Authors:
Zhang, HC
McComsey, DF
White, KB
Addo, MF
Andrade-Gordon, P
Derian, CK
Oksenberg, D
Maryanoff, BE
Citation: Hc. Zhang et al., Thrombin receptor (PAR-1) antagonists. Solid-phase synthesis of indole-based peptide mimetics by anchoring to a secondary amide, BIOORG MED, 11(16), 2001, pp. 2105-2109
Authors:
Andrade-Gordon, P
Derian, CK
Maryanoff, BE
Zhang, HC
Addo, MF
Cheung, WM
Damiano, BP
D'Andrea, MR
Darrow, AL
De Garavilla, L
Eckardt, AJ
Giardino, EC
Haertlein, BJ
McComsey, DF
Citation: P. Andrade-gordon et al., Administration of a potent antagonist of protease-activated receptor-1 (PAR-1) attenuates vascular restenosis following balloon angioplasty in rats, J PHARM EXP, 298(1), 2001, pp. 34-42
Authors:
Zhang, HC
Derian, CK
Andrade-Gordon, P
Hoekstra, WJ
McComsey, DF
White, KB
Poulter, BL
Addo, MF
Cheung, WM
Damiano, BP
Oksenberg, D
Reynolds, EE
Pandey, A
Scarborough, RM
Maryanoff, BE
Citation: Hc. Zhang et al., Discovery and optimization of a novel series of thrombin receptor (PAR-1) antagonists: Potent, selective peptide mimetics based on indole and indazole templates, J MED CHEM, 44(7), 2001, pp. 1021-1024
Authors:
Maryanoff, BE
Santulli, RJ
McComsey, DF
Hoekstra, WJ
Hoey, K
Smith, CE
Addo, M
Darrow, AL
Andrade-Gordon, P
Citation: Be. Maryanoff et al., Protease-activated receptor-2 (PAR-2): Structure-function study of receptor activation by diverse peptides related to tethered-ligand epitopes, ARCH BIOCH, 386(2), 2001, pp. 195-204
Citation: Df. Mccomsey et Be. Maryanoff, 3-aza-Cope rearrangement of quaternary N-allyl enammonium salts. Stereospecific 1,3 allyl migration from nitrogen to carbon on a tricyclic template, J ORG CHEM, 65(16), 2000, pp. 4938-4943
Authors:
Ceruso, MA
McComsey, DF
Leo, GC
Andrade-Gordon, P
Addo, MF
Scarborough, RM
Oksenberg, D
Maryanoff, BE
Citation: Ma. Ceruso et al., Thrombin receptor-activating peptides (TRAPs): Investigation of bioactive conformations via structure-activity, spectroscopic, and computational studies, BIO MED CH, 7(11), 1999, pp. 2353-2371
Authors:
Andrade-Gordon, P
Mayanoff, BE
Derian, CK
Zhang, HC
Addo, MF
Darrow, AL
Eckardt, AJ
Hoekstra, WJ
McComsey, DF
Oksenberg, D
Reynolds, EE
Santulli, RJ
Scarborough, RM
Smith, CE
White, KB
Citation: P. Andrade-gordon et al., Design, synthesis, and biological characterization of a peptide-mimetic antagonist for a tethered-ligand receptor, P NAS US, 96(22), 1999, pp. 12257-12262
Authors:
Hoekstra, WJ
Maryanoff, BE
Damiano, BP
Andrade-Gordon, P
Cohen, JH
Costanzo, MJ
Haertlein, BJ
Hecker, LR
Hulshizer, BL
Kauffman, JA
Keane, P
McComsey, DF
Mitchell, JA
Scott, L
Shah, RD
Yabut, SC
Citation: Wj. Hoekstra et al., Potent, orally active GPIIb/IIIa antagonists containing a nipecotic acid subunit. Structure-activity studies leading to the discovery of RWJ-53308, J MED CHEM, 42(25), 1999, pp. 5254-5265