Authors:
Liu, G
Huth, JR
Olejniczak, ET
Mendoza, R
DeVries, P
Leitza, S
Reilly, EB
Okasinski, GF
Fesik, SW
von Geldern, TW
Citation: G. Liu et al., Novel p-arylthio cinnamides as antagonists of leukocyte function-associated antigen-1/intracellular adhesion molecule-1 interaction. 2. Mechanism of inhibition and structure-based improvement of pharmaceutical properties, J MED CHEM, 44(8), 2001, pp. 1202-1210
Authors:
Winn, M
Reilly, EB
Liu, G
Huth, JR
Jae, HS
Freeman, J
Pei, ZH
Xin, ZL
Lynch, J
Kester, J
von Geldern, TW
Leitza, S
DeVries, P
Dickinson, R
Mussatto, D
Okasinski, GF
Citation: M. Winn et al., Discovery of novel p-arylthio cinnamides as antagonists of leukocyte function-associated antigen-1/intercellular adhesion molecule-1 interaction. 4. Structure-activity relationship of substituents on the benzene ring of the cinnamide, J MED CHEM, 44(25), 2001, pp. 4393-4403
Authors:
Pei, ZH
Xin, ZL
Liu, G
Li, YH
Reilly, EB
Lubbers, NL
Huth, JR
Link, JT
von Geldern, TW
Cox, BF
Leitza, S
Gao, Y
Marsh, KC
DeVries, P
Okasinski, GF
Citation: Zh. Pei et al., Discovery of potent antagonists of leukocyte function-associated antigen-1/intercellular adhesion molecule-1 interaction. 3. Amide (C-ring) structure-activity relationship and improvement of overall properties of arylthio cinnamides, J MED CHEM, 44(18), 2001, pp. 2913-2920
Authors:
Huth, JR
Olejniczak, ET
Mendoza, R
Liang, H
Harris, EAS
Lupher, ML
Wilson, AE
Fesik, SW
Staunton, DE
Citation: Jr. Huth et al., NMR and mutagenesis evidence for an I domain allosteric site that regulates lymphocyte function-associated antigen 1 ligand binding, P NAS US, 97(10), 2000, pp. 5231-5236