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Results: 1-10 |
Results: 10
INHIBITION OF HUMAN NEUTROPHIL ELASTASE - 4 - DESIGN, SYNTHESIS, X-RAY CRYSTALLOGRAPHIC ANALYSIS, AND STRUCTURE-ACTIVITY-RELATIONSHIPS FOR A SERIES OF P-2-MODIFIED, ORALLY-ACTIVE PEPTIDYL PENTAFLUOROETHYL KETONES
Authors: CREGGE RJ DURHAM SL FARR RA GALLION SL HARE CM HOFFMAN RV JANUSZ MJ KIM HO KOEHL JR MEHDI S METZ WA PEET NP PELTON JT SCHREUDER HA SUNDER S TARDIF C
Citation: Rj. Cregge et al., INHIBITION OF HUMAN NEUTROPHIL ELASTASE - 4 - DESIGN, SYNTHESIS, X-RAY CRYSTALLOGRAPHIC ANALYSIS, AND STRUCTURE-ACTIVITY-RELATIONSHIPS FOR A SERIES OF P-2-MODIFIED, ORALLY-ACTIVE PEPTIDYL PENTAFLUOROETHYL KETONES, Journal of medicinal chemistry, 41(14), 1998, pp. 2461-2480
HUMAN CHONDROSARCOMA CELLS STABLY TRANSFECTED WITH A STROMELYSIN (MMP-3) PROMOTER REPORTER CONSTRUCT PROVIDE A METHOD OF ASSESSING TRANSCRIPTIONAL INHIBITORS
Authors: JANUSZ MJ HARE CM DURHAM SL WOESSNER RD
Citation: Mj. Janusz et al., HUMAN CHONDROSARCOMA CELLS STABLY TRANSFECTED WITH A STROMELYSIN (MMP-3) PROMOTER REPORTER CONSTRUCT PROVIDE A METHOD OF ASSESSING TRANSCRIPTIONAL INHIBITORS, Inflammation research, 46, 1997, pp. 159-160
INHIBITION OF CARTILAGE DEGRADATION IN RAT COLLAGEN-INDUCED ARTHRITISBUT NOT ADJUVANT ARTHRITIS BY THE NEUTROPHIL ELASTASE INHIBITOR MDL-101,146
Authors: JANUSZ MJ DURHAM SL
Citation: Mj. Janusz et Sl. Durham, INHIBITION OF CARTILAGE DEGRADATION IN RAT COLLAGEN-INDUCED ARTHRITISBUT NOT ADJUVANT ARTHRITIS BY THE NEUTROPHIL ELASTASE INHIBITOR MDL-101,146, Inflammation research, 46(12), 1997, pp. 503-508
PHARMACOLOGICAL EVALUATION OF SELECTED, ORALLY-ACTIVE, PEPTIDYL INHIBITORS OF HUMAN NEUTROPHIL ELASTASE
Authors: JANUSZ MJ DURHAM SL HARE CM GEARY JL MANDAGERE AK POOLE JC THOMPSON TN XU D ANGELASTRO MR BURKHART JP CHEN TM MARQUART AL PEET NP HWANG KK
Citation: Mj. Janusz et al., PHARMACOLOGICAL EVALUATION OF SELECTED, ORALLY-ACTIVE, PEPTIDYL INHIBITORS OF HUMAN NEUTROPHIL ELASTASE, The Journal of pharmacology and experimental therapeutics, 275(3), 1995, pp. 1233-1238
INHIBITION OF HUMAN NEUTROPHIL ELASTASE .3. AN ORALLY-ACTIVE ENOL ACETATE PRODRUG
Authors: BURKHART JP KOEHL JR MEHDI S DURHAM SL JANUSZ MJ HUBER EW ANGELASTRO MR SUNDER S METZ WA SHUM PW CHEN TM BEY P CREGGE RJ PEET NP
Citation: Jp. Burkhart et al., INHIBITION OF HUMAN NEUTROPHIL ELASTASE .3. AN ORALLY-ACTIVE ENOL ACETATE PRODRUG, Journal of medicinal chemistry, 38(2), 1995, pp. 223-233
INHIBITION OF HUMAN NEUTROPHIL ELASTASE AND CATHEPSIN-G BY A BIPHENYLDISULFONIC ACID COPOLYMER
Authors: JANUSZ MJ HARE M
Citation: Mj. Janusz et M. Hare, INHIBITION OF HUMAN NEUTROPHIL ELASTASE AND CATHEPSIN-G BY A BIPHENYLDISULFONIC ACID COPOLYMER, International journal of immunopharmacology, 16(8), 1994, pp. 623-632
PHARMACOLOGY OF FLUORO-1-(1-METHYLETHYL)-2-OXOBUTYL]-L-PROLINAMIDE (MDL-101,146) - A POTENT ORALLY-ACTIVE INHIBITOR OF HUMAN NEUTROPHIL ELASTASE (VOL 270, PG 185, 1994)
Authors: DURHAM SL HARE CM ANGELASTRO MR BURKHART JP KOEHL JR MARQUART AL MEHDI S PEET NP JANUSZ MJ
Citation: Sl. Durham et al., PHARMACOLOGY OF FLUORO-1-(1-METHYLETHYL)-2-OXOBUTYL]-L-PROLINAMIDE (MDL-101,146) - A POTENT ORALLY-ACTIVE INHIBITOR OF HUMAN NEUTROPHIL ELASTASE (VOL 270, PG 185, 1994), The Journal of pharmacology and experimental therapeutics, 271(3), 1994, pp. 1720-1720
PHARMACOLOGY OF FLUORO-1-(1-METHYLETHYL)-2-OXOBUTYL]-L-PROLINAMIDE (MDL-101,146) - A POTENT ORALLY-ACTIVE INHIBITOR OF HUMAN NEUTROPHIL ELASTASE
Authors: DURHAM SL HARE CM ANGELASTRO MR BURKHART JP KOEHL JR MARQUART AL MEHDI S FEET NP JANUSZ MJ
Citation: Sl. Durham et al., PHARMACOLOGY OF FLUORO-1-(1-METHYLETHYL)-2-OXOBUTYL]-L-PROLINAMIDE (MDL-101,146) - A POTENT ORALLY-ACTIVE INHIBITOR OF HUMAN NEUTROPHIL ELASTASE, The Journal of pharmacology and experimental therapeutics, 270(1), 1994, pp. 185-191
INHIBITION OF HUMAN NEUTROPHIL ELASTASE WITH PEPTIDYL ELECTROPHILIC KETONES .2. ORALLY-ACTIVE P-G-VAL-PRO-VAL PENTAFLUOROETHYL KETONES
Authors: ANGELASTRO MR BAUGH LE BEY P BURKHART JP CHEN TM DURHAM SL HARE CM HUBER EW JANUSZ MJ KOEHL JR MARQUART AL MEHDI S PEET NP
Citation: Mr. Angelastro et al., INHIBITION OF HUMAN NEUTROPHIL ELASTASE WITH PEPTIDYL ELECTROPHILIC KETONES .2. ORALLY-ACTIVE P-G-VAL-PRO-VAL PENTAFLUOROETHYL KETONES, Journal of medicinal chemistry, 37(26), 1994, pp. 4538-4553
MDL 101,146, A POTENT ORALLY ACTIVE INHIBITOR OF HUMAN NEUTROPHIL ELASTASE INDUCED ACUTE PULMONARY HEMORRHAGE IN RATS AND HAMSTERS
Authors: DURHAM SL HARE CM ANGELASTRO MR BURKHART JP KOEHL JR MARQUART AL MEHDI S PEET NP JANUSZ MJ
Citation: Sl. Durham et al., MDL 101,146, A POTENT ORALLY ACTIVE INHIBITOR OF HUMAN NEUTROPHIL ELASTASE INDUCED ACUTE PULMONARY HEMORRHAGE IN RATS AND HAMSTERS, The American review of respiratory disease, 147(4), 1993, pp. 675-675
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