Authors:
SALL DJ
BRIGGS SL
CHIRGADZE NY
CLAWSON DK
GIFFORDMOORE DS
KLIMKOWSKI VJ
MCCOWAN JR
SMITH GF
WIKEL JH
Citation: Dj. Sall et al., DIBASIC BENZO[B]THIOPHENE DERIVATIVES AS A NOVEL CLASS OF ACTIVE-SITE-DIRECTED THROMBIN INHIBITORS - 2 - EXPLORING INTERACTIONS AT THE PROXIMAL (S-2) BINDING-SITE, Bioorganic & medicinal chemistry letters, 8(18), 1998, pp. 2527-2532
Authors:
CHIRGADZE NY
SALL DJ
KLIMKOWSKI VJ
CLAWSON DK
BRIGGS SL
HERMANN R
SMITH GF
GIFFORDMOORE DS
WERY JP
Citation: Ny. Chirgadze et al., THE CRYSTAL-STRUCTURE OF HUMAN ALPHA-THROMBIN COMPLEXED WITH LY178550, A NONPEPTIDYL, ACTIVE-SITE-DIRECTED INHIBITOR, Protein science, 6(7), 1997, pp. 1412-1417
Authors:
SALL DJ
BASTIAN JA
BRIGGS SL
BUBEN JA
CHIRGADZE NY
CLAWSON DK
DENNEY ML
GIERA DD
GIFFORDMOORE DS
HARPER RW
HAUSER KL
KLIMKOWSKI VJ
KOHN TJ
LIN HS
MCCOWAN JR
PALKOWITZ AD
SMITH GF
TAKEUCHI K
THRASHER KJ
TINSLEY JM
UTTERBACK BG
YAN SCB
ZHANG MS
Citation: Dj. Sall et al., DIBASIC BENZO[B]THIOPHENE DERIVATIVES AS A NOVEL CLASS OF ACTIVE-SITE-DIRECTED THROMBIN INHIBITORS .1. DETERMINATION OF THE SERINE-PROTEASESELECTIVITY, STRUCTURE-ACTIVITY-RELATIONSHIPS, AND BINDING ORIENTATION, Journal of medicinal chemistry, 40(22), 1997, pp. 3489-3493
Authors:
XIA JL
DUBIN PL
KIM Y
MUHOBERAC BB
KLIMKOWSKI VJ
Citation: Jl. Xia et al., ELECTROPHORETIC AND QUASI-ELASTIC LIGHT-SCATTERING OF SOLUBLE-PROTEINPOLYELECTROLYTE COMPLEXES, Journal of physical chemistry, 97(17), 1993, pp. 4528-4534