Authors:
NAYLOROLSEN AM
PONTICELLO GS
LEWIS SD
MULICHAK AM
CHEN ZG
HABECKER CN
PHILLIPS BT
SANDERS WM
TUCKER TJ
SHAFER JA
VACCA JP
Citation: Am. Naylorolsen et al., IDENTIFICATION AND SAR FOR A SELECTIVE, NONPEPTIDYL THROMBIN INHIBITOR, Bioorganic & medicinal chemistry letters, 8(13), 1998, pp. 1697-1702
Authors:
TUCKER TJ
LUMMA WC
MULICHAK AM
CHEN ZG
NAYLOROLSEN AM
LEWIS SD
LUCAS R
FREIDINGER RM
KUO LC
Citation: Tj. Tucker et al., DESIGN OF HIGHLY POTENT NONCOVALENT THROMBIN INHIBITORS THAT UTILIZE A NOVEL LIPOPHILIC BINDING POCKET IN THE THROMBIN ACTIVE-SITE, Journal of medicinal chemistry, 40(6), 1997, pp. 830-832
Authors:
FENG DM
GARDELL SJ
LEWIS SD
BOCK MG
CHEN ZG
FREIDINGER RM
NAYLOROLSEN AM
RAMJIT HG
WOLTMANN R
BASKIN EP
LYNCH JJ
LUCAS R
SHAFER JA
DANCHECK KB
CHEN IW
MAO SS
KRUEGER JA
HARE TR
MULICHAK AM
VACCA JP
Citation: Dm. Feng et al., DISCOVERY OF A NOVEL, SELECTIVE, AND ORALLY BIOAVAILABLE CLASS OF THROMBIN INHIBITORS INCORPORATING AMINOPYRIDYL MOIETIES AT THE P1 POSITION, Journal of medicinal chemistry, 40(23), 1997, pp. 3726-3733
Authors:
THAISRIVONGS S
WATENPAUGH KD
HOWE WJ
TOMICH PK
DOLAK LA
CHONG KT
TOMICH CSC
TOMASSELLI AG
TURNER SR
STROHBACH JW
MULICHAK AM
JANAKIRAMAN MN
MOON JB
LYNN JC
HORNG MM
HINSHAW RR
CURRY KA
ROTHROCK DJ
Citation: S. Thaisrivongs et al., STRUCTURE-BASED DESIGN OF NOVEL HIV PROTEASE INHIBITORS - CARBOXAMIDE-CONTAINING 4-HYDROXYCOUMARINS AND 4-HYDROXY-2-PYRONES AS POTENT NONPEPTIDIC INHIBITORS, Journal of medicinal chemistry, 38(18), 1995, pp. 3624-3637
Authors:
ROMINES KR
WATENPAUGH KD
TOMICH PK
HOWE WJ
MORRIS JK
LOVASZ KD
MULICHAK AM
FINZEL BC
LYNN JC
HORNG MM
SCHWENDE FJ
RUWART MJ
ZIPP GL
CHONG KT
DOLAK LA
TOTH LN
HOWARD GM
RUSH BD
WILKINSON KF
POSSERT PL
DALGA RJ
HINSHAW RR
Citation: Kr. Romines et al., USE OF MEDIUM-SIZED CYCLOALKYL RINGS TO ENHANCE SECONDARY BINDING - DISCOVERY OF A NEW CLASS OF HUMAN-IMMUNODEFICIENCY-VIRUS (HIV) PROTEASEINHIBITORS, Journal of medicinal chemistry, 38(11), 1995, pp. 1884-1891
Authors:
CHEN ZG
LI Y
MULICHAK AM
LEWIS SD
SHAFER JA
Citation: Zg. Chen et al., CRYSTAL-STRUCTURE OF HUMAN ALPHA-THROMBIN COMPLEXED WITH HIRUGEN AND P-AMIDINOPHENYLPYRUVATE AT 1.6 ANGSTROM RESOLUTION, Archives of biochemistry and biophysics, 322(1), 1995, pp. 198-203
Authors:
THAISRIVONGS S
TOMICH PK
WATENPAUGH KD
CHONG KT
HOWE WJ
YANG CP
STROHBACH JW
TURNER SR
MCGRATH JP
BOHANON MJ
LYNN JC
MULICHAK AM
SPINELLI PA
HINSHAW RR
PAGANO PJ
MOON JB
RUWART MJ
WILKINSON KF
RUSH BD
ZIPP GL
DALGA RJ
SCHWENDE FJ
HOWARD GM
PADBURY GE
TOTH LN
ZHAO ZY
KOEPLINGER KA
KAKUK TJ
COLE SL
ZAYA RM
PIPER RC
JEFFREY P
Citation: S. Thaisrivongs et al., STRUCTURE-BASED DESIGN OF HIV PROTEASE INHIBITORS - 4-HYDROXYCOUMARINS AND 4-HYDROXY-2-PYRONES AS NONPEPTIDIC INHIBITORS, Journal of medicinal chemistry, 37(20), 1994, pp. 3200-3204
Authors:
MULICHAK AM
HUI JO
TOMASSELLI AG
HEINRIKSON RL
CURRY KA
TOMICH CS
THAISRIVONGS S
SAWYER TK
WATENPAUGH KD
Citation: Am. Mulichak et al., THE CRYSTALLOGRAPHIC STRUCTURE OF THE PROTEASE FROM HUMAN-IMMUNODEFICIENCY-VIRUS TYPE-2 WITH 2 SYNTHETIC PEPTIDIC TRANSITION-STATE ANALOG INHIBITORS, The Journal of biological chemistry, 268(18), 1993, pp. 3103-3109