Authors:
Ichikawa, T
Kitazaki, T
Matsushita, Y
Yamada, M
Hayashi, R
Yamaguchi, M
Kiyota, Y
Okonogi, K
Itoh, K
Citation: T. Ichikawa et al., Optically active antifungal azoles. XII. Synthesis and antifungal activityof the water-soluble prodrugs of 1-[(1R,2R)-2-(2,4-Difluorophenyl)-2-hydroxy-1-methyl-3-(1H-1,2,4-triazol-1-yl)propyl]-3-[4-(1H-1-tetrazolyl)phenyl]-2-imidazolidinone, CHEM PHARM, 49(9), 2001, pp. 1102-1109
Authors:
Ichikawa, T
Yamada, M
Yamaguchi, M
Kitazaki, T
Matsushita, Y
Higashikawa, K
Itoh, K
Citation: T. Ichikawa et al., Optically active antifungal azoles. XIII. Synthesis of stereoisomers and metabolites of 1-[(1R,2R)-2-(2,4-difluorophenyl)-2-hydroxy-1-methyl-3(1H-1,2,4-triazol-1-yl)propyl]-3-[4-(1H-1-tetrazolyl)phenyl]-2-imidazolidinone (TAK-456), CHEM PHARM, 49(9), 2001, pp. 1110-1119
Authors:
Kitazaki, T
Ichikawa, T
Tasaka, A
Hosono, H
Matsushita, Y
Hayashi, R
Okonogi, K
Itoh, K
Citation: T. Kitazaki et al., Optically active antifungal azoles. X. Synthesis and antifungal activity of N-[4-(azolyl)phenyl]- and N-[4-(azolylmethyl)phenyl]-N '-[(1R,2R)-2-(2,4-difluorophenyl)-2-hydroxy-1-methyl-3-(1H-1,2,4-triazol-1-yl)propyl]-azolones, CHEM PHARM, 48(12), 2000, pp. 1935-1946
Authors:
Ichikawa, T
Kitazaki, T
Matsushita, Y
Hosono, H
Yamada, M
Mizuno, M
Itoh, K
Citation: T. Ichikawa et al., Optically active antifungal azoles. XI. An alternative synthetic route for1-[(1R,2R)-2-(2,4-difluarophenyl)-2-hydroxy-1-methyl-3-(1H-1,2,4-triazol-1-yl)propyl]-3-[4-(1H-1-tetrazolyl)phenyl]-2-imidazolidinone (TAK-456) and its analog, CHEM PHARM, 48(12), 2000, pp. 1947-1953
Authors:
Kitazaki, T
Tasaka, A
Hosono, H
Matsushita, Y
Itoh, K
Citation: T. Kitazaki et al., Optically active antifungal azoles. VIII. Synthesis and antifungal activity of 1-[(1R,2R)-2-(2,4-difluoro- and 2-fluorophenyl)-2-hydroxy-1-methyl-3-(1H-1,2,4-triazol-1-yl)propyl]-3-(4-substituted phenyl)-2(1H,3H)-imidazolones and 2-imidazolidinones, CHEM PHARM, 47(3), 1999, pp. 351-359
Authors:
Kitazaki, T
Tasaka, A
Hosono, H
Matsushita, Y
Itoh, K
Citation: T. Kitazaki et al., Optically active antifungal azoles. IX. An alternative synthetic route for2-[(1R,2R)-2-(2,4-difluorophenyl)-2-hydroxy-1-methyl-3-(1H-1,2,4-triazol-1-yl)propyl]-4-[4-(2,2,3,3-tetrafluoropropoxy)phenyl]-3(2H,4H)-1,2,4-triazolone and its analogs, CHEM PHARM, 47(3), 1999, pp. 360-368