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Results: 1-25 | 26-50 | 51-59
Results: 1-25/59
3'-AMIDATED 3'-DEOXYXYLOFURANOSE ANALOGS OF N-6-CYCLOPENTYLADENOSINES- A NEW CLASS OF NONXANTHINE ANTAGONISTS AT THE ADENOSINE A(1) RECEPTOR
Authors: VANCALENBERGH S IJZERMAN AP HERDEWIJN P
Citation: S. Vancalenbergh et al., 3'-AMIDATED 3'-DEOXYXYLOFURANOSE ANALOGS OF N-6-CYCLOPENTYLADENOSINES- A NEW CLASS OF NONXANTHINE ANTAGONISTS AT THE ADENOSINE A(1) RECEPTOR, Nucleosides & nucleotides, 17(9-11), 1998, pp. 1571-1576
A FUNCTIONAL SCREENING OF ADENOSINE-ANALOGS AT THE ADENOSINE A(2B) RECEPTOR - A SEARCH FOR POTENT AGONISTS
Authors: DEZWART M LINK R KUNZEL JKV CRISTALLI G JACOBSON KA TOWNSENDNICHOLSON A IJZERMAN AP
Citation: M. Dezwart et al., A FUNCTIONAL SCREENING OF ADENOSINE-ANALOGS AT THE ADENOSINE A(2B) RECEPTOR - A SEARCH FOR POTENT AGONISTS, Nucleosides & nucleotides, 17(6), 1998, pp. 969-985
MOLECULAR RECEPTORS MODELING OF G-PROTEIN-COUPLED
Authors: IJZERMAN AP
Citation: Ap. Ijzerman, MOLECULAR RECEPTORS MODELING OF G-PROTEIN-COUPLED, Naunyn-Schmiedeberg's archives of pharmacology, 358(1), 1998, pp. 125-125
MOLECULAR MODELING OF G-PROTEIN-COUPLED RECEPTORS
Authors: IJZERMAN AP
Citation: Ap. Ijzerman, MOLECULAR MODELING OF G-PROTEIN-COUPLED RECEPTORS, Naunyn-Schmiedeberg's archives of pharmacology, 358(1), 1998, pp. 133-133
METABOLIC AND CARDIOVASCULAR EFFECTS OF THE ADENOSINE A(1) RECEPTOR AGONIST N-6-(P-SULFOPHENYL)ADENOSINE IN DIABETIC ZUCKER RATS - INFLUENCE OF THE DISEASE ON THE SELECTIVITY OF ACTION
Authors: VANSCHAICK EA ZUIDEVELD KP TUKKER HE LANGEMEIJER MWE IJZERMAN AP DANHOF M
Citation: Ea. Vanschaick et al., METABOLIC AND CARDIOVASCULAR EFFECTS OF THE ADENOSINE A(1) RECEPTOR AGONIST N-6-(P-SULFOPHENYL)ADENOSINE IN DIABETIC ZUCKER RATS - INFLUENCE OF THE DISEASE ON THE SELECTIVITY OF ACTION, The Journal of pharmacology and experimental therapeutics, 287(1), 1998, pp. 21-30
A NOVEL CLASS OF ADENOSINE A(3) RECEPTOR LIGANDS - 1 - 3-(2-PYRIDINYL)ISOQUINOLINE DERIVATIVES
Authors: VANMUIJLWIJKKOEZEN JE TIMMERMAN H LINK R VANDERGOOT H IJZERMAN AP
Citation: Je. Vanmuijlwijkkoezen et al., A NOVEL CLASS OF ADENOSINE A(3) RECEPTOR LIGANDS - 1 - 3-(2-PYRIDINYL)ISOQUINOLINE DERIVATIVES, Journal of medicinal chemistry, 41(21), 1998, pp. 3987-3993
DERIVATIVES OF THE TRIAZOLOQUINAZOLINE ADENOSINE ANTAGONIST (CGS-15943) HAVING HIGH POTENCY AT THE HUMAN A(2B) AND A(3) RECEPTOR SUBTYPES
Authors: KIM YC DEZWART M CHANG L MORO S KUNZEL JKVD MELMAN N IJZERMAN AP JACOBSON KA
Citation: Yc. Kim et al., DERIVATIVES OF THE TRIAZOLOQUINAZOLINE ADENOSINE ANTAGONIST (CGS-15943) HAVING HIGH POTENCY AT THE HUMAN A(2B) AND A(3) RECEPTOR SUBTYPES, Journal of medicinal chemistry, 41(15), 1998, pp. 2835-2845
5'-SUBSTITUTED ADENOSINE-ANALOGS AS NEW HIGH-AFFINITY PARTIAL AGONISTS FOR THE ADENOSINE A(1) RECEPTOR
Authors: VANDERWENDEN EM CARNIELLI M ROELEN HCPF LORENZEN A VONFRIJTAG JK KUNZEL D IJZERMAN AP
Citation: Em. Vanderwenden et al., 5'-SUBSTITUTED ADENOSINE-ANALOGS AS NEW HIGH-AFFINITY PARTIAL AGONISTS FOR THE ADENOSINE A(1) RECEPTOR, Journal of medicinal chemistry, 41(1), 1998, pp. 102-108
ROLE OF CERAMIDE-1 IN THE MOLECULAR-ORGANIZATION OF THE STRATUM-CORNEUM LIPIDS
Authors: BOUWSTRA JA GOORIS GS DUBBELAAR FER WEERHEIM AM IJZERMAN AP PONEC M
Citation: Ja. Bouwstra et al., ROLE OF CERAMIDE-1 IN THE MOLECULAR-ORGANIZATION OF THE STRATUM-CORNEUM LIPIDS, Journal of lipid research, 39(1), 1998, pp. 186-196
SELECTIVITY OF ACTION OF 8-ALKYLAMINO ANALOGS OF N-6-CYCLOPENTYLADENOSINE IN-VIVO - HEMODYNAMIC VERSUS ANTI-LIPOLYTIC RESPONSES IN RATS
Authors: VANSCHAICK EA TUKKER HE ROELEN HCPF IJZERMAN AP DANHOF M
Citation: Ea. Vanschaick et al., SELECTIVITY OF ACTION OF 8-ALKYLAMINO ANALOGS OF N-6-CYCLOPENTYLADENOSINE IN-VIVO - HEMODYNAMIC VERSUS ANTI-LIPOLYTIC RESPONSES IN RATS, British Journal of Pharmacology, 124(3), 1998, pp. 607-618
THERMODYNAMICS OF FULL AGONIST, PARTIAL AGONIST, AND ANTAGONIST BINDING TO WILD-TYPE AND MUTANT ADENOSINE A(1) RECEPTORS
Authors: DALPIAZ A TOWNSENDNICHOLSON A BEUKERS MW SCHOFIELD PR IJZERMAN AP
Citation: A. Dalpiaz et al., THERMODYNAMICS OF FULL AGONIST, PARTIAL AGONIST, AND ANTAGONIST BINDING TO WILD-TYPE AND MUTANT ADENOSINE A(1) RECEPTORS, Biochemical pharmacology, 56(11), 1998, pp. 1437-1445
IDENTIFICATION OF CLASS-DETERMINING RESIDUES IN G-PROTEIN-COUPLED RECEPTORS BY SEQUENCE-ANALYSIS
Authors: KUIPERS W OLIVEIRA L VRIEND G IJZERMAN AP
Citation: W. Kuipers et al., IDENTIFICATION OF CLASS-DETERMINING RESIDUES IN G-PROTEIN-COUPLED RECEPTORS BY SEQUENCE-ANALYSIS, Receptors & channels, 5(3-4), 1997, pp. 159-174
PHYSIOLOGICAL INDIRECT EFFECT MODELING OF THE ANTILIPOLYTIC EFFECTS OF ADENOSINE A(1)-RECEPTOR AGONISTS
Authors: VANSCHAICK EA DEGREEF HJMM IJZERMAN AP DANHOF M
Citation: Ea. Vanschaick et al., PHYSIOLOGICAL INDIRECT EFFECT MODELING OF THE ANTILIPOLYTIC EFFECTS OF ADENOSINE A(1)-RECEPTOR AGONISTS, Journal of pharmacokinetics and biopharmaceutics, 25(6), 1997, pp. 673-694
TIME-COURSE OF ACTION OF 3 ADENOSINE A(1) RECEPTOR AGONISTS WITH DIFFERING LIPOPHILICITY IN RATS - COMPARISON OF PHARMACOKINETIC, HEMODYNAMIC AND EEG EFFECTS
Authors: VANSCHAICK EA KULKARNI C KUNZEL JKVD MATHOT RAA CRISTALLI G IJZERMAN AP DANHOF M
Citation: Ea. Vanschaick et al., TIME-COURSE OF ACTION OF 3 ADENOSINE A(1) RECEPTOR AGONISTS WITH DIFFERING LIPOPHILICITY IN RATS - COMPARISON OF PHARMACOKINETIC, HEMODYNAMIC AND EEG EFFECTS, Naunyn-Schmiedeberg's archives of pharmacology, 356(6), 1997, pp. 827-837
FUNCTIONAL-CHARACTERIZATION OF N-6, C8-DISUBSTITUTED ADENOSINE DERIVATIVES AS PARTIAL AGONISTS AT RAT-BRAIN ADENOSINE A(1) RECEPTORS
Authors: LORENZEN A SEBASTIAO AM SELLINK A VOGT H SCHWABE U RIBEIRO JA IJZERMAN AP
Citation: A. Lorenzen et al., FUNCTIONAL-CHARACTERIZATION OF N-6, C8-DISUBSTITUTED ADENOSINE DERIVATIVES AS PARTIAL AGONISTS AT RAT-BRAIN ADENOSINE A(1) RECEPTORS, Naunyn-Schmiedeberg's archives of pharmacology, 356(4), 1997, pp. 153-153
POTENCY AND EFFICACY OF PARTIAL AGONISTS OF THE ADENOSINE A(1) RECEPTOR IN G-PROTEIN ACTIVATION AND INHIBITION OF ADENYLATE-CYCLASE
Authors: LORENZEN A VOGT H VANDERWENDEN EM ROELEN HCPF CARNIELLI M IJZERMAN AP SCHWABE U
Citation: A. Lorenzen et al., POTENCY AND EFFICACY OF PARTIAL AGONISTS OF THE ADENOSINE A(1) RECEPTOR IN G-PROTEIN ACTIVATION AND INHIBITION OF ADENYLATE-CYCLASE, Naunyn-Schmiedeberg's archives of pharmacology, 355(4), 1997, pp. 110-110
STUDY OF THE INTERACTION BETWEEN ARYLOXYPROPANOLAMINES AND ASN386 IN HELIX-VII OF THE HUMAN 5-HYDROXYTRYPTAMINE(1A) RECEPTOR
Authors: KUIPERS W LINK R STANDAAR PJ STOIT AR VANWIJNGAARDEN I LEURS R IJZERMAN AP
Citation: W. Kuipers et al., STUDY OF THE INTERACTION BETWEEN ARYLOXYPROPANOLAMINES AND ASN386 IN HELIX-VII OF THE HUMAN 5-HYDROXYTRYPTAMINE(1A) RECEPTOR, Molecular pharmacology, 51(5), 1997, pp. 889-896
8-ALKYLAMINO-SUBSTITUTED ANALOGS OF N-6-CYCLOPENTYLADENOSINE ARE PARTIAL AGONISTS FOR THE CARDIOVASCULAR ADENOSINE A(1) RECEPTORS IN-VIVO
Authors: VANSCHAICK EA MATHOT RAA GUBBENSSTIBBE JM LANGEMEIJER MWE ROELEN HCPF IJZERMAN AP DANHOF M
Citation: Ea. Vanschaick et al., 8-ALKYLAMINO-SUBSTITUTED ANALOGS OF N-6-CYCLOPENTYLADENOSINE ARE PARTIAL AGONISTS FOR THE CARDIOVASCULAR ADENOSINE A(1) RECEPTORS IN-VIVO, The Journal of pharmacology and experimental therapeutics, 283(2), 1997, pp. 800-808
MECHANISM-BASED PHARMACOKINETIC-PHARMACODYNAMIC MODELING OF THE EFFECTS OF N-6-CYCLOPENTYLADENOSINE ANALOGS ON HEART-RATE IN RAT - ESTIMATION OF IN-VIVO OPERATIONAL AFFINITY AND EFFICACY AT ADENOSINE A(1) RECEPTORS
Authors: VANDERGRAAF PH VANSCHAICK EA MATHOT RAA IJZERMAN AP DANHOF M
Citation: Ph. Vandergraaf et al., MECHANISM-BASED PHARMACOKINETIC-PHARMACODYNAMIC MODELING OF THE EFFECTS OF N-6-CYCLOPENTYLADENOSINE ANALOGS ON HEART-RATE IN RAT - ESTIMATION OF IN-VIVO OPERATIONAL AFFINITY AND EFFICACY AT ADENOSINE A(1) RECEPTORS, The Journal of pharmacology and experimental therapeutics, 283(2), 1997, pp. 809-816
DETERMINATION OF DEXMEDETOMIDINE IN RAT PLASMA BY A SENSITIVE [H-3] CLONIDINE RADIORECEPTOR ASSAY
Authors: BOL CJJG IJZERMAN AP DANHOF M MANDEMA JW
Citation: Cjjg. Bol et al., DETERMINATION OF DEXMEDETOMIDINE IN RAT PLASMA BY A SENSITIVE [H-3] CLONIDINE RADIORECEPTOR ASSAY, Journal of pharmaceutical sciences, 86(7), 1997, pp. 822-826
5-HT1A-VERSUS D-2-RECEPTOR SELECTIVITY OF FLESINOXAN AND ANALOGOUS N-4-SUBSTITUTED N-1-ARYLPIPERAZINES
Authors: KUIPERS W KRUSE CG VANWIJNGAARDEN I STANDAAR PJ TULP MTM VELDMAN N SPEK AL IJZERMAN AP
Citation: W. Kuipers et al., 5-HT1A-VERSUS D-2-RECEPTOR SELECTIVITY OF FLESINOXAN AND ANALOGOUS N-4-SUBSTITUTED N-1-ARYLPIPERAZINES, Journal of medicinal chemistry, 40(3), 1997, pp. 300-312
CYCLOPENTYL-3'-SUBSTITUTED-XYLOFURANOSYLADENOSINES - A NEW CLASS OF NONXANTHINE ADENOSINE A(1) RECEPTOR ANTAGONISTS
Authors: VANCALENBERGH S VONFRIJTAG JK KUNZEL D BLATON NM PEETERS OM ROZENSKI J VANAERSCHOT A DEBRUYN A DEKEUKELEIRE D IJZERMAN AP HERDEWIJN P
Citation: S. Vancalenbergh et al., CYCLOPENTYL-3'-SUBSTITUTED-XYLOFURANOSYLADENOSINES - A NEW CLASS OF NONXANTHINE ADENOSINE A(1) RECEPTOR ANTAGONISTS, Journal of medicinal chemistry, 40(23), 1997, pp. 3765-3772
BIOLOGICAL-ACTIVITIES OF N-6,C8-DISUBSTITUTED ADENOSINE DERIVATIVES AS PARTIAL AGONISTS AT RAT-BRAIN ADENOSINE A(1) RECEPTORS
Authors: LORENZEN A SEBASTIAO AM SELLINK A VOGT H SCHWABE U RIBEIRO JA IJZERMAN AP
Citation: A. Lorenzen et al., BIOLOGICAL-ACTIVITIES OF N-6,C8-DISUBSTITUTED ADENOSINE DERIVATIVES AS PARTIAL AGONISTS AT RAT-BRAIN ADENOSINE A(1) RECEPTORS, European journal of pharmacology, 334(2-3), 1997, pp. 299-307
MUTATIONAL ANALYSIS OF THE PUTATIVE DEVAZEPIDE BINDING-SITE OF THE CCKA RECEPTOR
Authors: SMEETS RLL IJZERMAN AP HERMSEN HPH OPHORST OJAE VRIES SEV DEPONT JJHHM WILLEMS PHGM
Citation: Rll. Smeets et al., MUTATIONAL ANALYSIS OF THE PUTATIVE DEVAZEPIDE BINDING-SITE OF THE CCKA RECEPTOR, European journal of pharmacology, 325(1), 1997, pp. 93-99
PHARMACOKINETIC-PHARMACODYNAMIC MODELING OF THE ANTI-LIPOLYTIC AND ANTI-KETOTIC EFFECTS OF THE ADENOSINE A(1)-RECEPTOR AGONIST N-6-(P-SULPHOPHENYL)ADENOSINE IN RATS
Authors: VANSCHAICK EA DEGREEF HJMM LANGEMEIJER MWE SHEEHAN MJ IJZERMAN AP DANHOF M
Citation: Ea. Vanschaick et al., PHARMACOKINETIC-PHARMACODYNAMIC MODELING OF THE ANTI-LIPOLYTIC AND ANTI-KETOTIC EFFECTS OF THE ADENOSINE A(1)-RECEPTOR AGONIST N-6-(P-SULPHOPHENYL)ADENOSINE IN RATS, British Journal of Pharmacology, 122(3), 1997, pp. 525-533
Risultati: 1-25 | 26-50 | 51-59