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Results: 1-9 |
Results: 9
3-aryl[1,2,4]triazino[4,3-alpha]benzimidazol-4(10H)-ones: A new class of selective A(1) adenosine receptor antagonists
Authors: Da Settimo, F Primofiore, G Taliani, S Marini, AM La Motta, C Novellino, E Greco, G Lavecchia, A Trincavelli, L Martini, C
Citation: F. Da Settimo et al., 3-aryl[1,2,4]triazino[4,3-alpha]benzimidazol-4(10H)-ones: A new class of selective A(1) adenosine receptor antagonists, J MED CHEM, 44(3), 2001, pp. 316-327
[1,2,4]triazino[4,3-a]benzimidazole acetic acid derivatives: A new class of selective aldose reductase inhibitors
Authors: Da Settimo, F Primofiore, G Da Settimo, A La Motta, C Taliani, S Simorini, F Novellino, E Greco, G Lavecchia, A Boldrini, E
Citation: F. Da Settimo et al., [1,2,4]triazino[4,3-a]benzimidazole acetic acid derivatives: A new class of selective aldose reductase inhibitors, J MED CHEM, 44(25), 2001, pp. 4359-4369
Structure-based design, synthesis, and biological evaluation of conformationally restricted novel 2-alkylthio-6-[1-(2,6-difluorophenyl)alkyl]-3,4-dihydro-5-alkylpyrimidin-4(3H)-ones as non-nucleoside inhibitors of HIV-1 reverse transcriptase
Authors: Mai, A Sbardella, G Artico, M Ragno, R Massa, S Novellino, E Greco, G Lavecchia, A Musiu, C La Colla, M Murgioni, C La Colla, P Loddo, R
Citation: A. Mai et al., Structure-based design, synthesis, and biological evaluation of conformationally restricted novel 2-alkylthio-6-[1-(2,6-difluorophenyl)alkyl]-3,4-dihydro-5-alkylpyrimidin-4(3H)-ones as non-nucleoside inhibitors of HIV-1 reverse transcriptase, J MED CHEM, 44(16), 2001, pp. 2544-2554
Novel N-(arylalkyl) indol-3-ylglyoxylylamides targeted as ligands of the benzodiazepine receptor: Synthesis, biological evaluation, and molecular modeling analysis of the structure-activity relationships
Authors: Primofiore, G Da Settimo, F Taliani, S Marini, AM Novellino, E Greco, G Lavecchia, A Besnard, F Trincavelli, L Costa, B Martini, C
Citation: G. Primofiore et al., Novel N-(arylalkyl) indol-3-ylglyoxylylamides targeted as ligands of the benzodiazepine receptor: Synthesis, biological evaluation, and molecular modeling analysis of the structure-activity relationships, J MED CHEM, 44(14), 2001, pp. 2286-2297
Computer-assisted design, synthesis and biological evaluation of novel pyrrolyl heteroaryl sulfones targeted at HIV-1 reverse transcriptase as non-nucleoside inhibitors
Authors: Silvestri, R Artico, M De Martino, G Novellino, E Greco, G Lavecchia, A Massa, S Loi, AG Doratiotto, S La Colla, P
Citation: R. Silvestri et al., Computer-assisted design, synthesis and biological evaluation of novel pyrrolyl heteroaryl sulfones targeted at HIV-1 reverse transcriptase as non-nucleoside inhibitors, BIO MED CH, 8(9), 2000, pp. 2305-2309
Structure-activity relationship studies on potential non-nucleoside DABO-like inhibitors of HIV-1 reverse transcriptase
Authors: Costi, R Di Santo, R Artico, M Massa, S Lavecchia, A Marceddu, T Sanna, L La Colla, P Marongiu, ME
Citation: R. Costi et al., Structure-activity relationship studies on potential non-nucleoside DABO-like inhibitors of HIV-1 reverse transcriptase, ANTIVIR CHE, 11(2), 2000, pp. 117-133
Synthesis, molecular modeling, and opioid receptor affinity of 9,10-diazatricyclo[4.2.1.1(2,5)]decanes and 2,7-diazatricyclo[4.4.0.0(3,8)]decanes structurally related to 3,8-diazabicyclo[3.2.1]octanes
Authors: Vianello, P Albinati, A Pinna, GA Lavecchia, A Marinelli, L Borea, PA Gessi, S Fadda, P Tronci, S Cignarella, G
Citation: P. Vianello et al., Synthesis, molecular modeling, and opioid receptor affinity of 9,10-diazatricyclo[4.2.1.1(2,5)]decanes and 2,7-diazatricyclo[4.4.0.0(3,8)]decanes structurally related to 3,8-diazabicyclo[3.2.1]octanes, J MED CHEM, 43(11), 2000, pp. 2115-2123
Modeling of kappa-opioid receptor/agonists interactions using pharmacophore-based and docking simulations
Authors: Lavecchia, A Greco, G Novellino, E Vittorio, F Ronsisvalle, G
Citation: A. Lavecchia et al., Modeling of kappa-opioid receptor/agonists interactions using pharmacophore-based and docking simulations, J MED CHEM, 43(11), 2000, pp. 2124-2134
Solution conformation of a potent cyclic analogue of tuftsin: Low-temperature nuclear magnetic resonance study in a cryoprotective mixture
Authors: D'Ursi, A Albrizio, S Fattorusso, C Lavecchia, A Zanotti, G Temussi, PA
Citation: A. D'Ursi et al., Solution conformation of a potent cyclic analogue of tuftsin: Low-temperature nuclear magnetic resonance study in a cryoprotective mixture, J MED CHEM, 42(10), 1999, pp. 1705-1713
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