AAAAAA

   
Results: 1-14 |
Results: 14
2,2'-DITHIOBISBENZAMIDES DERIVED FROM ALPHA-AMINO-ACIDS, BETA-AMINO-ACIDS AND GAMMA-AMINO-ACIDS POSSESSING ANTI-HIV ACTIVITIES - SYNTHESIS AND STRUCTURE-ACTIVITY RELATIONSHIP
Authors: PRASAD JVNV LOO JA BOYER FE STIER MA GOGLIOTTI RD TURNER WJ HARVEY PJ KRAMER MR MACK DP SCHOLTEN JD GRACHECK SJ DOMAGALA JM
Citation: Jvnv. Prasad et al., 2,2'-DITHIOBISBENZAMIDES DERIVED FROM ALPHA-AMINO-ACIDS, BETA-AMINO-ACIDS AND GAMMA-AMINO-ACIDS POSSESSING ANTI-HIV ACTIVITIES - SYNTHESIS AND STRUCTURE-ACTIVITY RELATIONSHIP, Bioorganic & medicinal chemistry, 6(10), 1998, pp. 1707-1730
IN-VITRO ACTIVITY OF CLINAFLOXACIN, TROVAFLOXACIN, AND CIPROFLOXACIN
Authors: COHEN MA HUBAND MD GAGE JW YODER SL ROLAND GE GRACHECK SJ
Citation: Ma. Cohen et al., IN-VITRO ACTIVITY OF CLINAFLOXACIN, TROVAFLOXACIN, AND CIPROFLOXACIN, Journal of antimicrobial chemotherapy, 40(2), 1997, pp. 205-211
SYNTHESIS OF 5,6-DIHYDRO-4-HYDROXY-2-PYRONES AS HIV-1 PROTEASE INHIBITORS - THE PROFOUND EFFECT OF POLARITY ON ANTIVIRAL ACTIVITY
Authors: HAGEN SE PRASAD JVNV BOYER FE DOMAGALA JM ELLSWORTH EL GAJDA C HAMILTON HW MARKOSKI LJ STEINBAUGH BA TAIT BD LUNNEY EA TUMMINO PJ FERGUSON D HUPE D NOUHAN C GRACHECK SJ SAUNDERS JM VANDERROEST S
Citation: Se. Hagen et al., SYNTHESIS OF 5,6-DIHYDRO-4-HYDROXY-2-PYRONES AS HIV-1 PROTEASE INHIBITORS - THE PROFOUND EFFECT OF POLARITY ON ANTIVIRAL ACTIVITY, Journal of medicinal chemistry, 40(23), 1997, pp. 3707-3711
4-HYDROXY-5,6-DIHYDROPYRONES .2. POTENT NONPEPTIDE INHIBITORS OF HIV PROTEASE
Authors: TAIT BD HAGEN S DOMAGALA J ELLSWORTH EL GAJDA C HAMILTON HW PRASAD JVNV FERGUSON D GRAHAM N HUPE D NOUHAN C TUMMINO PJ HUMBLET C LUNNEY EA PAVLOVSKY A RUBIN J GRACHECK SJ BALDWIN ET BHAT TN ERICKSON JW GULNIK SV LIU BS
Citation: Bd. Tait et al., 4-HYDROXY-5,6-DIHYDROPYRONES .2. POTENT NONPEPTIDE INHIBITORS OF HIV PROTEASE, Journal of medicinal chemistry, 40(23), 1997, pp. 3781-3792
STRUCTURE-ACTIVITY-RELATIONSHIPS OF QUINOLONE AGENTS AGAINST MYCOBACTERIA - EFFECT OF STRUCTURAL MODIFICATIONS AT THE 8-POSITION
Authors: RENAU TE GAGE JW DEVER JA ROLAND GE JOANNIDES ET SHAPIRO MA SANCHEZ JP GRACHECK SJ DOMAGALA JM JACOBS MR REYNOLDS RC
Citation: Te. Renau et al., STRUCTURE-ACTIVITY-RELATIONSHIPS OF QUINOLONE AGENTS AGAINST MYCOBACTERIA - EFFECT OF STRUCTURAL MODIFICATIONS AT THE 8-POSITION, Antimicrobial agents and chemotherapy, 40(10), 1996, pp. 2363-2368
STRUCTURE-ACTIVITY-RELATIONSHIPS OF THE QUINOLONE ANTIBACTERIALS AGAINST MYCOBACTERIA - EFFECT OF STRUCTURAL-CHANGES AT N-1 AND C-7
Authors: RENAU TE SANCHEZ JP GAGE JW DEVER JA SHAPIRO MA GRACHECK SJ DOMAGALA JM
Citation: Te. Renau et al., STRUCTURE-ACTIVITY-RELATIONSHIPS OF THE QUINOLONE ANTIBACTERIALS AGAINST MYCOBACTERIA - EFFECT OF STRUCTURAL-CHANGES AT N-1 AND C-7, Journal of medicinal chemistry, 39(3), 1996, pp. 729-735
NONPEPTIDIC HIV PROTEASE INHIBITORS - 4-HYDROXY-PYRAN-2-ONE INHIBITORS WITH FUNCTIONAL TETHERS TO P-1 PHENYL RING TO REACH S-3 POCKET OF THE ENZYME
Authors: PRASAD JVNV TUMMINO PJ FERGUSON D SAUNDERS J VANDERROEST S MCQUADE TJ HELDSINGER A REYNER EL STEWART BH GUTTENDORF RJ PARA KS LUNNEY EA GRACHECK SJ DOMAGALA JM
Citation: Jvnv. Prasad et al., NONPEPTIDIC HIV PROTEASE INHIBITORS - 4-HYDROXY-PYRAN-2-ONE INHIBITORS WITH FUNCTIONAL TETHERS TO P-1 PHENYL RING TO REACH S-3 POCKET OF THE ENZYME, Biochemical and biophysical research communications, 221(3), 1996, pp. 815-820
COMPOUNDS THAT TARGET NOVEL CELLULAR-COMPONENTS INVOLVED IN HIV-1 TRANSCRIPTION
Authors: BUTERA ST ROBERTS BD CRITCHFIELD JW FANG G MCQUADE T GRACHECK SJ FOLKS TM
Citation: St. Butera et al., COMPOUNDS THAT TARGET NOVEL CELLULAR-COMPONENTS INVOLVED IN HIV-1 TRANSCRIPTION, Molecular medicine, 1(7), 1995, pp. 758-767
NONPEPTIDIC POTENT HIV-1 PROTEASE INHIBITORS - -HYDROXY-6-PHENYL-2-OXO-2H-PYRAN-3-YL)THIOMETHANES THAT SPAN P-1-P-2' SUBSITES IN A UNIQUE MODE OF ACTIVE-SITE BINDING
Authors: PRASAD JVN PARA KS TUMMINO PJ FERGUSON D MCQUADE TJ LUNNEY EA RAPUNDALO ST BATLEY BL HINGORANI G DOMAGALA JM GRACHECK SJ BHAT TN LIU BS BALDWIN ET ERICKSON JW SAWYER TK
Citation: Jvn. Prasad et al., NONPEPTIDIC POTENT HIV-1 PROTEASE INHIBITORS - -HYDROXY-6-PHENYL-2-OXO-2H-PYRAN-3-YL)THIOMETHANES THAT SPAN P-1-P-2' SUBSITES IN A UNIQUE MODE OF ACTIVE-SITE BINDING, Journal of medicinal chemistry, 38(6), 1995, pp. 898-905
THE SYNTHESIS, STRUCTURE-ACTIVITY, AND STRUCTURE-SIDE EFFECT RELATIONSHIPS OF A SERIES OF 8-ALKOXYQUINOLONE AND 5-AMINO-8-ALKOXYQUINOLONE ANTIBACTERIAL AGENTS
Authors: SANCHEZ JP GOGLIOTTI RD DOMAGALA JM GRACHECK SJ HUBAND MD SESNIE JA COHEN MA SHAPIRO MA
Citation: Jp. Sanchez et al., THE SYNTHESIS, STRUCTURE-ACTIVITY, AND STRUCTURE-SIDE EFFECT RELATIONSHIPS OF A SERIES OF 8-ALKOXYQUINOLONE AND 5-AMINO-8-ALKOXYQUINOLONE ANTIBACTERIAL AGENTS, Journal of medicinal chemistry, 38(22), 1995, pp. 4478-4487
EFFECT OF LIPOPHILICITY AT N-1 ON ACTIVITY OF FLUOROQUINOLONES AGAINST MYCOBACTERIA
Authors: RENAU TE SANCHEZ JP SHAPIRO MA DEVER JA GRACHECK SJ DOMAGALA JM
Citation: Te. Renau et al., EFFECT OF LIPOPHILICITY AT N-1 ON ACTIVITY OF FLUOROQUINOLONES AGAINST MYCOBACTERIA, Journal of medicinal chemistry, 38(15), 1995, pp. 2974-2977
GENETIC-RELATIONSHIP BETWEEN SOXRS AND MAR LOCI IN PROMOTING MULTIPLEANTIBIOTIC-RESISTANCE IN ESCHERICHIA-COLI
Authors: MILLER PF GAMBINO LF SULAVIK MC GRACHECK SJ
Citation: Pf. Miller et al., GENETIC-RELATIONSHIP BETWEEN SOXRS AND MAR LOCI IN PROMOTING MULTIPLEANTIBIOTIC-RESISTANCE IN ESCHERICHIA-COLI, Antimicrobial agents and chemotherapy, 38(8), 1994, pp. 1773-1779
SYNTHESIS AND ANTIBACTERIAL ACTIVITY OF NEW QUINOLONES CONTAINING A 7-[3-(1-AMINO-1-METHYLETHYL)-1-PYRROLIDINYL] MOIETY - GRAM-POSITIVE AGENTS WITH EXCELLENT ORAL ACTIVITY AND LOW SIDE-EFFECT POTENTIAL
Authors: HAGEN SE DOMAGALA JM GRACHECK SJ SESNIE JA STIER MA SUTO MJ
Citation: Se. Hagen et al., SYNTHESIS AND ANTIBACTERIAL ACTIVITY OF NEW QUINOLONES CONTAINING A 7-[3-(1-AMINO-1-METHYLETHYL)-1-PYRROLIDINYL] MOIETY - GRAM-POSITIVE AGENTS WITH EXCELLENT ORAL ACTIVITY AND LOW SIDE-EFFECT POTENTIAL, Journal of medicinal chemistry, 37(6), 1994, pp. 733-738
OVEREXPRESSION OF THE MARA POSITIVE REGULATOR IS SUFFICIENT TO CONFERMULTIPLE ANTIBIOTIC-RESISTANCE IN ESCHERICHIA-COLI
Authors: GAMBINO L GRACHECK SJ MILLER PF
Citation: L. Gambino et al., OVEREXPRESSION OF THE MARA POSITIVE REGULATOR IS SUFFICIENT TO CONFERMULTIPLE ANTIBIOTIC-RESISTANCE IN ESCHERICHIA-COLI, Journal of bacteriology, 175(10), 1993, pp. 2888-2894
Risultati: 1-14 |