AAAAAA

   
Results: 1-25 | 26-50 | 51-61
Results: 1-25/61
Ribose modified nucleosides and nucleotides as ligands for purine receptors
Authors: Jacobson, KA Ravi, RG Nandanan, E Kim, HS Moro, S Kim, YC Lee, K Barak, D Marquez, VE Ji, XD
Citation: Ka. Jacobson et al., Ribose modified nucleosides and nucleotides as ligands for purine receptors, NUCLEOS NUC, 20(4-7), 2001, pp. 333-341
Synthesis using ring closure metathesis and effect on nucleoside transportof a (N)-methanocarba S-(4-nitrobenzyl)thioinosine derivative
Authors: Lee, K Cass, C Jacobson, KA
Citation: K. Lee et al., Synthesis using ring closure metathesis and effect on nucleoside transportof a (N)-methanocarba S-(4-nitrobenzyl)thioinosine derivative, ORG LETT, 3(4), 2001, pp. 597-599
Synthesis and purine receptor affinity of 6-oxopurine nucleosides and nucleotides containing (N)-methanocarba-pseudoribose rings
Authors: Ravi, G Lee, K Ji, XD Kim, HS Soltysiak, KA Marquez, VE Jacobson, KA
Citation: G. Ravi et al., Synthesis and purine receptor affinity of 6-oxopurine nucleosides and nucleotides containing (N)-methanocarba-pseudoribose rings, BIOORG MED, 11(17), 2001, pp. 2295-2300
Ring-constrained (N)-methanocarba nucleosides as adenosine receptor agonists: Independent 5 '-uronamide and 2 '-deoxy modifications
Authors: Lee, K Ravi, G Ji, XD Marquez, VE Jacobson, KA
Citation: K. Lee et al., Ring-constrained (N)-methanocarba nucleosides as adenosine receptor agonists: Independent 5 '-uronamide and 2 '-deoxy modifications, BIOORG MED, 11(10), 2001, pp. 1333-1337
Induction of cortical oscillations in spreading cells by depolymerization of microtubules
Authors: Pletjushkina, OJ Rajfur, Z Pomorski, P Oliver, TN Vasiliev, JM Jacobson, KA
Citation: Oj. Pletjushkina et al., Induction of cortical oscillations in spreading cells by depolymerization of microtubules, CELL MOTIL, 48(4), 2001, pp. 235-244
Cardioprotective effects of adenosine A(1) and A(3) receptor activation during hypoxia in isolated rat cardiac myocytes
Authors: Safran, N Shneyvays, V Balas, N Jacobson, KA Nawrath, H Shainberg, A
Citation: N. Safran et al., Cardioprotective effects of adenosine A(1) and A(3) receptor activation during hypoxia in isolated rat cardiac myocytes, MOL C BIOCH, 217(1-2), 2001, pp. 143-152
Actions of a series of PPADS analogs at P2X(1) and P2X(3) receptors
Authors: Brown, SG Kim, YC Kim, SA Jacobson, KA Burnstock, G King, BF
Citation: Sg. Brown et al., Actions of a series of PPADS analogs at P2X(1) and P2X(3) receptors, DRUG DEV R, 53(4), 2001, pp. 281-291
Two distinct P2Y receptors are involved in purine- and pyrimidine-evoked Ca2+ elevation in mammalian brain astrocytic cultures
Authors: Bolego, C Centemeri, C Abbracchio, MP Ceruti, S Cattabeni, F Jacobson, KA Puglisi, L Rovati, GE Burnstock, G Nicosia, S
Citation: C. Bolego et al., Two distinct P2Y receptors are involved in purine- and pyrimidine-evoked Ca2+ elevation in mammalian brain astrocytic cultures, DRUG DEV R, 52(1-2), 2001, pp. 122-132
Probing adenosine and P2 receptors: Design of novel purines and nonpurinesas selective ligands
Authors: Jacobson, KA
Citation: Ka. Jacobson, Probing adenosine and P2 receptors: Design of novel purines and nonpurinesas selective ligands, DRUG DEV R, 52(1-2), 2001, pp. 178-186
Adenosine A(1) and A(3) receptors: Distinct cardioprotection
Authors: Liang, BT Stewart, D Jacobson, KA
Citation: Bt. Liang et al., Adenosine A(1) and A(3) receptors: Distinct cardioprotection, DRUG DEV R, 52(1-2), 2001, pp. 366-378
Angiotensin II-induced apoptosis in rat cardiomyocyte culture: a possible role of AT(1) and AT(2) receptors
Authors: Goldenberg, I Grossman, E Jacobson, KA Shneyvays, V Shainberg, A
Citation: I. Goldenberg et al., Angiotensin II-induced apoptosis in rat cardiomyocyte culture: a possible role of AT(1) and AT(2) receptors, J HYPERTENS, 19(9), 2001, pp. 1681-1689
P1 and P2 purine and pyrimidine receptor ligands
Authors: Jacobson, KA Knutsen, LJS
Citation: Ka. Jacobson et Ljs. Knutsen, P1 and P2 purine and pyrimidine receptor ligands, HANDB EXP P, 151, 2001, pp. 129-175
Allosteric modulation of A(3) adenosine receptors by a series of 3-(2-pyridinyl)isoquinoline derivatives
Authors: Gao, ZG Van Muijlwijk-Koezen, JE Chen, AS Muller, CE IJzerman, AP Jacobson, KA
Citation: Zg. Gao et al., Allosteric modulation of A(3) adenosine receptors by a series of 3-(2-pyridinyl)isoquinoline derivatives, MOLEC PHARM, 60(5), 2001, pp. 1057-1063
Structure-activity relationships of pyridoxal phosphate derivatives as potent and selective antagonists of P2X(1) receptors
Authors: Kim, YC Brown, SG Harden, TK Boyer, JL Dubyak, G King, BF Burnstock, G Jacobson, KA
Citation: Yc. Kim et al., Structure-activity relationships of pyridoxal phosphate derivatives as potent and selective antagonists of P2X(1) receptors, J MED CHEM, 44(3), 2001, pp. 340-349
Neoceptor concept based on molecular complementarity in GPCRs: A mutant adenosine A(3) receptor with selectively enhanced affinity for amine-modifiednucleosides
Authors: Jacobson, KA Gao, ZG Chen, AS Barak, D Kim, SA Lee, K Link, A Van Rompaey, P van Calenbergh, S Liang, BT
Citation: Ka. Jacobson et al., Neoceptor concept based on molecular complementarity in GPCRs: A mutant adenosine A(3) receptor with selectively enhanced affinity for amine-modifiednucleosides, J MED CHEM, 44(24), 2001, pp. 4125-4136
Acyclic and cyclopropyl analogues of adenosine bisphosphate antagonists ofthe P2Y(1) receptor: Structure-activity relationships and receptor docking
Authors: Kim, HS Barak, D Harden, TK Boyer, JL Jacobson, KA
Citation: Hs. Kim et al., Acyclic and cyclopropyl analogues of adenosine bisphosphate antagonists ofthe P2Y(1) receptor: Structure-activity relationships and receptor docking, J MED CHEM, 44(19), 2001, pp. 3092-3108
Fluorosulfonyl- and bis-(beta-chloroethyl)amino-phenylamino functionalizedpyrazolo[4,3-e]1,2,4-triazolo[1,5-c]pyrimidine derivatives: Irreversible antagonists at the human A(3) adenosine receptor and molecular modeling studies
Authors: Baraldi, PG Cacciari, B Moro, S Romagnoli, R Ji, XD Jacobson, KA Gessi, S Borea, PA Spalluto, G
Citation: Pg. Baraldi et al., Fluorosulfonyl- and bis-(beta-chloroethyl)amino-phenylamino functionalizedpyrazolo[4,3-e]1,2,4-triazolo[1,5-c]pyrimidine derivatives: Irreversible antagonists at the human A(3) adenosine receptor and molecular modeling studies, J MED CHEM, 44(17), 2001, pp. 2735-2742
[H-3]MRS 1754, a selective antagonist radioligand for A(2B) adenosine receptors
Authors: Ji, XD Kim, YC Ahern, DG Linden, J Jacobson, KA
Citation: Xd. Ji et al., [H-3]MRS 1754, a selective antagonist radioligand for A(2B) adenosine receptors, BIOCH PHARM, 61(6), 2001, pp. 657-663
Constitutive activation of A(3) adenosine receptors by site-directed mutagenesis
Authors: Chen, A Gao, ZG Barak, D Liang, BT Jacobson, KA
Citation: A. Chen et al., Constitutive activation of A(3) adenosine receptors by site-directed mutagenesis, BIOC BIOP R, 284(3), 2001, pp. 596-601
Structure-activity relationships for G2 checkpoint inhibition by caffeine analogs
Authors: Jiang, XX Lim, LY Daly, JW Li, AH Jacobson, KA Roberge, M
Citation: Xx. Jiang et al., Structure-activity relationships for G2 checkpoint inhibition by caffeine analogs, INT J ONCOL, 16(5), 2000, pp. 971-978
The utilization of a unified pharmacophore query in the discovery of new antagonists of the adenosine receptor family
Authors: Webb, TR Melman, N Lvovskiy, D Ji, XD Jacobson, KA
Citation: Tr. Webb et al., The utilization of a unified pharmacophore query in the discovery of new antagonists of the adenosine receptor family, BIOORG MED, 10(1), 2000, pp. 31-34
Distinct cardioprotective effects of adenosine mediated by differential coupling of receptor subtypes to phospholipases C and D
Authors: Parsons, M Young, L Lee, JE Jacobson, KA Liang, BT
Citation: M. Parsons et al., Distinct cardioprotective effects of adenosine mediated by differential coupling of receptor subtypes to phospholipases C and D, FASEB J, 14(10), 2000, pp. 1423-1431
Inhibition of ecto-apyrase and ecto-ATPase by pyridoxal phosphate-related compounds
Authors: Hoffmann, C Heine, P Pradel, G Kim, YC Jacobson, KA Zimmermann, H
Citation: C. Hoffmann et al., Inhibition of ecto-apyrase and ecto-ATPase by pyridoxal phosphate-related compounds, DRUG DEV R, 51(3), 2000, pp. 153-158
Purification and recognition of recombinant mouse P2X(1) receptors expressed in a baculovirus system
Authors: Chen, LP Hardwick, JP McPhie, P Sitkovsky, MV Jacobson, KA
Citation: Lp. Chen et al., Purification and recognition of recombinant mouse P2X(1) receptors expressed in a baculovirus system, DRUG DEV R, 51(1), 2000, pp. 7-19
Activity of novel adenine nucleotide derivatives as agonists and antagonists at recombinant rat P2X receptors
Authors: Brown, SG King, BF Kim, YC Jang, SY Burnstock, G Jacobson, KA
Citation: Sg. Brown et al., Activity of novel adenine nucleotide derivatives as agonists and antagonists at recombinant rat P2X receptors, DRUG DEV R, 49(4), 2000, pp. 253-259
Risultati: 1-25 | 26-50 | 51-61