Authors:
PRASAD JVNV
TUMMINO PJ
FERGUSON D
SAUNDERS J
VANDERROEST S
MCQUADE TJ
HELDSINGER A
REYNER EL
STEWART BH
GUTTENDORF RJ
PARA KS
LUNNEY EA
GRACHECK SJ
DOMAGALA JM
Citation: Jvnv. Prasad et al., NONPEPTIDIC HIV PROTEASE INHIBITORS - 4-HYDROXY-PYRAN-2-ONE INHIBITORS WITH FUNCTIONAL TETHERS TO P-1 PHENYL RING TO REACH S-3 POCKET OF THE ENZYME, Biochemical and biophysical research communications, 221(3), 1996, pp. 815-820
Authors:
PRASAD JVN
PARA KS
TUMMINO PJ
FERGUSON D
MCQUADE TJ
LUNNEY EA
RAPUNDALO ST
BATLEY BL
HINGORANI G
DOMAGALA JM
GRACHECK SJ
BHAT TN
LIU BS
BALDWIN ET
ERICKSON JW
SAWYER TK
Citation: Jvn. Prasad et al., NONPEPTIDIC POTENT HIV-1 PROTEASE INHIBITORS - -HYDROXY-6-PHENYL-2-OXO-2H-PYRAN-3-YL)THIOMETHANES THAT SPAN P-1-P-2' SUBSITES IN A UNIQUE MODE OF ACTIVE-SITE BINDING, Journal of medicinal chemistry, 38(6), 1995, pp. 898-905
Authors:
ISLAM I
NG KY
CHONG KT
MCQUADE TJ
HUI JO
WILKINSON KF
RUSH BD
RUWART MJ
BORCHARDT RT
FISHER JF
Citation: I. Islam et al., EVALUATION OF A VITAMIN-CLOAKING STRATEGY FOR OLIGOPEPTIDE THERAPEUTICS - BIOTINYLATED HIV-1 PROTEASE INHIBITORS, Journal of medicinal chemistry, 37(2), 1994, pp. 293-304
Authors:
SAWYER TK
FISHER JF
HESTER JB
SMITH CW
TOMASSELLI AG
TARPLEY WG
BURTON PS
HUI JO
MCQUADE TJ
CONRADI RA
BRADFORD VS
LIU L
KINNER JH
TUSTIN J
ALEXANDER DL
HARRISON AW
EMMERT DE
STAPLES DJ
MAGGIORA LL
ZHANG YZ
POORMAN RA
DUNN BM
RAO C
SCARBOROUGH PE
LOWTHER WT
CRAIK C
DECAMP D
MOON J
HOWE WJ
HEINRIKSON RL
Citation: Tk. Sawyer et al., PEPTIDOMIMETIC INHIBITORS OF HUMAN-IMMUNODEFICIENCY-VIRUS PROTEASE (HIV-PR) - DESIGN, ENZYME BINDING AND SELECTIVITY, ANTIVIRAL EFFICACY, AND CELL-PERMEABILITY PROPERTIES, Bioorganic & medicinal chemistry letters, 3(5), 1993, pp. 819-824
Authors:
THAISRIVONGS S
TURNER SR
STROHBACH JW
TENBRINK RE
TARPLEY WG
MCQUADE TJ
HEINRIKSON RL
TOMASSELLI AG
HUI JO
HOWE WJ
Citation: S. Thaisrivongs et al., INHIBITORS OF THE PROTEASE FROM HUMAN-IMMUNODEFICIENCY-VIRUS - SYNTHESIS, ENZYME-INHIBITION, AND ANTIVIRAL ACTIVITY OF A SERIES OF COMPOUNDS CONTAINING THE DIHYDROXYETHYLENE TRANSITION-STATE ISOSTERE, Journal of medicinal chemistry, 36(8), 1993, pp. 941-952