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Results: 1-13 |
Results: 13
Synthesis and receptor binding affinity of new selective GluR5 ligands
Authors: Bunch, L Johansen, TH Brauner-Osborne, H Stensbol, TB Johansen, TN Krogsgaard-Larsen, P Madsen, U
Citation: L. Bunch et al., Synthesis and receptor binding affinity of new selective GluR5 ligands, BIO MED CH, 9(4), 2001, pp. 875-879
Resolution, configurational assignment, and enantiopharmacology at glutamate receptors of 2-amino-3-(3-carboxy-5-methyl-4-isoxazolyl)propionic acid (ACPA) and demethyl-ACPA
Authors: Johansen, TN Stensbol, TB Nielsen, B Vogensen, SB Frydenvang, K Slok, FA Brauner-Osborne, H Madsen, U Krogsgaard-Larsen, P
Citation: Tn. Johansen et al., Resolution, configurational assignment, and enantiopharmacology at glutamate receptors of 2-amino-3-(3-carboxy-5-methyl-4-isoxazolyl)propionic acid (ACPA) and demethyl-ACPA, CHIRALITY, 13(9), 2001, pp. 523-532
A convenient synthesis of 4-substituted 3-ethoxy-5-methylisoxazoles by palladium-catalyzed coupling reactions
Authors: Kromann, H Slok, FA Johansen, TN Krogsgaard-Larsen, P
Citation: H. Kromann et al., A convenient synthesis of 4-substituted 3-ethoxy-5-methylisoxazoles by palladium-catalyzed coupling reactions, TETRAHEDRON, 57(11), 2001, pp. 2195-2201
Synthesis and pharmacology of 3-isoxazolol amino acids as selective antagonists at group I metabotropic glutamic acid receptors
Authors: Madsen, U Brauner-Osborne, H Frydenvang, K Hvene, L Johansen, TN Nielsen, B Sanchez, C Stensbol, TB Bischoff, F Krogsgaard-Larsen, P
Citation: U. Madsen et al., Synthesis and pharmacology of 3-isoxazolol amino acids as selective antagonists at group I metabotropic glutamic acid receptors, J MED CHEM, 44(7), 2001, pp. 1051-1059
Stereochemistry and molecular pharmacology of (S)-thio-ATPA, a new potent and selective GluR5 agonist
Authors: Stensbol, TB Jensen, HS Nielsen, B Johansen, TN Egebjerg, J Frydenvang, K Krogsgaard-Larsen, P
Citation: Tb. Stensbol et al., Stereochemistry and molecular pharmacology of (S)-thio-ATPA, a new potent and selective GluR5 agonist, EUR J PHARM, 411(3), 2001, pp. 245-253
Resolution, configurational assignment, and enantiopharmacology of 2-amino-3-[3-hydroxy-5-(2-methyl-2H-tetrazol-5-yl)isoxazol-4-yl]propionic acid, a potent GluR3-and GluR4-preferring AMPA receptor agonist
Authors: Vogensen, SB Jensen, HS Stensbol, TB Frydenvang, K Bang-Andersen, B Johansen, TN Egebjerg, J Krogsgaard-Larsen, P
Citation: Sb. Vogensen et al., Resolution, configurational assignment, and enantiopharmacology of 2-amino-3-[3-hydroxy-5-(2-methyl-2H-tetrazol-5-yl)isoxazol-4-yl]propionic acid, a potent GluR3-and GluR4-preferring AMPA receptor agonist, CHIRALITY, 12(10), 2000, pp. 705-713
A new structural class of subtype-selective inhibitor of cloned excitatoryamino acid transporter, EAAT2
Authors: Brauner-Osborne, H Hermit, MB Nielsen, B Krogsgaard-Larsen, P Johansen, TN
Citation: H. Brauner-osborne et al., A new structural class of subtype-selective inhibitor of cloned excitatoryamino acid transporter, EAAT2, EUR J PHARM, 406(1), 2000, pp. 41-44
Resolution, absolute stereochemistry, and enantiopharmacology of the GluR1-4 and GluR5 antagonist 2-amino-3-[5-tert-butyl-3-(phosphonomethoxy)-4-isoxazolyl]propionic acid
Authors: Moller, EH Egebjerg, J Brehm, L Stensbol, TB Johansen, TN Madsen, U Krogsgaard-Larsen, P
Citation: Eh. Moller et al., Resolution, absolute stereochemistry, and enantiopharmacology of the GluR1-4 and GluR5 antagonist 2-amino-3-[5-tert-butyl-3-(phosphonomethoxy)-4-isoxazolyl]propionic acid, CHIRALITY, 11(10), 1999, pp. 752-759
Synthesis of deuterium and tritium labelled (RS)-2-amino-3-(5-tert-butyl-3-hydroxy-4-isoxazolyl) propionic acid (ATPA), a selective kainic acid receptor agonist
Authors: Johansen, TN Hawes, CR Ellis, GJ Ebert, B Stensbol, TB Thrige, DD Krogsgaard-Larsen, P
Citation: Tn. Johansen et al., Synthesis of deuterium and tritium labelled (RS)-2-amino-3-(5-tert-butyl-3-hydroxy-4-isoxazolyl) propionic acid (ATPA), a selective kainic acid receptor agonist, J LABEL C R, 42(10), 1999, pp. 937-947
3-Pyrazolone analogues of the 3-isoxazolol metabotropic excitatory amino acid receptor agonist homo-AMPA. Synthesis and pharmacological testing
Authors: Zimmermann, D Janin, YL Brehm, L Brauner-Osborne, H Ebert, B Johansen, TN Madsen, U Krogsgaard-Larsen, P
Citation: D. Zimmermann et al., 3-Pyrazolone analogues of the 3-isoxazolol metabotropic excitatory amino acid receptor agonist homo-AMPA. Synthesis and pharmacological testing, EUR J MED C, 34(11), 1999, pp. 967-976
Synthesis and pharmacology of the baclofen homologues 5-amino-4-(4-chlorophenyl)pentanoic acid and the R- and S-enantiomers of 5-amino-3-(4-chlorophenyl)pentanoic acid
Authors: Karla, R Ebert, B Thorkildsen, C Herdeis, C Johansen, TN Nielsen, B Krogsgaard-Larsen, P
Citation: R. Karla et al., Synthesis and pharmacology of the baclofen homologues 5-amino-4-(4-chlorophenyl)pentanoic acid and the R- and S-enantiomers of 5-amino-3-(4-chlorophenyl)pentanoic acid, J MED CHEM, 42(11), 1999, pp. 2053-2059
Resolution, absolute stereochemistry and molecular pharmacology of the enantiomers of ATPA
Authors: Stensbol, TB Borre, L Johansen, TN Egebjerg, J Madsen, U Ebert, B Krogsgaard-Larsen, P
Citation: Tb. Stensbol et al., Resolution, absolute stereochemistry and molecular pharmacology of the enantiomers of ATPA, EUR J PHARM, 380(2-3), 1999, pp. 153-162
Multiple conformations of an intercalated (-)-(7S,8R,9S,10R)-N-6-[10-(7,8,9,10-tetrahydrobenzo[a]pyrenyl)]-2 '-deoxyadenosyl adduct in the N-ras codon 61 sequence
Authors: Zegar, IS Chary, P Jabil, RJ Tamura, PJ Johansen, TN Lloyd, RS Harris, CM Harris, TM Stone, MP
Citation: Is. Zegar et al., Multiple conformations of an intercalated (-)-(7S,8R,9S,10R)-N-6-[10-(7,8,9,10-tetrahydrobenzo[a]pyrenyl)]-2 '-deoxyadenosyl adduct in the N-ras codon 61 sequence, BIOCHEM, 37(47), 1998, pp. 16516-16528
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