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Results: 1-12 |
Results: 12
OPTIMIZATION OF 3-(1H-INDAZOL-3-YLMETHYL)-1,5-BENZODIAZEPINES AS POTENT, ORALLY-ACTIVE CCK-A AGONISTS
Authors: HENKE BR AQUINO CJ BIRKEMO LS CROOM DK DOUGHERTY RW ERVIN GN GRIZZLE MK HIRST GC JAMES MK JOHNSON MF QUEEN KL SHERRILL RG SUGG EE SUH EM SZEWCZYK JW UNWALLA RJ YINGLING J WILLSON TM
Citation: Br. Henke et al., OPTIMIZATION OF 3-(1H-INDAZOL-3-YLMETHYL)-1,5-BENZODIAZEPINES AS POTENT, ORALLY-ACTIVE CCK-A AGONISTS, Journal of medicinal chemistry, 40(17), 1997, pp. 2706-2725
DISCOVERY OF 1,5-BENZODIAZEPINES WITH PERIPHERAL CHOLECYSTOKININ (CCK-A) RECEPTOR AGONIST ACTIVITY .2. OPTIMIZATION OF THE C3 AMINO SUBSTITUENT
Authors: HIRST GC AQUINO C BIRKEMO L CROOM DK DEZUBE M DOUGHERTY RW ERVIN GN GRIZZLE MK HENKE B JAMES MK JOHNSON MF MOMTAHEN T QUEEN KL SHERRILL RG SZEWCZYK J WILLSON TM SUGG EE
Citation: Gc. Hirst et al., DISCOVERY OF 1,5-BENZODIAZEPINES WITH PERIPHERAL CHOLECYSTOKININ (CCK-A) RECEPTOR AGONIST ACTIVITY .2. OPTIMIZATION OF THE C3 AMINO SUBSTITUENT, Journal of medicinal chemistry, 39(26), 1996, pp. 5236-5245
DISCOVERY OF 1,5-BENZODIAZEPINES WITH PERIPHERAL CHOLECYSTOKININ (CCK-A) RECEPTOR AGONIST ACTIVITY .1. OPTIMIZATION OF THE AGONIST TRIGGER
Authors: AQUINO CJ ARMOUR DR BERMAN JM BIRKEMO LS CARR RAE CROOM DK DEZUBE M DOUGHERTY RW ERVIN GN GRIZZLE MK HEAD JE HIRST GC JAMES MK JOHNSON MF MILLER LJ QUEEN KL RIMELE TJ SMITH DN SUGG EE
Citation: Cj. Aquino et al., DISCOVERY OF 1,5-BENZODIAZEPINES WITH PERIPHERAL CHOLECYSTOKININ (CCK-A) RECEPTOR AGONIST ACTIVITY .1. OPTIMIZATION OF THE AGONIST TRIGGER, Journal of medicinal chemistry, 39(2), 1996, pp. 562-569
3-[2-(N-PHENYLACETAMIDE)]-1,5-BENZODIAZEPINES - ORALLY-ACTIVE, BINDING SELECTIVE CCK-A AGONISTS
Authors: WILLSON TM HENKE BR MOMTAHEN TM MYERS PL SUGG EE UNWALLA RJ CROOM DK DOUGHERTY RW GRIZZLE MK JOHNSON MF QUEEN KL RIMELE TJ YINGLING JD JAMES MK
Citation: Tm. Willson et al., 3-[2-(N-PHENYLACETAMIDE)]-1,5-BENZODIAZEPINES - ORALLY-ACTIVE, BINDING SELECTIVE CCK-A AGONISTS, Journal of medicinal chemistry, 39(15), 1996, pp. 3030-3034
3-(1H-INDAZOL-3-YLMETHYL)-1,5-BENZODIAZEPINES - CCK-A AGONISTS THAT DEMONSTRATE ORAL ACTIVITY AS SATIETY AGENTS
Authors: HENKE BR WILLSON TM SUGG EE CROOM DK DOUGHERTY RW QUEEN KL BIRKEMO LS ERVIN GN GRIZZLE MK JOHNSON MF JAMES MK
Citation: Br. Henke et al., 3-(1H-INDAZOL-3-YLMETHYL)-1,5-BENZODIAZEPINES - CCK-A AGONISTS THAT DEMONSTRATE ORAL ACTIVITY AS SATIETY AGENTS, Journal of medicinal chemistry, 39(14), 1996, pp. 2655-2658
MODIFICATION OF RECEPTOR SELECTIVITY AND FUNCTIONAL-ACTIVITY IN CHOLECYSTOKININ PEPTOID LIGANDS
Authors: DEZUBE M SUGG EE BIRKEMO LS CROOM DK DOUGHERTY RW ERVIN GN GRIZZLE MK JAMES MK JOHNSON MF MOSHER JT QUEEN KL RIMELE TJ SAULS HR TRIANTAFILLOU JA
Citation: M. Dezube et al., MODIFICATION OF RECEPTOR SELECTIVITY AND FUNCTIONAL-ACTIVITY IN CHOLECYSTOKININ PEPTOID LIGANDS, Journal of medicinal chemistry, 38(17), 1995, pp. 3384-3390
STRUCTURE-ACTIVITY-RELATIONSHIPS FOR INHIBITION OF TYPE-1 AND 2 HUMAN5-ALPHA-REDUCTASE AND HUMAN ADRENAL 3-BETA-HYDROXY-DELTA(5)-STEROID DEHYDROGENASE 3-KETO-DELTA(5)-STEROID ISOMERASE BY 6-AZAANDROST-4-EN-3-ONES - OPTIMIZATION OF THE C17 SUBSTITUENT/
Authors: FRYE SV HAFFNER CD MALONEY PR HINER RN DORSEY GF NOE RA UNWALLA RJ BATCHELOR KW BRAMSON HN STUART JD SCHWEIKER SL VANAMOLD J BICKETT DM MOSS ML TIAN GC LEE FW TIPPIN TK JAMES MK GRIZZLE MK LONG JE CROOM DK
Citation: Sv. Frye et al., STRUCTURE-ACTIVITY-RELATIONSHIPS FOR INHIBITION OF TYPE-1 AND 2 HUMAN5-ALPHA-REDUCTASE AND HUMAN ADRENAL 3-BETA-HYDROXY-DELTA(5)-STEROID DEHYDROGENASE 3-KETO-DELTA(5)-STEROID ISOMERASE BY 6-AZAANDROST-4-EN-3-ONES - OPTIMIZATION OF THE C17 SUBSTITUENT/, Journal of medicinal chemistry, 38(14), 1995, pp. 2621-2627
REDUCTION OF PROSTATIC DIHYDROTESTOSTERONE (DHT) IN RATS BY A SERIES OF 6-AZASTEROID 5-ALPHA REDUCTASE (5AR) INHIBITORS
Authors: JAMES MK GRIZZLE MK SCHUSTER SV LONG JE FRYE SV HAFFNER CD MALONEY PR MOOK RA DORSEY GF HINER RN
Citation: Mk. James et al., REDUCTION OF PROSTATIC DIHYDROTESTOSTERONE (DHT) IN RATS BY A SERIES OF 6-AZASTEROID 5-ALPHA REDUCTASE (5AR) INHIBITORS, The FASEB journal, 8(5), 1994, pp. 10000638-10000638
REDUCTION IN THE PROSTATE WEIGHT OF RATS BY A SERIES OF 6-AZASTEROID 5-ALPHA-REDUCTASE (5AR) INHIBITORS
Authors: GRIZZLE MK JAMES MK SCHUSTER SV LONG JE FRYE SV HAFFNER CD MALONEY PR MOOK RA DORSEY GF HINER RN
Citation: Mk. Grizzle et al., REDUCTION IN THE PROSTATE WEIGHT OF RATS BY A SERIES OF 6-AZASTEROID 5-ALPHA-REDUCTASE (5AR) INHIBITORS, The FASEB journal, 8(5), 1994, pp. 10000638-10000638
6-AZASTEROIDS - STRUCTURE-ACTIVITY-RELATIONSHIPS FOR INHIBITION OF TYPE-1 AND TYPE-2 HUMAN 5-ALPHA-REDUCTASE AND HUMAN ADRENAL 3-BETA-HYDROXY-DELTA(5)-STEROID DEHYDROGENASE 3-KETO-DELTA(5)-STEROID ISOMERASE
Authors: FRYE SV HAFFNER CD MALONEY PR MOOK RA DORSEY GF HINER RN CRIBBS CM WHEELER TN RAY JA ANDREWS RC BATCHELOR KW BRAMSON HN STUART JD SCHWEIKER SL VANARNOLD J CROOM S BICKETT DM MOSS ML TIAN GC UNWALLA RJ LEE FW TIPPIN TK JAMES MK GRIZZLE MK LONG JE SCHUSTER SV
Citation: Sv. Frye et al., 6-AZASTEROIDS - STRUCTURE-ACTIVITY-RELATIONSHIPS FOR INHIBITION OF TYPE-1 AND TYPE-2 HUMAN 5-ALPHA-REDUCTASE AND HUMAN ADRENAL 3-BETA-HYDROXY-DELTA(5)-STEROID DEHYDROGENASE 3-KETO-DELTA(5)-STEROID ISOMERASE, Journal of medicinal chemistry, 37(15), 1994, pp. 2352-2360
THE INOTROPIC AND BETA-BLOCKING EFFECTS OF A CHIMERIC MOLECULE THAT PUTATIVELY INHIBITS BOTH TYPE-III PHOSPHODIESTERASE AND BETA-ADRENOCEPTORS IN ANESTHETIZED DOGS
Authors: SHAFFER JE GRIZZLE MK ANDERSON DK WHEELER TN
Citation: Je. Shaffer et al., THE INOTROPIC AND BETA-BLOCKING EFFECTS OF A CHIMERIC MOLECULE THAT PUTATIVELY INHIBITS BOTH TYPE-III PHOSPHODIESTERASE AND BETA-ADRENOCEPTORS IN ANESTHETIZED DOGS, The Journal of pharmacology and experimental therapeutics, 265(3), 1993, pp. 1105-1112
6-AZASTEROIDS - POTENT DUAL INHIBITORS OF HUMAN TYPE-1 AND 2 STEROID 5-ALPHA-REDUCTASE
Authors: FRYE SV HAFFNER CD MALONEY PR MOOK RA HINER RN BATCHELOR KW BRAMSON HN STUART JD SCHWEIKER SL VANARNOLD J BICKETT DM MOSS ML TIAN GC UNWALLA RJ LEE FW TIPPIN TK JAMES MK GRIZZLE MK LONG JE SCHUSTER SV DORSEY GF
Citation: Sv. Frye et al., 6-AZASTEROIDS - POTENT DUAL INHIBITORS OF HUMAN TYPE-1 AND 2 STEROID 5-ALPHA-REDUCTASE, Journal of medicinal chemistry, 36(26), 1993, pp. 4313-4315
Risultati: 1-12 |