Authors:
Miller, WH
Bondinell, WE
Cousins, RD
Erhard, KF
Jakas, DR
Keenan, RM
Ku, TW
Newlander, KA
Ross, ST
Haltiwanger, RC
Bradbeer, J
Drake, FH
Gowen, M
Hoffman, SJ
Hwang, SM
James, IE
Lark, MW
Lechowska, B
Rieman, DJ
Stroup, GB
Vasko-Moser, JA
Zembryki, DL
Azzarano, LM
Adams, PC
Salyers, KL
Smith, BR
Ward, KW
Johanson, KO
Huffman, WF
Citation: Wh. Miller et al., Orally bioavailable nonpeptide vitronectin receptor antagonists with efficacy in an osteoporosis model, BIOORG MED, 9(13), 1999, pp. 1807-1812
Authors:
Sarau, HM
Foley, JJ
Schmidt, DB
Martin, LD
Webb, EF
Tzimas, MN
Breton, JJ
Chabot-Fletcher, M
Underwood, DC
Hay, DWP
Kingsbury, WD
Chambers, PA
Pendrak, I
Jakas, DR
Sathe, GM
Van Horn, S
Daines, RA
Griswold, DE
Citation: Hm. Sarau et al., In vitro and in vivo pharmacological characterization of SB 201993, an eicosanoid-like LTB4 receptor antagonist with anti-inflammatory activity, PROS LEUK E, 61(1), 1999, pp. 55-64
Authors:
Ward, KW
Azzarano, LM
Bondinell, WE
Cousins, RD
Huffman, WF
Jakas, DR
Keenan, RM
Ku, TW
Lundberg, D
Miller, WH
Mumaw, JA
Newlander, KA
Pirhalla, JL
Roethke, TJ
Salyers, KL
Souder, PR
Stelman, GJ
Smith, BR
Citation: Kw. Ward et al., Preclinical pharmacokinetics and interspecies scaling of a novel vitronectin receptor antagonist, DRUG META D, 27(11), 1999, pp. 1232-1241
Authors:
Keenan, RM
Callahan, JF
Samanen, JM
Bondinell, WE
Calvo, RR
Chen, LC
DeBrosse, C
Eggleston, DS
Haltiwanger, RC
Hwang, SM
Jakas, DR
Ku, TW
Miller, WH
Newlander, KA
Nichols, A
Parker, MF
Southhall, LS
Uzinskas, I
Vasko-Moser, JA
Venslavsky, JW
Wong, AS
Huffman, WF
Citation: Rm. Keenan et al., Conformational preferences in a benzodiazepine series of potent nonpeptidefibrinogen receptor antagonists, J MED CHEM, 42(4), 1999, pp. 545-559
Authors:
Keenan, RM
Miller, WH
Lago, MA
Ali, FE
Bondinell, WE
Callahan, JF
Calvo, RR
Cousins, RD
Hwang, SM
Jakas, DR
Ku, TW
Kwon, C
Nguyen, TT
Reader, VA
Rieman, DJ
Ross, ST
Takata, DT
Uzinskas, IN
Yuan, CCK
Smith, BR
Citation: Rm. Keenan et al., Benzimidazole derivatives as arginine mimetics in 1,4-benzodiazepine nonpeptide vitronectin receptor (alpha v beta 3) antagonists, BIOORG MED, 8(22), 1998, pp. 3165-3170
Authors:
Keenan, RM
Lago, MA
Miller, WH
Ali, FE
Cousins, RD
Hall, LB
Hwang, SM
Jakas, DR
Kwon, C
Louden, C
Nguyen, TT
Ohlstein, EH
Rieman, DJ
Ross, ST
Samanen, JM
Smith, BR
Stadel, J
Takata, DT
Vickery, L
Yuan, CCK
Yue, TL
Citation: Rm. Keenan et al., Discovery of an imidazopyridine-containing 1,4-benzodiazepine nonpeptide vitronectin receptor (alpha v beta 3) antagonist with efficacy in a restenosis model, BIOORG MED, 8(22), 1998, pp. 3171-3176