Authors:
SANDERSON PEJ
LYLE TA
CUTRONA KJ
DYER DL
DORSEY BD
MCDONOUGH CM
NAYLOROLSEN AM
CHEN IW
CHEN ZG
COOK JJ
COOPER CM
GARDELL SJ
HARE TR
KRUEGER JA
LEWIS SD
LIN JH
LUCAS BJ
LYLE EA
LYNCH JJ
STRANIERI MT
VASTAG K
YAN YW
SHAFER JA
VACCA JP
Citation: Pej. Sanderson et al., EFFICACIOUS, ORALLY BIOAVAILABLE THROMBIN INHIBITORS BASED ON 3-AMINOPYRIDINONE OR 3-AMINOPYRAZINONE ACETAMIDE PEPTIDOMIMETIC TEMPLATES, Journal of medicinal chemistry, 41(23), 1998, pp. 4466-4474
Authors:
HOLLOWAY MK
WAI JM
HALGREN TA
FITZGERALD PMD
VACCA JP
DORSEY BD
LEVIN RB
THOMPSON WJ
CHEN LJ
DESOLMS SJ
GAFFIN N
GHOSH AK
GIULIANI EA
GRAHAM SL
GUARE JP
HUNGATE RW
LYLE TA
SANDERS WM
TUCKER TJ
WIGGINS M
WISCOUNT CM
WOLTERSDORF OW
YOUNG SD
DARKE PL
ZUGAY JA
Citation: Mk. Holloway et al., A-PRIORI PREDICTION OF ACTIVITY FOR HIV-1 PROTEASE INHIBITORS EMPLOYING ENERGY MINIMIZATION IN THE ACTIVE-SITE (VOL 38, PG 308, 1995), Journal of medicinal chemistry, 39(11), 1996, pp. 2280-2280
Authors:
YOUNG SD
BRITCHER SF
TRAN LO
PAYNE LS
LUMMA WC
LYLE TA
HUFF JR
ANDERSON PS
OLSEN DB
CARROLL SS
PETTIBONE DJ
OBRIEN JA
BALL RG
BALANI SK
LIN JH
CHEN IW
SCHLEIF WA
SARDANA VV
LONG WJ
BYRNES VW
EMINI EA
Citation: Sd. Young et al., L-743,726 (DMP-266) - A NOVEL, HIGHLY POTENT NONNUCLEOSIDE INHIBITOR OF THE HUMAN-IMMUNODEFICIENCY-VIRUS TYPE-1 REVERSE-TRANSCRIPTASE, Antimicrobial agents and chemotherapy, 39(12), 1995, pp. 2602-2605
Authors:
HOLLOWAY MK
WAI JM
HALGREN TA
FITZGERALD PMD
VACCA JP
DORSEY BD
LEVIN RB
THOMPSON WJ
CHEN LJ
DESOLMS SJ
GAFFIN N
GHOSH AK
GIULIANI EA
GRAHAM SL
GUARE JP
HUNGATE RW
LYLE TA
SANDERS WM
TUCKER TJ
WIGGINS M
WISCOUNT CM
WOLTERSDORF OW
YOUNG SD
DARKE PL
ZUGAY JA
Citation: Mk. Holloway et al., A-PRIORI PREDICTION OF ACTIVITY FOR HIV-1 PROTEASE INHIBITORS EMPLOYING ENERGY MINIMIZATION IN THE ACTIVE-SITE, Journal of medicinal chemistry, 38(2), 1995, pp. 305-317
Authors:
TUCKER TJ
LYLE TA
WISCOUNT CM
BRITCHER SF
YOUNG SD
SANDERS WM
LUMMA WC
GOLDMAN ME
OBRIEN JA
BALL RG
HOMNICK CF
SCHLEIF WA
EMINI EA
HUFF JR
ANDERSON PS
Citation: Tj. Tucker et al., SYNTHESIS OF A SERIES OF ORO-4-CYCLOPROPYL-3,4-DIHYDROQUINAZOLIN-2(1H)-ONES AS NOVEL NONNUCLEOSIDE HIV-1 REVERSE-TRANSCRIPTASE INHIBITORS, Journal of medicinal chemistry, 37(15), 1994, pp. 2437-2444