Authors:
LUM RT
NELSON MG
JOLY A
HORSMA AG
LEE G
MEYER SM
WICK MM
SCHOW SR
Citation: Rt. Lum et al., SELECTIVE-INHIBITION OF THE CHYMOTRYPSIN-LIKE ACTIVITY OF THE 20S PROTEASOME BY 5-METHOXY-1-INDANONE DIPEPTIDE BENZAMIDES, Bioorganic & medicinal chemistry letters, 8(3), 1998, pp. 209-214
Authors:
LUM RT
KERWAR SS
MEYER SM
NELSON MG
SCHOW SR
SHIFFMAN D
WICK MM
JOLY A
Citation: Rt. Lum et al., A NEW STRUCTURAL CLASS OF PROTEASOME INHIBITORS THAT PREVENT NF-KAPPA-B ACTIVATION, Biochemical pharmacology, 55(9), 1998, pp. 1391-1397
Authors:
SCHOW SR
MACKMAN RL
BLUM CL
BROOKS E
HORSMA AG
JOLY A
KERWAR SS
LEE G
SHIFFMAN D
NELSON MG
WANG XB
WICK MM
ZHANG XM
LUM RT
Citation: Sr. Schow et al., SYNTHESIS AND ACTIVITY OF 2,6,9-TRISUBSTITUTED PURINES, Bioorganic & medicinal chemistry letters, 7(21), 1997, pp. 2697-2702
Authors:
MEYER S
LUM RT
NELSON MG
SCHOW SR
SHIFFMAN D
KERWAR SS
WICK MM
JOLY A
Citation: S. Meyer et al., INHIBITION OF THE CHYMOTRYPSIN-LIKE ACTIVITY OF THE PROTEASOME PREVENTS LIPOPOLYSACCHARIDE-INDUCED NF-KAPPA-B ACTIVATION, The FASEB journal, 11(9), 1997, pp. 2180-2180
Authors:
PFISTER JR
BELARDINELLI L
LEE G
LUM RT
MILNER P
STANLEY WC
LINDEN J
BAKER SP
SCHREINER G
Citation: Jr. Pfister et al., SYNTHESIS AND BIOLOGICAL EVALUATION OF THE ENANTIOMERS OF THE POTENT AND SELECTIVE A(1)-ADENOSINE ANTAGONIST 1,3-DIPROPYL-8-[2-(5,6-EPOXYNORBONYL)]XANTHINE, Journal of medicinal chemistry, 40(12), 1997, pp. 1773-1778
Authors:
THOMPSON SK
EPPLEY AM
FRAZEE JS
DARCY MG
LUM RT
TOMASZEK TA
IVANOFF LA
MORRIS JF
STERNBERG EJ
LAMBERT DM
FERNANDEZ AV
PETTEWAY SR
MEEK TD
METCALF BW
GLEASON JG
Citation: Sk. Thompson et al., SYNTHESIS AND ANTIVIRAL ACTIVITY OF A NOVEL CLASS OF HIV-1 PROTEASE INHIBITORS CONTAINING A HETEROCYCLIC P-1'-P-2' AMIDE BOND ISOSTERE, Bioorganic & medicinal chemistry letters, 4(20), 1994, pp. 2441-2446