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Results: 5

Authors: PRASAD JVNV TUMMINO PJ FERGUSON D SAUNDERS J VANDERROEST S MCQUADE TJ HELDSINGER A REYNER EL STEWART BH GUTTENDORF RJ PARA KS LUNNEY EA GRACHECK SJ DOMAGALA JM
Citation: Jvnv. Prasad et al., NONPEPTIDIC HIV PROTEASE INHIBITORS - 4-HYDROXY-PYRAN-2-ONE INHIBITORS WITH FUNCTIONAL TETHERS TO P-1 PHENYL RING TO REACH S-3 POCKET OF THE ENZYME, Biochemical and biophysical research communications, 221(3), 1996, pp. 815-820

Authors: PRASAD JVN PARA KS TUMMINO PJ FERGUSON D MCQUADE TJ LUNNEY EA RAPUNDALO ST BATLEY BL HINGORANI G DOMAGALA JM GRACHECK SJ BHAT TN LIU BS BALDWIN ET ERICKSON JW SAWYER TK
Citation: Jvn. Prasad et al., NONPEPTIDIC POTENT HIV-1 PROTEASE INHIBITORS - -HYDROXY-6-PHENYL-2-OXO-2H-PYRAN-3-YL)THIOMETHANES THAT SPAN P-1-P-2' SUBSITES IN A UNIQUE MODE OF ACTIVE-SITE BINDING, Journal of medicinal chemistry, 38(6), 1995, pp. 898-905

Authors: ISLAM I NG KY CHONG KT MCQUADE TJ HUI JO WILKINSON KF RUSH BD RUWART MJ BORCHARDT RT FISHER JF
Citation: I. Islam et al., EVALUATION OF A VITAMIN-CLOAKING STRATEGY FOR OLIGOPEPTIDE THERAPEUTICS - BIOTINYLATED HIV-1 PROTEASE INHIBITORS, Journal of medicinal chemistry, 37(2), 1994, pp. 293-304

Authors: SAWYER TK FISHER JF HESTER JB SMITH CW TOMASSELLI AG TARPLEY WG BURTON PS HUI JO MCQUADE TJ CONRADI RA BRADFORD VS LIU L KINNER JH TUSTIN J ALEXANDER DL HARRISON AW EMMERT DE STAPLES DJ MAGGIORA LL ZHANG YZ POORMAN RA DUNN BM RAO C SCARBOROUGH PE LOWTHER WT CRAIK C DECAMP D MOON J HOWE WJ HEINRIKSON RL
Citation: Tk. Sawyer et al., PEPTIDOMIMETIC INHIBITORS OF HUMAN-IMMUNODEFICIENCY-VIRUS PROTEASE (HIV-PR) - DESIGN, ENZYME BINDING AND SELECTIVITY, ANTIVIRAL EFFICACY, AND CELL-PERMEABILITY PROPERTIES, Bioorganic & medicinal chemistry letters, 3(5), 1993, pp. 819-824

Authors: THAISRIVONGS S TURNER SR STROHBACH JW TENBRINK RE TARPLEY WG MCQUADE TJ HEINRIKSON RL TOMASSELLI AG HUI JO HOWE WJ
Citation: S. Thaisrivongs et al., INHIBITORS OF THE PROTEASE FROM HUMAN-IMMUNODEFICIENCY-VIRUS - SYNTHESIS, ENZYME-INHIBITION, AND ANTIVIRAL ACTIVITY OF A SERIES OF COMPOUNDS CONTAINING THE DIHYDROXYETHYLENE TRANSITION-STATE ISOSTERE, Journal of medicinal chemistry, 36(8), 1993, pp. 941-952
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