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Results: 1-15 |
Results: 15
NEW NONSTEROIDAL ANDROGEN RECEPTOR MODULATORS BASED ON 4(TRIFLUOROMETHYL)-2 (1H)-PYRROLIDINO[3,2-G] QUINOLINONE
Authors: EDWARDS JP WEST SJ POOLEY CLF MARSCHKE KB FARMER LJ JONES TK
Citation: Jp. Edwards et al., NEW NONSTEROIDAL ANDROGEN RECEPTOR MODULATORS BASED ON 4(TRIFLUOROMETHYL)-2 (1H)-PYRROLIDINO[3,2-G] QUINOLINONE, Bioorganic & medicinal chemistry letters, 8(7), 1998, pp. 745-750
NONSTEROIDAL PROGESTERONE-RECEPTOR ANTAGONISTS BASED ON A CONFORMATIONALLY-RESTRICTED SUBSERIES OF 6-ARYL-1,2-DIHYDRO-2,2,4-TRIMETHYLQUINOLINES
Authors: HAMANN LG WINN DT POOLEY CLF TEGLEY CM WEST SJ FARMER LJ ZHI L EDWARDS JP MARSCHKE KB MAIS DE GOLDMAN ME JONES TK
Citation: Lg. Hamann et al., NONSTEROIDAL PROGESTERONE-RECEPTOR ANTAGONISTS BASED ON A CONFORMATIONALLY-RESTRICTED SUBSERIES OF 6-ARYL-1,2-DIHYDRO-2,2,4-TRIMETHYLQUINOLINES, Bioorganic & medicinal chemistry letters, 8(19), 1998, pp. 2731-2736
SYNTHESIS AND BIOLOGICAL-ACTIVITY OF A NOVEL SERIES OF NONSTEROIDAL, PERIPHERALLY SELECTIVE ANDROGEN RECEPTOR ANTAGONISTS DERIVED FROM 1,2-DIHYDROPYRIDONO[5,6-G] QUINOLINES
Authors: HAMANN LG HIGUCHI RI ZHI L EDWARDS JP WANG XN MARSCHKE KB KONG JW FARMER LJ JONES TK
Citation: Lg. Hamann et al., SYNTHESIS AND BIOLOGICAL-ACTIVITY OF A NOVEL SERIES OF NONSTEROIDAL, PERIPHERALLY SELECTIVE ANDROGEN RECEPTOR ANTAGONISTS DERIVED FROM 1,2-DIHYDROPYRIDONO[5,6-G] QUINOLINES, Journal of medicinal chemistry, 41(4), 1998, pp. 623-639
5-ARYL-1,2-DIHYDROCHROMENO[3,4-F]QUINOLINES - A NOVEL CLASS OF NONSTEROIDAL HUMAN PROGESTERONE-RECEPTOR AGONISTS
Authors: ZHI L TEGLEY CM KALLEL EA MARSCHKE KB MAIS DE GOTTARDIS MM JONES TK
Citation: L. Zhi et al., 5-ARYL-1,2-DIHYDROCHROMENO[3,4-F]QUINOLINES - A NOVEL CLASS OF NONSTEROIDAL HUMAN PROGESTERONE-RECEPTOR AGONISTS, Journal of medicinal chemistry, 41(3), 1998, pp. 291-302
5-ARYL-1,2-DIHYDRO-5H-CHROMENO[3,4-F]QUINOLINES AS POTENT, ORALLY-ACTIVE, NONSTEROIDAL PROGESTERONE-RECEPTOR AGONISTS - THE EFFECT OF D-RING SUBSTITUENTS
Authors: EDWARDS JP WEST SJ MARSCHKE KB MAIS DE GOTTARDIS MM JONES TK
Citation: Jp. Edwards et al., 5-ARYL-1,2-DIHYDRO-5H-CHROMENO[3,4-F]QUINOLINES AS POTENT, ORALLY-ACTIVE, NONSTEROIDAL PROGESTERONE-RECEPTOR AGONISTS - THE EFFECT OF D-RING SUBSTITUENTS, Journal of medicinal chemistry, 41(3), 1998, pp. 303-310
5-BENZYLIDENE 1,2-DIHYDROCHROMENO[3,4-F]QUINOLINES, A NOVEL CLASS OF NONSTEROIDAL HUMAN PROGESTERONE-RECEPTOR AGONISTS
Authors: TEGLEY CM ZHI L MARSCHKE KB GOTTARDIS MM YANG QC JONES TK
Citation: Cm. Tegley et al., 5-BENZYLIDENE 1,2-DIHYDROCHROMENO[3,4-F]QUINOLINES, A NOVEL CLASS OF NONSTEROIDAL HUMAN PROGESTERONE-RECEPTOR AGONISTS, Journal of medicinal chemistry, 41(22), 1998, pp. 4354-4359
DISCOVERY AND PRELIMINARY SAR STUDIES OF A NOVEL, NONSTEROIDAL PROGESTERONE-RECEPTOR ANTAGONIST PHARMACOPHORE
Authors: POOLEY CLF EDWARDS JP GOLDMAN ME WANG MW MARSCHKE KB CROMBIE DL JONES TK
Citation: Clf. Pooley et al., DISCOVERY AND PRELIMINARY SAR STUDIES OF A NOVEL, NONSTEROIDAL PROGESTERONE-RECEPTOR ANTAGONIST PHARMACOPHORE, Journal of medicinal chemistry, 41(18), 1998, pp. 3461-3466
ANDROGEN RECEPTOR-MEDIATED ANTAGONISM OF ESTROGEN-DEPENDENT LOW-DENSITY-LIPOPROTEIN RECEPTOR TRANSCRIPTION IN CULTURED-HEPATOCYTES
Authors: CROSTON GE MILAN LB MARSCHKE KB REICHMAN M BRIGGS MR
Citation: Ge. Croston et al., ANDROGEN RECEPTOR-MEDIATED ANTAGONISM OF ESTROGEN-DEPENDENT LOW-DENSITY-LIPOPROTEIN RECEPTOR TRANSCRIPTION IN CULTURED-HEPATOCYTES, Endocrinology, 138(9), 1997, pp. 3779-3786
ESTROGEN AND ESTROGEN-RECEPTOR ANTAGONISTS STIMULATE TRANSCRIPTION FROM THE HUMAN RETINOIC ACID RECEPTOR-ALPHA-1 PROMOTER VIA A NOVEL SEQUENCE
Authors: ELGORT MG ZOU A MARSCHKE KB ALLEGRETTO EA
Citation: Mg. Elgort et al., ESTROGEN AND ESTROGEN-RECEPTOR ANTAGONISTS STIMULATE TRANSCRIPTION FROM THE HUMAN RETINOIC ACID RECEPTOR-ALPHA-1 PROMOTER VIA A NOVEL SEQUENCE, Molecular endocrinology, 10(5), 1996, pp. 477-487
SPECIFICITY OF SIMPLE HORMONE RESPONSE ELEMENTS IN ANDROGEN-REGULATEDGENES
Authors: MARSCHKE KB TAN JA KUPFER SR WILSON EM FRENCH FS
Citation: Kb. Marschke et al., SPECIFICITY OF SIMPLE HORMONE RESPONSE ELEMENTS IN ANDROGEN-REGULATEDGENES, Endocrine, 3(11), 1995, pp. 819-825
ANDROGEN RECEPTOR DEFECTS - HISTORICAL, CLINICAL, AND MOLECULAR PERSPECTIVES
Authors: QUIGLEY CA DEBELLIS A MARSCHKE KB ELAWADY MK WILSON EM FRENCH FS
Citation: Ca. Quigley et al., ANDROGEN RECEPTOR DEFECTS - HISTORICAL, CLINICAL, AND MOLECULAR PERSPECTIVES, Endocrine reviews, 16(3), 1995, pp. 271-321
CHARACTERIZATION OF A HEPATIC PROTEIN IN NONHUMAN-PRIMATES THAT BINDSMIBOLERONE BUT NOT DIHYDROTESTOSTERONE OR METHYLTRIENOLONE
Authors: KORITNIK DR MARSCHKE KB KOSHY A
Citation: Dr. Koritnik et al., CHARACTERIZATION OF A HEPATIC PROTEIN IN NONHUMAN-PRIMATES THAT BINDSMIBOLERONE BUT NOT DIHYDROTESTOSTERONE OR METHYLTRIENOLONE, Steroids, 60(11), 1995, pp. 759-767
CHARACTERIZATION OF MUTANT ANDROGEN RECEPTORS CAUSING PARTIAL ANDROGEN INSENSITIVITY SYNDROME
Authors: DEBELLIS A QUIGLEY CA MARSCHKE KB ELAWADY MK LANE MV SMITH EP SAR M WILSON EM FRENCH FS
Citation: A. Debellis et al., CHARACTERIZATION OF MUTANT ANDROGEN RECEPTORS CAUSING PARTIAL ANDROGEN INSENSITIVITY SYNDROME, The Journal of clinical endocrinology and metabolism, 78(3), 1994, pp. 513-522
A COMPLEX RESPONSE ELEMENT IN INTRON-1 OF THE ANDROGEN-REGULATED 20-KDA PROTEIN GENE DISPLAYS CELL TYPE-DEPENDENT ANDROGEN RECEPTOR SPECIFICITY
Authors: HO KC MARSCHKE KB TAN JA POWER SGA WILSON EM FRENCH FS
Citation: Kc. Ho et al., A COMPLEX RESPONSE ELEMENT IN INTRON-1 OF THE ANDROGEN-REGULATED 20-KDA PROTEIN GENE DISPLAYS CELL TYPE-DEPENDENT ANDROGEN RECEPTOR SPECIFICITY, The Journal of biological chemistry, 268(36), 1993, pp. 27226-27235
RECEPTOR ACCESSORY FACTOR ENHANCES SPECIFIC DNA-BINDING OF ANDROGEN AND GLUCOCORTICOID RECEPTORS
Authors: KUPFER SR MARSCHKE KB WILSON EM FRENCH FS
Citation: Sr. Kupfer et al., RECEPTOR ACCESSORY FACTOR ENHANCES SPECIFIC DNA-BINDING OF ANDROGEN AND GLUCOCORTICOID RECEPTORS, The Journal of biological chemistry, 268(23), 1993, pp. 17519-17527
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