Citation: Ys. Choe et Ja. Katzenellenbogen, SYNTHESIS OF C-6 FLUOROANDROGENS - EVALUATION OF LIGANDS FOR TUMOR RECEPTOR IMAGING, Steroids, 60(5), 1995, pp. 414-422
Citation: Dy. Chi et al., CRYSTAL-STRUCTURE OF DOISYNOLIC ACID AND THE STRUCTURE OF OTHER PRODUCTS FORMED DURING ITS SYNTHESIS, Steroids, 60(3), 1995, pp. 261-264
Authors:
CHOE YS
LIDSTROM PJ
CHI DY
BONASERA TA
WELCH MJ
KATZENELLENBOGEN JA
Citation: Ys. Choe et al., SYNTHESIS OF 11-BETA-[F-18]FLUORO-5-ALPHA-DIHYDROTESTOSTERONE AND TA-[F-18]FLUORO-19-NOR-5-ALPHA-DIHYDROTESTOSTERONE - PREPARATION VIA HALOFLUORINATION-REDUCTION, RECEPTOR-BINDING, AND TISSUE DISTRIBUTION, Journal of medicinal chemistry, 38(5), 1995, pp. 816-825
Authors:
NAPOLITANO E
FIASCHI R
CARLSON KE
KATZENELLENBOGEN JA
Citation: E. Napolitano et al., 11-BETA-SUBSTITUTED ESTRADIOL DERIVATIVES, POTENTIAL HIGH-AFFINITY CARBON-11-LABELED PROBES FOR THE ESTROGEN-RECEPTOR - A STRUCTURE-AFFINITY RELATIONSHIP STUDY, Journal of medicinal chemistry, 38(3), 1995, pp. 429-434
Authors:
BUCKMAN BO
BONASERA TA
KIRSCHBAUM KS
WELCH MJ
KATZENELLENBOGEN JA
Citation: Bo. Buckman et al., FLUORINE-18-LABELED PROGESTIN 16A,L7A-DIOXOLANES - DEVELOPMENT OF HIGH-AFFINITY LIGANDS FOR THE PROGESTERONE-RECEPTOR WITH HIGH IN-VIVO TARGET SITE SELECTIVITY, Journal of medicinal chemistry, 38(2), 1995, pp. 328-337
Authors:
NAPOLITANO E
FIASCHI R
CARLSON KE
KATZENELLENBOGEN JA
Citation: E. Napolitano et al., 11-BETA-SUBSTITUTED ESTRADIOL DERIVATIVES .2. POTENTIAL CARBON-11-LABELED AND IODINE-LABELED PROBES FOR THE ESTROGEN-RECEPTOR, Journal of medicinal chemistry, 38(14), 1995, pp. 2774-2779
Authors:
CUSHMAN M
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KATZENELLENBOGEN JA
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Citation: M. Cushman et al., SYNTHESIS, ANTITUBULIN AND ANTIMITOTIC ACTIVITY, AND CYTOTOXICITY OF ANALOGS OF 2-METHOXYESTRADIOL, AN ENDOGENOUS MAMMALIAN METABOLITE OF ESTRADIOL THAT INHIBITS TUBULIN POLYMERIZATION BY BINDING TO THE COLCHICINE BINDING-SITE, Journal of medicinal chemistry, 38(12), 1995, pp. 2041-2049
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CHI DY
LIDSTROM PJ
CHOE YS
BONASERA TA
WELCH MJ
KATZENELLENBOGEN JA
Citation: Dy. Chi et al., BROMO[F-18]FLUORINATION OF CYCLOHEXENES - A METHOD FOR THE PREPARATION OF [F-18] FLUOROCYCLOHEXANES, Journal of fluorine chemistry, 71(1), 1995, pp. 143-147
Citation: Dy. Chi et al., CRYSTAL-STRUCTURE OF A BIS(AMIDO)BIS(THIOLATO)OXORHENIUM(V) COMPLEX THAT FORMS A METHANOL-SOLVATED SALT WITH CALCIUM EXTRACTED FROM SILICA-GEL, Inorganic chemistry, 34(6), 1995, pp. 1624-1625
Authors:
SEIELSTAD DA
CARLSON KE
KUSHNER PJ
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KATZENELLENBOGEN JA
Citation: Da. Seielstad et al., ANALYSIS OF THE STRUCTURAL CORE OF THE HUMAN ESTROGEN-RECEPTOR LIGAND-BINDING DOMAIN BY SELECTIVE PROTEOLYSIS MASS-SPECTROMETRIC ANALYSIS, Biochemistry, 34(39), 1995, pp. 12605-12615
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ONEIL JP
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Citation: Jp. Oneil et al., PROGESTIN RADIOPHARMACEUTICALS LABELED WITH TECHNETIUM AND RHENIUM - SYNTHESIS, BINDING-AFFINITY, AND IN-VIVO DISTRIBUTION OF A NEW PROGESTIN N2S2-METAL CONJUGATE, Bioconjugate chemistry, 5(3), 1994, pp. 182-193
Authors:
BERGMANN KE
CARLSON KE
KATZENELLENBOGEN JA
Citation: Ke. Bergmann et al., HEXESTROL DIAZIRINE PHOTOAFFINITY-LABELING REAGENT FOR THE ESTROGEN-RECEPTOR, Bioconjugate chemistry, 5(2), 1994, pp. 141-150
Authors:
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ROCQUE PG
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KATZENELLENBOGEN JA
Citation: Ke. Bergmann et al., OXOHEXESTROL DERIVATIVES LABELED WITH F-18 - SYNTHESIS, RECEPTOR-BINDING AND IN-VITRO DISTRIBUTION OF 2 NONSTEROIDAL ESTROGENS AS POTENTIALBREAST-TUMOR IMAGING AGENTS, Nuclear medicine and biology, 21(1), 1994, pp. 25-39
Authors:
BERGMANN KE
WOOGE CH
CARLSON KE
KATZENELLENBOGEN BS
KATZENELLENBOGEN JA
Citation: Ke. Bergmann et al., BIVALENT LIGANDS AS PROBES OF ESTROGEN-RECEPTOR ACTION, Journal of steroid biochemistry and molecular biology, 49(2-3), 1994, pp. 139-152
Authors:
BONASERA TA
ONEIL JP
CHOE YS
LICH LL
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WELCH MJ
KATZENELLENBOGEN JA
Citation: Ta. Bonasera et al., IMAGING THE PROSTATE IN BABOONS WITH F-18 LABELED ANDROGEN RECEPTOR LIGANDS, The Journal of nuclear medicine, 35(5), 1994, pp. 160000053-160000053
Authors:
DEHDASHTI F
MORTIMER JE
GRIFFETH LK
MCGUIRE AH
RADFORD DM
FUSSELMAN MJ
BURNEY RJ
BONASERA TA
SEIGEL BA
KATZENELLENBOGEN JA
WELCH MJ
Citation: F. Dehdashti et al., POSITRON TOMOGRAPHIC ASSESSMENT OF BREAST-LESIONS WITH FDG AND FES, The Journal of nuclear medicine, 35(5), 1994, pp. 160000141-160000141
Authors:
NAPOLITANO EN
DENCE CS
WELCH MJ
KATZENELLENBOGEN JA
Citation: En. Napolitano et al., C-11 LABELED ESTROGENS AS IMAGING AGENTS FOR BREAST-TUMORS, The Journal of nuclear medicine, 35(5), 1994, pp. 160000250-160000250
Authors:
KYM PR
WILSON SR
GRITTON WH
KATZENELLENBOGEN JA
Citation: Pr. Kym et al., NOVEL STEROIDS FROM CETYLTRIMETHYLAMMONIUM PERMANGANATE-INITIATED OXIDATIVE REARRANGEMENTS OF 16-DEHYDROPROGESTERONE, Tetrahedron letters, 35(18), 1994, pp. 2833-2836
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VANBROCKLIN HF
LIU AJ
WELCH MJ
ONEIL JP
KATZENELLENBOGEN JA
Citation: Hf. Vanbrocklin et al., THE SYNTHESIS OF 7-ALPHA-METHYL-SUBSTITUTED ESTROGENS LABELED WITH F-18 - POTENTIAL BREAST-TUMOR IMAGING AGENTS, Steroids, 59(1), 1994, pp. 34-45
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CHI DY
ONEIL JP
ANDERSON CJ
WELCH MJ
KATZENELLENBOGEN JA
Citation: Dy. Chi et al., HOMODIMERIC AND HETERODIMERIC BIS(AMINO THIOL) OXOMETAL COMPLEXES WITH RHENIUM(V) AND TECHNETIUM(V) - CONTROL OF HETERODIMERIC COMPLEX-FORMATION AND AN APPROACH TO METAL-COMPLEXES THAT MIMIC STEROID-HORMONES, Journal of medicinal chemistry, 37(7), 1994, pp. 928-937
Authors:
RAY S
TANDON A
DWIVEDY I
WILSON SR
ONEIL JP
KATZENELLENBOGEN JA
Citation: S. Ray et al., AN X-RAY CRYSTALLOGRAPHIC STUDY OF THE NONSTEROIDAL CONTRACEPTIVE AGENT CENTCHROMAN, Journal of medicinal chemistry, 37(5), 1994, pp. 696-700
Authors:
BUCKMAN BO
VANBROCKLIN HF
DENCE CS
BERGMANN SR
WELCH MJ
KATZENELLENBOGEN JA
Citation: Bo. Buckman et al., SYNTHESIS AND TISSUE BIODISTRIBUTION OF [OMEGA-C-11]PALMITIC ACID - ANOVEL PET IMAGING AGENT FOR CARDIAC FATTY-ACID METABOLISM, Journal of medicinal chemistry, 37(15), 1994, pp. 2481-2485
Citation: Jp. Oneil et al., PREPARATION AND STRUCTURAL CHARACTERIZATION OF MONOAMINE-MONOAMIDE BIS(THIOL) OXO COMPLEXES OF TECHNETIUM(V) AND RHENIUM(V), Inorganic chemistry, 33(2), 1994, pp. 319-323
Authors:
KATZENELLENBOGEN JA
MATHIAS CJ
VANBROCKLIN HF
BRODACK JW
WELCH MJ
Citation: Ja. Katzenellenbogen et al., TITRATION OF THE IN-VIVO UPTAKE OF 16-ALPHA-F-18!FLUOROESTRADIOL BY TARGET TISSUES IN THE RAT - COMPETITION BY TAMOXIFEN, AND IMPLICATIONSFOR QUANTITATING ESTROGEN-RECEPTORS IN-VIVO AND THE USE OF ANIMAL-MODELS IN RECEPTOR-BINDING RADIOPHARMACEUTICAL DEVELOPMENT, Nuclear medicine and biology, 20(6), 1993, pp. 735-745
Citation: Mj. Kochanny et al., SYNTHESIS AND NMR-SPECTRUM OF [C-13(18)]-MESO-HEXESTROL, A FULLY C-13SUBSTITUTED LIGAND FOR NMR-STUDIES OF THE ESTROGEN-RECEPTOR, Magnetic resonance in chemistry, 31(11), 1993, pp. 977-986