Authors:
HENKE BR
AQUINO CJ
BIRKEMO LS
CROOM DK
DOUGHERTY RW
ERVIN GN
GRIZZLE MK
HIRST GC
JAMES MK
JOHNSON MF
QUEEN KL
SHERRILL RG
SUGG EE
SUH EM
SZEWCZYK JW
UNWALLA RJ
YINGLING J
WILLSON TM
Citation: Br. Henke et al., OPTIMIZATION OF 3-(1H-INDAZOL-3-YLMETHYL)-1,5-BENZODIAZEPINES AS POTENT, ORALLY-ACTIVE CCK-A AGONISTS, Journal of medicinal chemistry, 40(17), 1997, pp. 2706-2725
Authors:
HIRST GC
AQUINO C
BIRKEMO L
CROOM DK
DEZUBE M
DOUGHERTY RW
ERVIN GN
GRIZZLE MK
HENKE B
JAMES MK
JOHNSON MF
MOMTAHEN T
QUEEN KL
SHERRILL RG
SZEWCZYK J
WILLSON TM
SUGG EE
Citation: Gc. Hirst et al., DISCOVERY OF 1,5-BENZODIAZEPINES WITH PERIPHERAL CHOLECYSTOKININ (CCK-A) RECEPTOR AGONIST ACTIVITY .2. OPTIMIZATION OF THE C3 AMINO SUBSTITUENT, Journal of medicinal chemistry, 39(26), 1996, pp. 5236-5245
Authors:
AQUINO CJ
ARMOUR DR
BERMAN JM
BIRKEMO LS
CARR RAE
CROOM DK
DEZUBE M
DOUGHERTY RW
ERVIN GN
GRIZZLE MK
HEAD JE
HIRST GC
JAMES MK
JOHNSON MF
MILLER LJ
QUEEN KL
RIMELE TJ
SMITH DN
SUGG EE
Citation: Cj. Aquino et al., DISCOVERY OF 1,5-BENZODIAZEPINES WITH PERIPHERAL CHOLECYSTOKININ (CCK-A) RECEPTOR AGONIST ACTIVITY .1. OPTIMIZATION OF THE AGONIST TRIGGER, Journal of medicinal chemistry, 39(2), 1996, pp. 562-569
Authors:
HENKE BR
WILLSON TM
SUGG EE
CROOM DK
DOUGHERTY RW
QUEEN KL
BIRKEMO LS
ERVIN GN
GRIZZLE MK
JOHNSON MF
JAMES MK
Citation: Br. Henke et al., 3-(1H-INDAZOL-3-YLMETHYL)-1,5-BENZODIAZEPINES - CCK-A AGONISTS THAT DEMONSTRATE ORAL ACTIVITY AS SATIETY AGENTS, Journal of medicinal chemistry, 39(14), 1996, pp. 2655-2658
Authors:
DEZUBE M
SUGG EE
BIRKEMO LS
CROOM DK
DOUGHERTY RW
ERVIN GN
GRIZZLE MK
JAMES MK
JOHNSON MF
MOSHER JT
QUEEN KL
RIMELE TJ
SAULS HR
TRIANTAFILLOU JA
Citation: M. Dezube et al., MODIFICATION OF RECEPTOR SELECTIVITY AND FUNCTIONAL-ACTIVITY IN CHOLECYSTOKININ PEPTOID LIGANDS, Journal of medicinal chemistry, 38(17), 1995, pp. 3384-3390
Authors:
FRYE SV
HAFFNER CD
MALONEY PR
HINER RN
DORSEY GF
NOE RA
UNWALLA RJ
BATCHELOR KW
BRAMSON HN
STUART JD
SCHWEIKER SL
VANAMOLD J
BICKETT DM
MOSS ML
TIAN GC
LEE FW
TIPPIN TK
JAMES MK
GRIZZLE MK
LONG JE
CROOM DK
Citation: Sv. Frye et al., STRUCTURE-ACTIVITY-RELATIONSHIPS FOR INHIBITION OF TYPE-1 AND 2 HUMAN5-ALPHA-REDUCTASE AND HUMAN ADRENAL 3-BETA-HYDROXY-DELTA(5)-STEROID DEHYDROGENASE 3-KETO-DELTA(5)-STEROID ISOMERASE BY 6-AZAANDROST-4-EN-3-ONES - OPTIMIZATION OF THE C17 SUBSTITUENT/, Journal of medicinal chemistry, 38(14), 1995, pp. 2621-2627
Authors:
JAMES MK
GRIZZLE MK
SCHUSTER SV
LONG JE
FRYE SV
HAFFNER CD
MALONEY PR
MOOK RA
DORSEY GF
HINER RN
Citation: Mk. James et al., REDUCTION OF PROSTATIC DIHYDROTESTOSTERONE (DHT) IN RATS BY A SERIES OF 6-AZASTEROID 5-ALPHA REDUCTASE (5AR) INHIBITORS, The FASEB journal, 8(5), 1994, pp. 10000638-10000638
Authors:
GRIZZLE MK
JAMES MK
SCHUSTER SV
LONG JE
FRYE SV
HAFFNER CD
MALONEY PR
MOOK RA
DORSEY GF
HINER RN
Citation: Mk. Grizzle et al., REDUCTION IN THE PROSTATE WEIGHT OF RATS BY A SERIES OF 6-AZASTEROID 5-ALPHA-REDUCTASE (5AR) INHIBITORS, The FASEB journal, 8(5), 1994, pp. 10000638-10000638
Authors:
FRYE SV
HAFFNER CD
MALONEY PR
MOOK RA
DORSEY GF
HINER RN
CRIBBS CM
WHEELER TN
RAY JA
ANDREWS RC
BATCHELOR KW
BRAMSON HN
STUART JD
SCHWEIKER SL
VANARNOLD J
CROOM S
BICKETT DM
MOSS ML
TIAN GC
UNWALLA RJ
LEE FW
TIPPIN TK
JAMES MK
GRIZZLE MK
LONG JE
SCHUSTER SV
Citation: Sv. Frye et al., 6-AZASTEROIDS - STRUCTURE-ACTIVITY-RELATIONSHIPS FOR INHIBITION OF TYPE-1 AND TYPE-2 HUMAN 5-ALPHA-REDUCTASE AND HUMAN ADRENAL 3-BETA-HYDROXY-DELTA(5)-STEROID DEHYDROGENASE 3-KETO-DELTA(5)-STEROID ISOMERASE, Journal of medicinal chemistry, 37(15), 1994, pp. 2352-2360
Authors:
SHAFFER JE
GRIZZLE MK
ANDERSON DK
WHEELER TN
Citation: Je. Shaffer et al., THE INOTROPIC AND BETA-BLOCKING EFFECTS OF A CHIMERIC MOLECULE THAT PUTATIVELY INHIBITS BOTH TYPE-III PHOSPHODIESTERASE AND BETA-ADRENOCEPTORS IN ANESTHETIZED DOGS, The Journal of pharmacology and experimental therapeutics, 265(3), 1993, pp. 1105-1112
Authors:
FRYE SV
HAFFNER CD
MALONEY PR
MOOK RA
HINER RN
BATCHELOR KW
BRAMSON HN
STUART JD
SCHWEIKER SL
VANARNOLD J
BICKETT DM
MOSS ML
TIAN GC
UNWALLA RJ
LEE FW
TIPPIN TK
JAMES MK
GRIZZLE MK
LONG JE
SCHUSTER SV
DORSEY GF
Citation: Sv. Frye et al., 6-AZASTEROIDS - POTENT DUAL INHIBITORS OF HUMAN TYPE-1 AND 2 STEROID 5-ALPHA-REDUCTASE, Journal of medicinal chemistry, 36(26), 1993, pp. 4313-4315