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Results: 1-25 | 26-36
Results: 1-25/36
STRATEGIES TOWARD IDENTIFICATION OF NOVEL AND SELECTIVE PROTEIN-KINASE INHIBITORS
Authors: ZIMMERMANN J BUCHDUNGER E CAPRARO HG COLLINGWOOD S FABBRO D FURET P GEIGER T IMBACH P METT H MEYER T RUETZ S TRAXLER P
Citation: J. Zimmermann et al., STRATEGIES TOWARD IDENTIFICATION OF NOVEL AND SELECTIVE PROTEIN-KINASE INHIBITORS, Annals of oncology, 9, 1998, pp. 11-11
PHARMACODYNAMIC CONFIRMATION OF CGP-48664 AS AN INHIBITOR OF THE POLYAMINE BIOSYNTHETIC ENZYME S-DENOSYLMETHIONINE DECARBOXYLASE (SAMDC) INAN ADVANCED MELANOMA PATIENT
Authors: PORTER CW SIU L KRAMER DL METT H BARBET N LINNARTZ R ECKHARDT SG
Citation: Cw. Porter et al., PHARMACODYNAMIC CONFIRMATION OF CGP-48664 AS AN INHIBITOR OF THE POLYAMINE BIOSYNTHETIC ENZYME S-DENOSYLMETHIONINE DECARBOXYLASE (SAMDC) INAN ADVANCED MELANOMA PATIENT, Annals of oncology, 9, 1998, pp. 491-491
S-ADENOSYLMETHIONINE DECARBOXYLASE OF ONCHOCERCA-VOLVULUS AS A TARGETFOR CHEMOTHERAPY
Authors: DADARA AA METT H MULLER S WALTER RD
Citation: Aa. Dadara et al., S-ADENOSYLMETHIONINE DECARBOXYLASE OF ONCHOCERCA-VOLVULUS AS A TARGETFOR CHEMOTHERAPY, Naunyn-Schmiedeberg's archives of pharmacology, 358(1), 1998, pp. 4419-4419
S-ADENOSYLMETHIONINE DECARBOXYLASE OF ONCHOCERCA-VOLVULUS AS A TARGETFOR CHEMOTHERAPY
Authors: DADARA AA METT H MULLER S WALTER RD
Citation: Aa. Dadara et al., S-ADENOSYLMETHIONINE DECARBOXYLASE OF ONCHOCERCA-VOLVULUS AS A TARGETFOR CHEMOTHERAPY, Naunyn-Schmiedeberg's archives of pharmacology, 358(1), 1998, pp. 103-103
SELECTIVE-INHIBITION OF THE PLATELET-DERIVED GROWTH-FACTOR SIGNAL-TRANSDUCTION PATHWAY BY A PROTEIN-TYROSINE KINASE INHIBITOR OF THE 2-PHENYLAMINOPYRIMIDINE CLASS (VOL 92, PG 2558, 1995)
Authors: BUCHDUNGER E ZIMMERMANN J METT H MEYER T MULLER M REGENASS U LYDON NB
Citation: E. Buchdunger et al., SELECTIVE-INHIBITION OF THE PLATELET-DERIVED GROWTH-FACTOR SIGNAL-TRANSDUCTION PATHWAY BY A PROTEIN-TYROSINE KINASE INHIBITOR OF THE 2-PHENYLAMINOPYRIMIDINE CLASS (VOL 92, PG 2558, 1995), Proceedings of the National Academy of Sciences of the United Statesof America, 95(20), 1998, pp. 12069-12069
4,5-DIANILINOPHTHALIMIDE - A PROTEIN-TYROSINE KINASE INHIBITOR WITH SELECTIVITY FOR THE EPIDERMAL GROWTH-FACTOR RECEPTOR SIGNAL-TRANSDUCTION PATHWAY AND POTENT IN-VIVO ANTITUMOR-ACTIVITY (VOL 91, PG 2334, 1994)
Authors: BUCHDUNGER E TRINKS U METT H REGENASS U MULLER M MEYER T MCGLYNN E PINNA LA TRAXLER P LYDON NB
Citation: E. Buchdunger et al., 4,5-DIANILINOPHTHALIMIDE - A PROTEIN-TYROSINE KINASE INHIBITOR WITH SELECTIVITY FOR THE EPIDERMAL GROWTH-FACTOR RECEPTOR SIGNAL-TRANSDUCTION PATHWAY AND POTENT IN-VIVO ANTITUMOR-ACTIVITY (VOL 91, PG 2334, 1994), Proceedings of the National Academy of Sciences of the United Statesof America, 95(20), 1998, pp. 12069-12069
A POTENT PROTEIN-TYROSINE KINASE INHIBITOR WHICH SELECTIVELY BLOCKS PROLIFERATION OF EPIDERMAL GROWTH-FACTOR RECEPTOR-EXPRESSING TUMOR-CELLS IN-VITRO AND IN-VIVO
Authors: LYDON NB METT H MUELLER M BECKER M COZENS RM STOVER D DANIELS D TRAXLER P BUCHDUNGER E
Citation: Nb. Lydon et al., A POTENT PROTEIN-TYROSINE KINASE INHIBITOR WHICH SELECTIVELY BLOCKS PROLIFERATION OF EPIDERMAL GROWTH-FACTOR RECEPTOR-EXPRESSING TUMOR-CELLS IN-VITRO AND IN-VIVO, International journal of cancer, 76(1), 1998, pp. 154-163
LYSOSOMAL SEQUESTRATION OF POLYAMINE ANALOGS IN CHINESE-HAMSTER OVARYCELLS RESISTANT TO THE S-ADENOSYLMETHIONINE DECARBOXYLASE INHIBITOR, CGP-48664
Authors: KRAMER DL BLACK JD METT H BERGERON RJ PORTER CW
Citation: Dl. Kramer et al., LYSOSOMAL SEQUESTRATION OF POLYAMINE ANALOGS IN CHINESE-HAMSTER OVARYCELLS RESISTANT TO THE S-ADENOSYLMETHIONINE DECARBOXYLASE INHIBITOR, CGP-48664, Cancer research, 58(17), 1998, pp. 3883-3890
POTENT AND SELECTIVE INHIBITORS OF THE ABL-KINASE - PHENYLAMINO-PYRIMIDINE (PAP) DERIVATIVES
Authors: ZIMMERMANN J BUCHDUNGER E METT H MEYER T LYDON NB
Citation: J. Zimmermann et al., POTENT AND SELECTIVE INHIBITORS OF THE ABL-KINASE - PHENYLAMINO-PYRIMIDINE (PAP) DERIVATIVES, Bioorganic & medicinal chemistry letters, 7(2), 1997, pp. 187-192
CGP-48664, A POTENT AND SPECIFIC S-ADENOSYLMETHIONINE DECARBOXYLASE INHIBITOR - EFFECTS ON REGULATION AND STABILITY OF THE ENZYME
Authors: SVENSSON F METT H PERSSON L
Citation: F. Svensson et al., CGP-48664, A POTENT AND SPECIFIC S-ADENOSYLMETHIONINE DECARBOXYLASE INHIBITOR - EFFECTS ON REGULATION AND STABILITY OF THE ENZYME, Biochemical journal, 322, 1997, pp. 297-302
ALTERATIONS IN ORNITHINE DECARBOXYLASE CHARACTERISTICS ACCOUNT FOR TOLERANCE OF TRYPANOSOMA-BRUCEI-RHODESIENSE TO D,L-ALPHA-DIFLUOROMETHYLORNITHINE
Authors: ITEN M METT H EVANS A ENYARU JCK BRUN R KAMINSKY R
Citation: M. Iten et al., ALTERATIONS IN ORNITHINE DECARBOXYLASE CHARACTERISTICS ACCOUNT FOR TOLERANCE OF TRYPANOSOMA-BRUCEI-RHODESIENSE TO D,L-ALPHA-DIFLUOROMETHYLORNITHINE, Antimicrobial agents and chemotherapy, 41(9), 1997, pp. 1922-1925
USE OF A PHARMACOPHORE MODEL FOR THE DESIGN OF EGF-R TYROSINE KINASE INHIBITORS - 4-(PHENYLAMINO)PYRAZOLO[3,4-D]PYRIMIDINES
Authors: TRAXLER P BOLD G FREI J LANG M LYDON N METT H BUCHDUNGER E MEYER T MUELLER M FURET P
Citation: P. Traxler et al., USE OF A PHARMACOPHORE MODEL FOR THE DESIGN OF EGF-R TYROSINE KINASE INHIBITORS - 4-(PHENYLAMINO)PYRAZOLO[3,4-D]PYRIMIDINES, Journal of medicinal chemistry, 40(22), 1997, pp. 3601-3616
SEMICOCHLIODINOL-A AND SEMICOCHLIODINOL-B - INHIBITORS OF HIV-1 PROTEASE AND EGF-R PROTEIN-TYROSINE KINASE RELATED TO ASTERRIQUINONES PRODUCED BY THE FUNGUS CHRYSOSPORIUM-MERDARIUM
Authors: FREDENHAGEN A PETERSEN F TINTELNOTBLOMLEY M ROSEL J METT H HUG P
Citation: A. Fredenhagen et al., SEMICOCHLIODINOL-A AND SEMICOCHLIODINOL-B - INHIBITORS OF HIV-1 PROTEASE AND EGF-R PROTEIN-TYROSINE KINASE RELATED TO ASTERRIQUINONES PRODUCED BY THE FUNGUS CHRYSOSPORIUM-MERDARIUM, Journal of antibiotics, 50(5), 1997, pp. 395-401
SYNTHESIS OF MODIFIED TRIPEPTIDES AND TETRAPEPTIDES AS POTENTIAL BISUBSTRATE INHIBITORS OF THE EPIDERMAL GROWTH-FACTOR RECEPTOR PROTEIN-TYROSINE KINASE
Authors: ROSSE G SEQUIN U METT H FURET P TRAXLER P FRETZ H
Citation: G. Rosse et al., SYNTHESIS OF MODIFIED TRIPEPTIDES AND TETRAPEPTIDES AS POTENTIAL BISUBSTRATE INHIBITORS OF THE EPIDERMAL GROWTH-FACTOR RECEPTOR PROTEIN-TYROSINE KINASE, Helvetica Chimica Acta, 80(3), 1997, pp. 653-670
ALTERATIONS IN ORNITHINE DECARBOXYLASE CHARACTERISTICS ACCOUNT FOR TOLERANCE OF TRYPANOSOMA-BRUCEI-RHODESIENSE TO D,L-ALPHA-DIFLUOROMETHYLORNITHINE (DFMO)
Authors: KAMINSKY R ITEN M METT H LITTLEWOOD A BRUN R
Citation: R. Kaminsky et al., ALTERATIONS IN ORNITHINE DECARBOXYLASE CHARACTERISTICS ACCOUNT FOR TOLERANCE OF TRYPANOSOMA-BRUCEI-RHODESIENSE TO D,L-ALPHA-DIFLUOROMETHYLORNITHINE (DFMO), TM & IH. Tropical medicine & international health, 1(6), 1996, pp. 32-33
PHENYLAMINO-PYRIMIDINE (PAP) - DERIVATIVES - A NEW CLASS OF POTENT AND HIGHLY SELECTIVE PDGF-RECEPTOR AUTOPHOSPHORYLATION INHIBITORS
Authors: ZIMMERMANN J BUCHDUNGER E METT H MEYER T LYDON NB TRAXLER P
Citation: J. Zimmermann et al., PHENYLAMINO-PYRIMIDINE (PAP) - DERIVATIVES - A NEW CLASS OF POTENT AND HIGHLY SELECTIVE PDGF-RECEPTOR AUTOPHOSPHORYLATION INHIBITORS, Bioorganic & medicinal chemistry letters, 6(11), 1996, pp. 1221-1226
PHENYLAMINO-PYRIMIDINE (PAP) DERIVATIVES - A NEW CLASS OF POTENT AND SELECTIVE INHIBITORS OF PROTEIN-KINASE-C (PKC)
Authors: ZIMMERMANN J CARAVATTI G METT H MEYER T MULLER M LYDON NB FABBRO D
Citation: J. Zimmermann et al., PHENYLAMINO-PYRIMIDINE (PAP) DERIVATIVES - A NEW CLASS OF POTENT AND SELECTIVE INHIBITORS OF PROTEIN-KINASE-C (PKC), Archiv der pharmazie, 329(7), 1996, pp. 371-376
SEQUENCE-SPECIFIC ANTISENSE OLIGONUCLEOTIDE ANALOG INTERFERENCE WITH SPERMIDINE SPERMINE N-1-ACETYLTRANSFERASE GENE-EXPRESSION/
Authors: FOGELPETROVIC M VUJCIC S HANER R REGENASS U METT H PORTER CW
Citation: M. Fogelpetrovic et al., SEQUENCE-SPECIFIC ANTISENSE OLIGONUCLEOTIDE ANALOG INTERFERENCE WITH SPERMIDINE SPERMINE N-1-ACETYLTRANSFERASE GENE-EXPRESSION/, Anticancer research, 16(5A), 1996, pp. 2517-2523
IN-VITRO TRYPANOCIDAL ACTIVITIES OF NEW S-ADENOSYLMETHIONINE DECARBOXYLASE INHIBITORS
Authors: BRUN R BUHLER Y SANDMEIER U KAMINSKY R BACCHI CJ RATTENDI D LANE S CROFT SL SNOWDON D YARDLEY V CARAVATTI G FREI J STANEK J METT H
Citation: R. Brun et al., IN-VITRO TRYPANOCIDAL ACTIVITIES OF NEW S-ADENOSYLMETHIONINE DECARBOXYLASE INHIBITORS, Antimicrobial agents and chemotherapy, 40(6), 1996, pp. 1442-1447
INHIBITION OF THE ABL PROTEIN-TYROSINE KINASE IN-VITRO AND IN-VIVO BYA 2-PHENYLAMINOPYRIMIDINE DERIVATIVE
Authors: BUCHDUNGER E ZIMMERMANN J METT H MEYER T MULLER M DRUKER BJ LYDON NB
Citation: E. Buchdunger et al., INHIBITION OF THE ABL PROTEIN-TYROSINE KINASE IN-VITRO AND IN-VIVO BYA 2-PHENYLAMINOPYRIMIDINE DERIVATIVE, Cancer research, 56(1), 1996, pp. 100-104
DETERMINATION OF DECARBOXYLASE ACTIVITY IN ADHERENT TISSUE-CULTURE CELLS
Authors: SCHACHER B REUTER R BUSSELL K METT H
Citation: B. Schacher et al., DETERMINATION OF DECARBOXYLASE ACTIVITY IN ADHERENT TISSUE-CULTURE CELLS, Analytical biochemistry, 234(1), 1996, pp. 97-99
4,5-BIS(4-FLUOROANILINO)PHTHALIMIDE - A SELECTIVE INHIBITOR OF THE EPIDERMAL GROWTH-FACTOR RECEPTOR SIGNAL-TRANSDUCTION PATHWAY WITH POTENTIN-VIVO ANTITUMOR-ACTIVITY
Authors: BUCHDUNGER E METT H TRINKS U REGENASS U MULLER M MEYER T BEILSTEIN P WIRZ B SCHNEIDER P TRAXLER P LYDON NB
Citation: E. Buchdunger et al., 4,5-BIS(4-FLUOROANILINO)PHTHALIMIDE - A SELECTIVE INHIBITOR OF THE EPIDERMAL GROWTH-FACTOR RECEPTOR SIGNAL-TRANSDUCTION PATHWAY WITH POTENTIN-VIVO ANTITUMOR-ACTIVITY, Clinical cancer research, 1(8), 1995, pp. 813-821
SELECTIVE-INHIBITION OF THE PLATELET-DERIVED GROWTH-FACTOR SIGNAL-TRANSDUCTION PATHWAY BY A NOVEL TYROSINE PROTEIN-KINASE INHIBITOR OF THE 2-PHENYLAMINO PYRIMIDINE CLASS
Authors: LYDON NB ZIMMERMANN J METT H MEYER T MULLER M REGENASS U BUCHDUNGER E
Citation: Nb. Lydon et al., SELECTIVE-INHIBITION OF THE PLATELET-DERIVED GROWTH-FACTOR SIGNAL-TRANSDUCTION PATHWAY BY A NOVEL TYROSINE PROTEIN-KINASE INHIBITOR OF THE 2-PHENYLAMINO PYRIMIDINE CLASS, Journal of cellular biochemistry, 1995, pp. 69-69
SELECTIVE-INHIBITION OF THE PLATELET-DERIVED GROWTH-FACTOR SIGNAL-TRANSDUCTION PATHWAY BY A PROTEIN-TYROSINE KINASE INHIBITOR OF THE 2-PHENYLAMINOPYRIMIDINE CLASS
Authors: BUCHDUNGER E ZIMMERMANN J METT H MEYER T MULLER M REGENASS U LYDON NB
Citation: E. Buchdunger et al., SELECTIVE-INHIBITION OF THE PLATELET-DERIVED GROWTH-FACTOR SIGNAL-TRANSDUCTION PATHWAY BY A PROTEIN-TYROSINE KINASE INHIBITOR OF THE 2-PHENYLAMINOPYRIMIDINE CLASS, Proceedings of the National Academy of Sciences of the United Statesof America, 92(7), 1995, pp. 2558-2562
[(ALKYLAMINO)METHYL]ACRYLOPHENONES - POTENT AND SELECTIVE INHIBITORS OF THE EPIDERMAL GROWTH-FACTOR RECEPTOR PROTEIN-TYROSINE KINASE
Authors: TRAXLER P TRINKS U BUCHDUNGER E METT H MEYER T MULLER M REGENASS U ROSEL J LYDON N
Citation: P. Traxler et al., [(ALKYLAMINO)METHYL]ACRYLOPHENONES - POTENT AND SELECTIVE INHIBITORS OF THE EPIDERMAL GROWTH-FACTOR RECEPTOR PROTEIN-TYROSINE KINASE, Journal of medicinal chemistry, 38(13), 1995, pp. 2441-2448
Risultati: 1-25 | 26-36