Citation: E. Kostenis et al., FUNCTIONAL-CHARACTERIZATION OF A SERIES OF MUTANT G-PROTEIN ALPHA(Q) SUBUNITS DISPLAYING PROMISCUOUS RECEPTOR COUPLING PROPERTIES, The Journal of biological chemistry, 273(28), 1998, pp. 17886-17892
Citation: E. Kostenis et al., IMPORTANCE OF THE AMINO-TERMINAL EXTENSION OF G-ALPHA-Q IN RECEPTOR G-PROTEIN COUPLING SPECIFICITY/, The FASEB journal, 11(9), 1997, pp. 1137-1137
Citation: C. Trankle et al., G-PROTEIN COUPLING SPECIFICITY AND SENSITIVITY TOWARDS ALLOSTERIC MODULATION OF MUSCARINIC M-2 AND M-3 RECEPTORS, Naunyn-Schmiedeberg's archives of pharmacology, 355(4), 1997, pp. 63-63
Authors:
WESS J
LIU J
BLIN N
YUN J
LERCHE C
KOSTENIS E
Citation: J. Wess et al., STRUCTURAL BASIS OF RECEPTOR G-PROTEIN COUPLING SELECTIVITY STUDIED WITH MUSCARINIC RECEPTORS AS MODEL SYSTEMS, Life sciences, 60(13-14), 1997, pp. 1007-1014
Citation: E. Kostenis et al., GENETIC-ANALYSIS OF RECEPTOR-G-ALPHA(Q) COUPLING SELECTIVITY, The Journal of biological chemistry, 272(38), 1997, pp. 23675-23681
Authors:
KOSTENIS E
DEGTYAREV MY
CONKLIN BR
WESS J
Citation: E. Kostenis et al., THE N-TERMINAL EXTENSION OF G-ALPHA(Q) IS CRITICAL FOR CONSTRAINING THE SELECTIVITY OF RECEPTOR COUPLING, The Journal of biological chemistry, 272(31), 1997, pp. 19107-19110
Citation: E. Kostenis et al., MOLECULAR-BASIS OF RECEPTOR G PROTEIN COUPLING SELECTIVITY STUDIED BYCOEXPRESSION OF WILD-TYPE AND MUTANT M2 MUSCARINIC RECEPTORS WITH MUTANT G-ALPHA(Q) SUBUNITS/, Biochemistry, 36(6), 1997, pp. 1487-1495
Citation: E. Kostenis et K. Mohr, 2-POINT KINETIC-EXPERIMENTS TO QUANTIFY ALLOSTERIC EFFECTS ON RADIOLIGAND DISSOCIATION, Trends in pharmacological sciences, 17(8), 1996, pp. 280-283
Citation: C. Trankle et al., SEARCH FOR LEAD STRUCTURES TO DEVELOP NEW ALLOSTERIC MODULATORS OF MUSCARINIC RECEPTORS, The Journal of pharmacology and experimental therapeutics, 279(2), 1996, pp. 926-933
Citation: E. Kostenis et al., EVIDENCE FOR A MULTIPLE BINDING MODE OF BISPYRIDINIUM-TYPE ALLOSTERICMODULATORS OF MUSCARINIC RECEPTORS, European journal of pharmacology, 314(3), 1996, pp. 385-392
Authors:
GASTEIGER J
HOLZGRABE U
KOSTENIS E
MOHR K
SURIG U
WAGENER M
Citation: J. Gasteiger et al., VARIATION OF THE OXIME FUNCTION OF BISPYRIDINIUM-TYPE ALLOSTERIC MODULATORS OF M(2)-CHOLINOCEPTORS, Die Pharmazie, 50(2), 1995, pp. 99-105
Citation: A. Maass et al., POTENTIATION OF THE ACTION OF N-METHYLSCOPOLAMINE IN GUINEA-PIG ATRIABY THE ALLOSTERIC ANTAGONISTS TETRA-W84, W84, AND ALCURONIUM, Life sciences, 56(11-12), 1995, pp. 1008-1008
Citation: E. Kostenis et al., SIDE-CHAIN VARIATIONS IN BISPYRIDINIUM-TYPE ALLOSTERIC MODULATORS OF M(2)-CHOLINOCEPTORS, Life sciences, 56(11-12), 1995, pp. 1009-1009
Citation: A. Maass et al., POTENTIATION BY ALCURONIUM OF THE ANTIMUSCARINIC EFFECT OF N-METHYLSCOPOLAMINE IN GUINEA-PIG LEFT ATRIA, European journal of pharmacology, 272(1), 1995, pp. 103-106
Authors:
PFAFFENDORF M
BATINK HD
KOSTENIS E
TRANKLE C
MOHR K
VANZWIETEN PA
Citation: M. Pfaffendorf et al., INFLUENCE OF W84, AN ALLOSTERIC MODULAR OF MUSCARINIC M2-RECEPTORS, ON THE DISSOCIATION CHARACTERISTICS OF [3H]PRAZOSIN AND [I-125] IODOCYANO-PINDOLOL IN RAT CARDIAC TISSUES, British Journal of Pharmacology, 114, 1995, pp. 436-436
Citation: E. Kostenis et al., ALLOSTERIC EFFECT ON MUSCARINIC M(2)-RECEPTORS OF DERIVATIVES OF THE ALKANE-BIS-AMMONIUM COMPOUND W84 - COMPARISON WITH BISPYRIDINIUM TYPE ALLOSTERIC MODULATORS, European journal of medicinal chemistry, 29(12), 1994, pp. 947-953
Authors:
CID MHB
HOLZGRABE U
KOSTENIS E
MOHR K
TRANKLE C
Citation: Mhb. Cid et al., SEARCH FOR THE PHARMACOPHORE OF BISPYRIDINIUM-TYPE ALLOSTERIC MODULATORS OF MUSCARINIC RECEPTORS, Journal of medicinal chemistry, 37(10), 1994, pp. 1439-1445