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LUESSEN HL
DELEEUW BJ
DEBOER BG
VERHOEF JC
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Citation: Af. Kotze et al., COMPARISON OF THE EFFECT OF DIFFERENT CHITOSAN SALTS AND N-TRIMETHYL CHITOSAN CHLORIDE ON THE PERMEABILITY OF INTESTINAL EPITHELIAL-CELLS (CACO-2), Journal of controlled release, 51(1), 1998, pp. 35-46
Authors:
KOTZE AF
LUESSEN HL
DELEEUW BJ
DEBOER BG
VERHOEF JC
JUNGINGER HE
Citation: Af. Kotze et al., N-TRIMETHYL CHITOSAN CHLORIDE AS A POTENTIAL ABSORPTION ENHANCER ACROSS MUCOSAL SURFACES - IN-VITRO EVALUATION IN INTESTINAL EPITHELIAL-CELLS (CACO-2), Pharmaceutical research, 14(9), 1997, pp. 1197-1202
Authors:
KOTZE AF
DELEEUW BJ
LUESSEN HL
DEBOER AG
VERHOEF JC
JUNGINGER HE
Citation: Af. Kotze et al., CHITOSANS FOR ENHANCED DELIVERY OF THERAPEUTIC PEPTIDES ACROSS INTESTINAL EPITHELIA - IN-VITRO EVALUATION IN CACO-2 CELL MONOLAYERS, International journal of pharmaceutics, 159(2), 1997, pp. 243-253
Authors:
LUESSEN HL
RENTEL CO
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DEBOER AG
VERHOEF JC
JUNGINGER HE
Citation: Hl. Luessen et al., MUCOADHESIVE POLYMERS IN PERORAL PEPTIDE DRUG-DELIVERY .4. POLYCARBOPHIL AND CHITOSAN ARE POTENT ENHANCERS OF PEPTIDE-TRANSPORT ACROSS INTESTINAL MUCOSAE IN-VITRO, Journal of controlled release, 45(1), 1997, pp. 15-23
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LUESSEN HL
LEHR CM
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JUNGINGER HE
Citation: F. Kaiho et al., DISINTEGRATION AND GEL-FORMING BEHAVIOR OF CARBOMER AND ITS SODIUM-SALT USED AS EXCIPIENTS FOR DIRECT COMPRESSION, STP pharma sciences, 6(6), 1996, pp. 385-389
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VERHOEF JC
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Citation: Hl. Luessen et al., MUCOADHESIVE POLYMERS IN PERORAL PEPTIDE DRUG-DELIVERY .1. INFLUENCE OF MUCOADHESIVE EXCIPIENTS ON THE PROTEOLYTIC ACTIVITY OF INTESTINAL ENZYMES, European journal of pharmaceutical sciences, 4(2), 1996, pp. 117-128
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DELEEUW BJ
LANGEMEYER MWE
DEBOER AG
VERHOEF JC
JUNGINGER HE
Citation: Hl. Luessen et al., MUCOADHESIVE POLYMERS IN PERORAL PEPTIDE DRUG-DELIVERY .6. CARBOMER AND CHITOSAN IMPROVE THE INTESTINAL-ABSORPTION OF THE PEPTIDE DRUG BUSERELIN IN-VIVO, Pharmaceutical research, 13(11), 1996, pp. 1668-1672
Authors:
LUESSEN HL
BOHNER V
PERARD D
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VERHOEF JC
DEBOER AG
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JUNGINGER HE
Citation: Hl. Luessen et al., MUCOADHESIVE POLYMERS IN PERORAL PEPTIDE DRUG-DELIVERY .5. EFFECT OF POLY(ACRYLATES) ON THE ENZYMATIC DEGRADATION OF PEPTIDE DRUGS BY INTESTINAL BRUSH-BORDER MEMBRANE-VESICLES, International journal of pharmaceutics, 141(1-2), 1996, pp. 39-52
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AKIYAMA Y
LUESSEN HL
DEBOER AG
VERHOEF JC
JUNGINGER HE
Citation: Y. Akiyama et al., NOVEL PERORAL DOSAGE FORMS WITH PROTEASE INHIBITORY ACTIVITIES .2. DESIGN OF FAST DISSOLVING POLY(ACRYLATE) AND CONTROLLED DRUG-RELEASING CAPSULE FORMULATIONS WITH TRYPSIN INHIBITING PROPERTIES, International journal of pharmaceutics, 138(1), 1996, pp. 13-23
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AKIYAMA Y
LUESSEN HL
DEBOER AG
VERHOEF JC
JUNGINGER HE
Citation: Y. Akiyama et al., NOVEL PERORAL DOSAGE FORMS WITH PROTEASE INHIBITORY ACTIVITIES .1. DESIGN OF CAPSULES WITH FAST GEL-FORMING AND FAST DRUG-RELEASING PROPERTIES, International journal of pharmaceutics, 136(1-2), 1996, pp. 155-163
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LUESSEN HL
DEBOER AG
VERHOEF JC
LEHR CM
JUNGINGER HE
Citation: G. Borchard et al., THE POTENTIAL OF MUCOADHESIVE POLYMERS IN ENHANCING INTESTINAL PEPTIDE DRUG ABSORPTION .3. EFFECTS OF CHITOSAN-GLUTAMATE AND CARBOMER ON EPITHELIAL TIGHT JUNCTIONS IN-VITRO, Journal of controlled release, 39(2-3), 1996, pp. 131-138
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LUESSEN HL
VERHOEF JC
BORCHARD G
LEHR CM
DEBOER AG
JUNGINGER HE
Citation: Hl. Luessen et al., MUCOADHESIVE POLYMERS IN PERORAL PEPTIDE DRUG-DELIVERY .2. CARBOMER AND POLYCARBOPHIL ARE POTENT INHIBITORS OF THE INTESTINAL PROTEOLYTIC-ENZYME TRYPSIN, Pharmaceutical research, 12(9), 1995, pp. 1293-1298
Authors:
LUESSEN HL
NOACH ABJ
DEBOER AG
VERHOEF JC
JUNGINGER HE
Citation: Hl. Luessen et al., EFFECT OF POLYCARBOPHIL ON THE PARACELLULAR PERMEABILITY OF A HYDROPHILIC MODEL-COMPOUND AFTER APPLICATION ON A CACO-2 CELL-LINE, Journal of controlled release, 28(1-3), 1994, pp. 288-288
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LUESSEN HL
VERHOEF JC
LEHR CM
DEBOER AG
JUNGINGER HE
Citation: Hl. Luessen et al., 2 DERIVATIVES OF POLY(ACRYLIC ACID) ARE ABLE 2 INHIBIT TRYPSIN ACTIVITY, Journal of controlled release, 28(1-3), 1994, pp. 316-316