 5-HT4 RECEPTORS BY SB-207710, A SELECTIVE AND HIGH-AFFINITY 5-HT4 RECEPTOR ANTAGONIST, Naunyn-Schmiedeberg's archives of pharmacology, 349(5), 1994, pp. 546-548
TISSUE AND AGONIST-DEPENDENT NON-SURMOUNTABLE ANTAGONISM BY THE SELECTIVE 5-HT4 RECEPTOR ANTAGONIST SB-204070
Authors: BAXTER GS SANGER GJ GASTER LM WARDLE KA
Citation: Gs. Baxter et al., TISSUE AND AGONIST-DEPENDENT NON-SURMOUNTABLE ANTAGONISM BY THE SELECTIVE 5-HT4 RECEPTOR ANTAGONIST SB-204070, British Journal of Pharmacology, 112, 1994, pp. 210000055-210000055
THE EFFECTS OF SB-204070, A HIGHLY POTENT AND SELECTIVE 5-HT4 RECEPTOR ANTAGONIST, ON GUINEA-PIG DISTAL COLON
Authors: WARDLE KA ELLIS ES BAXTER GS KENNETT GA GASTER LM SANGER GJ
Citation: Ka. Wardle et al., THE EFFECTS OF SB-204070, A HIGHLY POTENT AND SELECTIVE 5-HT4 RECEPTOR ANTAGONIST, ON GUINEA-PIG DISTAL COLON, British Journal of Pharmacology, 112(3), 1994, pp. 789-794
SYNTHESIS OF NOVEL MODIFIED DIPEPTIDE INHIBITORS OF HUMAN COLLAGENASE- BETA-MERCAPTO CARBOXYLIC-ACID DERIVATIVES
Authors: BESZANT B BIRD J GASTER LM HARPER GP HUGHES I KARRAN EH MARKWELL RE MILESWILLIAMS AJ SMITH SA
Citation: B. Beszant et al., SYNTHESIS OF NOVEL MODIFIED DIPEPTIDE INHIBITORS OF HUMAN COLLAGENASE- BETA-MERCAPTO CARBOXYLIC-ACID DERIVATIVES, Journal of medicinal chemistry, 36(25), 1993, pp. 4030-4039
(1-BUTYL-4-PIPERIDINYL)METHYL 8-AMINO-7-CHLORO-1,4-BENZODIOXANE-5-CARBOXYLATE HYDROCHLORIDE - A HIGHLY POTENT AND SELECTIVE 5-HT4 RECEPTOR ANTAGONIST DERIVED FROM METOCLOPRAMIDE
Authors: GASTER LM JENNINGS AJ JOINER GF KING FD MULHOLLAND KR RAHMAN SK STARR S WYMAN PA WARDLE KA ELLIS ES SANGER GJ
Citation: Lm. Gaster et al., (1-BUTYL-4-PIPERIDINYL)METHYL 8-AMINO-7-CHLORO-1,4-BENZODIOXANE-5-CARBOXYLATE HYDROCHLORIDE - A HIGHLY POTENT AND SELECTIVE 5-HT4 RECEPTOR ANTAGONIST DERIVED FROM METOCLOPRAMIDE, Journal of medicinal chemistry, 36(25), 1993, pp. 4121-4123
)3-AMINO-6-CARBOXAMIDO-1,2,3,4-TETRAHYDROCARBAZOLE - A CONFORMATIONALLY RESTRICTED ANALOG OF 5-CARBOXAMIDOTRYPTAMINE WITH SELECTIVITY FOR THE SEROTONIN 5-HT1D RECEPTOR (VOL 36, PG 1919, 1993)
Authors: KING FD BROWN AM GASTER LM KAUMANN AJ MEDHURST AD PARKER SG PARSONS AA PATCH TL RAVAL P
Citation: Fd. King et al., )3-AMINO-6-CARBOXAMIDO-1,2,3,4-TETRAHYDROCARBAZOLE - A CONFORMATIONALLY RESTRICTED ANALOG OF 5-CARBOXAMIDOTRYPTAMINE WITH SELECTIVITY FOR THE SEROTONIN 5-HT1D RECEPTOR (VOL 36, PG 1919, 1993), Journal of medicinal chemistry, 36(21), 1993, pp. 3218-3218
(+ -) 3-AMINO-6-CARBOXAMIDO-1,2,3,4-TETRAHYDROCARBAZOLE - A CONFORMATIONALLY RESTRICTED ANALOG OF 5-CARBOXAMIDOTRYPTAMINE WITH SELECTIVITY FOR THE SEROTONIN 5-HT1D RECEPTOR/
Authors: KING FD BROWN AM GASTER LM KAUMANN AJ MEDHURST AD PARKER SG PARSONS AA PATCH TL RAVAL P
Citation: Fd. King et al., (+ -) 3-AMINO-6-CARBOXAMIDO-1,2,3,4-TETRAHYDROCARBAZOLE - A CONFORMATIONALLY RESTRICTED ANALOG OF 5-CARBOXAMIDOTRYPTAMINE WITH SELECTIVITY FOR THE SEROTONIN 5-HT1D RECEPTOR/, Journal of medicinal chemistry, 36(13), 1993, pp. 1918-1919
SB-204070 - A HIGHLY POTENT AND SELECTIVE 5-HT4 RECEPTOR ANTAGONIST
Authors: WARDLE KA ELLIS ES GASTER LM KING FD SANGER GJ
Citation: Ka. Wardle et al., SB-204070 - A HIGHLY POTENT AND SELECTIVE 5-HT4 RECEPTOR ANTAGONIST, British Journal of Pharmacology, 110, 1993, pp. 160000015-160000015
Risultati: 1-16 |