Authors:
CINOTTI L
LEBARS D
GARCIALARREA L
PEYRON R
GREGOIRE MC
LAVENNE F
KROGSGAARDLARSEN P
COMAR D
MAUGUIERE F
Citation: L. Cinotti et al., GABA-A STIMULATION IN NORMAL VOLUNTEERS A ND DURING TEMPORAL EPILEPSYMEASURED BY (18)FDG WITH POSITRON EMISSION TOMOGRAPHY, Journal de chimie physique et de physico-chimie biologique, 93(1), 1996, pp. 48-52
Authors:
SOKILDE B
MIKKELSEN I
STENSBOL TB
ANDERSEN B
EBDRUP S
KROGSGAARDLARSEN P
FALCH E
Citation: B. Sokilde et al., ANALOGS OF CARBACHOLINE - SYNTHESIS AND RELATIONSHIP BETWEEN STRUCTURE AND AFFINITY FOR MUSCARINIC AND NICOTINIC ACETYLCHOLINE-RECEPTORS, Archiv der pharmazie, 329(2), 1996, pp. 95-104
Authors:
JOHANSEN TN
BALASUBRAMANIAN V
MADSEN U
FERKANY JW
KROGSGAARDLARSEN P
Citation: Tn. Johansen et al., SYNTHESIS OF TRITIATED -2-AMINO-2-(3-HYDROXY-5-METHYLISOXAZOL-4-YL)ACETIC ACID (AMAA), A POTENT AND SELECTIVE NMDA AGONIST, Journal of labelled compounds & radiopharmaceuticals, 38(10), 1996, pp. 915-922
Authors:
KROGSGAARDLARSEN P
EBERT B
LUND TM
BRAUNEROSBORNE H
SLOK FA
JOHANSEN TN
BREHM L
MADSEN U
Citation: P. Krogsgaardlarsen et al., DESIGN OF EXCITATORY AMINO-ACID RECEPTOR AGONISTS, PARTIAL AGONISTS AND ANTAGONISTS - IBOTENIC ACID AS A KEY LEAD STRUCTURE, European journal of medicinal chemistry, 31(7-8), 1996, pp. 515-537
Authors:
EBERT B
MADSEN U
SOBY KK
KROGSGAARDLARSEN P
Citation: B. Ebert et al., FUNCTIONAL PARTIAL AGONISM AT IONOTROPIC EXCITATORY AMINO-ACID RECEPTORS, Neurochemistry international, 29(3), 1996, pp. 309-316
Authors:
MADSEN U
BANGANDERSEN B
BREHM L
CHRISTENSEN IT
EBERT B
KRISTOFFERSEN ITS
LANG Y
KROGSGAARDLARSEN P
Citation: U. Madsen et al., SYNTHESIS AND PHARMACOLOGY OF HIGHLY SELECTIVE CARBOXY AND PHOSPHONO ISOXAZOLE AMINO-ACID AMPA RECEPTOR ANTAGONISTS, Journal of medicinal chemistry, 39(8), 1996, pp. 1682-1691
Authors:
JAROSZEWSKI JW
MATZEN L
FROLUND B
KROGSGAARDLARSEN P
Citation: Jw. Jaroszewski et al., NEUROACTIVE POLYAMINE WASP TOXINS - NUCLEAR-MAGNETIC-RESONANCE SPECTROSCOPIC ANALYSIS OF THE PROTOLYTIC PROPERTIES OF PHILANTHOTOXIN-343, Journal of medicinal chemistry, 39(2), 1996, pp. 515-521
Authors:
BRAUNEROSBORNE H
SLOK FA
SKJAERBAEK N
EBERT B
SEKIYAMA N
NAKANISHI S
KROGSGAARDLARSEN P
Citation: H. Braunerosborne et al., A NEW HIGHLY SELECTIVE METABOTROPIC EXCITATORY AMINO-ACID AGONIST - 2-AMINO-4-(3-HYDROXY-5-METHYLISOXAZOL-4-YL)BUTYRIC ACID, Journal of medicinal chemistry, 39(16), 1996, pp. 3188-3194
Authors:
MADSEN U
FRYDENVANG K
EBERT B
JOHANSEN TN
BREHM L
KROGSGAARDLARSEN P
Citation: U. Madsen et al., N-METHYL-D-ASPARTIC ACID RECEPTOR AGONISTS - RESOLUTION, ABSOLUTE STEREOCHEMISTRY, AND PHARMACOLOGY OF THE ENANTIOMERS OF 2-AMINO-2-(3-HYDROXY-5-METHYL-4-ISOXAZOLYL)ACETIC ACID, Journal of medicinal chemistry, 39(1), 1996, pp. 183-190
Authors:
BRAUNEROSBORNE H
EBERT B
BRANN MR
FALCH E
KROGSGAARDLARSEN P
Citation: H. Braunerosborne et al., FUNCTIONAL PARTIAL AGONISM AT CLONED HUMAN MUSCARINIC ACETYLCHOLINE-RECEPTORS, European journal of pharmacology, 313(1-2), 1996, pp. 145-150
Authors:
WAHL P
MADSEN U
BANKE T
KROGSGAARDLARSEN P
SCHOUSBOE A
Citation: P. Wahl et al., DIFFERENT CHARACTERISTICS OF AMPA RECEPTOR AGONISTS ACTING AT AMPA RECEPTORS EXPRESSED IN XENOPUS OOCYTES, European journal of pharmacology, 308(2), 1996, pp. 211-218
Authors:
NIELSEN M
WITT MR
EBERT B
KROGSGAARDLARSEN P
Citation: M. Nielsen et al., THIOMUSCIMOL, A NEW PHOTOAFFINITY LABEL FOR THE GABA(A) RECEPTOR, European journal of pharmacology. Molecular pharmacology section, 289(1), 1995, pp. 109-112
Authors:
FRYDENVANG K
KRISTIANSEN U
FROLUND B
HERDEIS C
KROGSGAARDLARSEN P
Citation: K. Frydenvang et al., GABA(B) ANTAGONISTS - ENANTIOPHARMACOLOGY OF 5-AMINO-4-HYDROXY-2-METHYLVALERIC ACID AND X-RAY STRUCTURE OF THE EUTOMER, Chirality, 7(7), 1995, pp. 526-533
Authors:
FROLUND B
JEPPESEN L
KROGSGAARDLARSEN P
HANSEN JJ
Citation: B. Frolund et al., GABA(A) AGONISTS - RESOLUTION AND PHARMACOLOGY OF (-ISOGUVACINE AND (-)-ISOGUVACINE OXIDE()), Chirality, 7(6), 1995, pp. 434-438
Authors:
FROLUND B
EBERT B
LAWRENCE LW
HURT SD
KROGSGAARDLARSEN P
Citation: B. Frolund et al., SYNTHESIS AND RECEPTOR-BINDING OF 5-AMINO[H-3](2)METHYL-3-ISOTHIAZOLOL ([H-3]THIOMUSCIMOL), A SPECIFIC GABA(A) AGONIST PHOTOAFFINITY LABEL, Journal of labelled compounds & radiopharmaceuticals, 36(9), 1995, pp. 877-889
Citation: B. Ebert et al., KETOBEMIDONE, METHADONE AND PETHIDINE ARE NONCOMPETITIVE N-METHYL-D-ASPARTATE (NMDA) ANTAGONISTS IN THE RAT CORTEX AND SPINAL-CORD, Neuroscience letters, 187(3), 1995, pp. 165-168
Authors:
SKJAERBAEK N
EBERT B
FALCH E
BREHM L
KROGSGAARDLARSEN P
Citation: N. Skjaerbaek et al., EXCITATORY AMINO-ACIDS - SYNTHESIS OF -3-(5-CYCLOPROPYL-3-HYDROXYISOXAZOL-4-YL)PROPIONIC ACID, A NEW POTENT AND SPECIFIC AMPA RECEPTOR AGONIST, Journal of the Chemical Society. Perkin transactions. I, (3), 1995, pp. 221-225
Authors:
LENZ SM
MEIER E
PEDERSEN H
FREDERIKSEN K
BOGESO KP
KROGSGAARDLARSEN P
Citation: Sm. Lenz et al., MUSCARINIC AGONISTS - SYNTHESES AND STRUCTURE-ACTIVITY-RELATIONSHIPS OF BICYCLIC ISOXAZOLE ESTER BIOISOSTERES OF NORARECOLINE, European journal of medicinal chemistry, 30(4), 1995, pp. 263-270
Authors:
JORGENSEN HB
EBERT B
KROGSGAARDLARSEN P
BRANN MR
FALCH E
Citation: Hb. Jorgensen et al., MOLECULAR PHARMACOLOGY OF O-ALKYL-THAO COMPOUNDS USING THE 5 CLONED MUSCARINIC ACETYLCHOLINE-RECEPTORS, Life sciences, 56(11-12), 1995, pp. 1007-1007
Citation: P. Krogsgaardlarsen, STRUCTURAL AND MOLECULAR PHARMACOLOGICAL STUDIES OF GABA-B RECEPTOR LIGANDS, Journal of neurochemistry, 65, 1995, pp. 61-61
Citation: J. Kardos et al., INTERACTIONS BETWEEN GABA-A AND GABA-B RECEPTORS IN CEREBELLAR GRANULE CELLS - DISINHIBITION AT THE CELLULAR-LEVEL, Journal of neurochemistry, 65, 1995, pp. 62-62
Authors:
FROLUND B
KRISTIANSEN U
BREHM L
HANSEN AB
KROGSGAARDLARSEN P
FALCH E
Citation: B. Frolund et al., PARTIAL GABA(A) RECEPTOR AGONISTS - SYNTHESIS AND IN-VITRO PHARMACOLOGY OF A SERIES OF NONANNULATED ANALOGS OF 4,5,6,7-TETRAHYDROISOXAZOLO[5,4-C]PYRIDIN-3-OL, Journal of medicinal chemistry, 38(17), 1995, pp. 3287-3296
Authors:
BRAUNEROSBORNE H
EBERT B
BRANN MR
FALCH E
KROGSGAARDLARSEN P
Citation: H. Braunerosborne et al., ANNULATED HETEROCYCLIC BIOISOSTERES OF NORARECOLINE - SYNTHESIS AND MOLECULAR PHARMACOLOGY AT 5 RECOMBINANT HUMAN MUSCARINIC ACETYLCHOLINE-RECEPTORS, Journal of medicinal chemistry, 38(12), 1995, pp. 2188-2195
Authors:
ARNT J
SANCHEZ C
LENZ SM
MADSEN U
KROGSGAARDLARSEN P
Citation: J. Arnt et al., DIFFERENTIATION OF IN-VIVO EFFECTS OF AMPA AND NMDA RECEPTOR LIGANDS USING DRUG DISCRIMINATION METHODS AND CONVULSANT ANTICONVULSANT ACTIVITY/, European journal of pharmacology, 285(3), 1995, pp. 289-297